Literature DB >> 24081753

The MABA approach: a new option to improve bronchodilator therapy.

Mario Cazzola1, Jose-Luis Lopez-Campos, Luis Puente-Maestu.   

Abstract

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Year:  2013        PMID: 24081753     DOI: 10.1183/09031936.00067013

Source DB:  PubMed          Journal:  Eur Respir J        ISSN: 0903-1936            Impact factor:   16.671


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  9 in total

Review 1.  Umeclidinium/vilanterol: a review of its use as maintenance therapy in adults with chronic obstructive pulmonary disease.

Authors:  Hannah A Blair; Emma D Deeks
Journal:  Drugs       Date:  2015-01       Impact factor: 9.546

2.  Navafenterol (AZD8871) in patients with mild asthma: a randomised placebo-controlled phase I study evaluating the safety, tolerability, pharmacokinetics, and pharmacodynamics of single ascending doses of this novel inhaled long-acting dual-pharmacology bronchodilator.

Authors:  Eulalia Jimenez; Carol Astbury; Muna Albayaty; Ulrika Wählby-Hamrén; Beatriz Seoane; Cristina Villarroel; Helena Pujol; Maria Jesus Bermejo; Ajay Aggarwal; Ioannis Psallidas
Journal:  Respir Res       Date:  2020-09-09

3.  Pharmacokinetics, Excretion, and Mass Balance of [14 C]-Batefenterol Following a Single Microtracer Intravenous Dose (Concomitant to an Inhaled Dose) or Oral Dose of Batefenterol in Healthy Men.

Authors:  Claire Ambery; Graeme Young; Teresa Fuller; Aili L Lazaar; Adrian Pereira; Adam Hughes; David Ramsay; Frans van den Berg; Peter Daley-Yates
Journal:  Clin Pharmacol Drug Dev       Date:  2018-09-19

4.  Randomized dose-finding study of batefenterol via dry powder inhaler in patients with COPD.

Authors:  Courtney Crim; Michael L Watkins; Eric D Bateman; Gregory J Feldman; Isabelle Schenkenberger; Edward M Kerwin; Catriona Crawford; Krishna Pudi; Shuyen Ho; Charlotte Baidoo; Ramiro Castro-Santamaria
Journal:  Int J Chron Obstruct Pulmon Dis       Date:  2019-03-08

5.  A randomized, controlled, repeat-dose study of batefenterol/fluticasone furoate compared with placebo in the treatment of COPD.

Authors:  Courtney Crim; Mark Gotfried; Selwyn Spangenthal; Michael Watkins; Amanda Emmett; Catriona Crawford; Charlotte Baidoo; Ramiro Castro-Santamaria
Journal:  BMC Pulm Med       Date:  2020-05-04       Impact factor: 3.317

Review 6.  Long-Acting Muscarinic Antagonists Under Investigational to Treat Chronic Obstructive Pulmonary Disease.

Authors:  Josuel Ora; Angelo Coppola; Mario Cazzola; Luigino Calzetta; Paola Rogliani
Journal:  J Exp Pharmacol       Date:  2020-12-08

Review 7.  The future of inhalation therapy in chronic obstructive pulmonary disease.

Authors:  Mario Cazzola; Josuel Ora; Luigino Calzetta; Paola Rogliani; Maria Gabriella Matera
Journal:  Curr Res Pharmacol Drug Discov       Date:  2022-02-17

8.  Population Pharmacokinetics and Pharmacodynamics of GSK961081 (Batefenterol), a Muscarinic Antagonist and β2-Agonist, in Moderate-to-Severe COPD Patients: Substudy of a Randomized Trial.

Authors:  Claire L Ambery; Pascal Wielders; Andrea Ludwig-Sengpiel; Robert Chan; John H Riley
Journal:  Drugs R D       Date:  2015-09

9.  In vitro anti-inflammatory effects of AZD8999, a novel bifunctional muscarinic acetylcholine receptor antagonist /β2-adrenoceptor agonist (MABA) compound in neutrophils from COPD patients.

Authors:  Javier Milara; Sonia Contreras; Alfredo de Diego; Marta Calbet; Mònica Aparici; Esteban Morcillo; Montserrat Miralpeix; Julio Cortijo
Journal:  PLoS One       Date:  2019-01-04       Impact factor: 3.240

  9 in total

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