Literature DB >> 24064757

Safety of Abiraterone Acetate in Castration-resistant Prostate Cancer Patients With Concomitant Cardiovascular Risk Factors.

Giuseppe Procopio1, Paolo Grassi, Isabella Testa, Elena Verzoni, Valter Torri, Roberto Salvioni, Riccardo Valdagni, Filippo de Braud.   

Abstract

OBJECTIVES: The aim of this study was to evaluate the safety profile of abiraterone acetate (AA) in metastatic castration-resistant prostate cancer (mCRPC) men with cardiovascular comorbidity, as little conclusive safety data are available in this patient subset. PATIENTS AND METHODS: A retrospective analysis of mCRPC patients with controlled cardiovascular comorbidities, receiving AA 1000 mg administered orally once daily and prednisone 5 mg twice daily, between April 2011 and July 2012, was performed. All clinical and instrumental variables and toxicity data were analyzed by descriptive statistics: mean, standard deviation, minimum and maximum values for continuous variables, and absolute and relative frequencies for categorical variables.
RESULTS: A total of 51 mCRPC patients were evaluated. Metastatic sites included the bone (74%), lungs, and liver (26%). All patients were previously treated with at least 2 lines of hormone and 1 docetaxel-based chemotherapy. Preexisting cardiac risk factors included hypertension (41%), cardiac ischemia (12%), arrhythmias (6%), dislipidemia (18%), and hyperglycemia (30%). No grade 3-4 adverse events were observed. Grade 1-2 adverse events included fluid retention (18%), asthenia (15%), and hypertension (16%). Median progression-free survival was 5.1 months (95% confidence interval, 0.5-12). Prostate specific antigen assessment revealed a good overall disease control rate (64%).
CONCLUSIONS: AA appears to be safe and well tolerated even in patients with cardiovascular comorbidities or with increased risk factors for cardiovascular diseases.

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Year:  2015        PMID: 24064757     DOI: 10.1097/COC.0b013e3182a790ce

Source DB:  PubMed          Journal:  Am J Clin Oncol        ISSN: 0277-3732            Impact factor:   2.339


  11 in total

1.  Safety of long-term exposure to abiraterone acetate in patients with castration-resistant prostate cancer and concomitant cardiovascular risk factors.

Authors:  Elena Verzoni; Paolo Grassi; Raffaele Ratta; Monica Niger; Filippo De Braud; Riccardo Valdagni; Giuseppe Procopio
Journal:  Ther Adv Med Oncol       Date:  2016-07-05       Impact factor: 8.168

Review 2.  Hormonal prostate cancer therapies and cardiovascular disease: a systematic review.

Authors:  Vittore Cereda; Pina T Falbo; Gaia Manna; Alessandro Iannace; Antonello Menghi; Michela Corona; Diana Semenova; Leonardo Calò; Roberto Carnevale; Giacomo Frati; Gaetano Lanzetta
Journal:  Heart Fail Rev       Date:  2022-01       Impact factor: 4.214

Review 3.  Abiraterone in the treatment of metastatic castration-resistant prostate cancer.

Authors:  Elahe A Mostaghel
Journal:  Cancer Manag Res       Date:  2014-01-28       Impact factor: 3.989

Review 4.  Androgen synthesis inhibitors in the treatment of castration-resistant prostate cancer.

Authors:  Mark N Stein; Neal Patel; Alexander Bershadskiy; Alisa Sokoloff; Eric A Singer
Journal:  Asian J Androl       Date:  2014 May-Jun       Impact factor: 3.285

5.  Feasibility of abiraterone acetate treatment in patients with metastatic castration-resistant prostate cancer and atrial fibrillation.

Authors:  Simon Rauch; Dominic Fong; Elisa Morra; Francesca Maines; Orazio Caffo; Gilbert Spizzo
Journal:  Prostate Int       Date:  2016-02-21

Review 6.  Association of Biomarkers with Serious Cardiac Adverse Events during Abiraterone Acetate Treatment in Castration Resistant Prostate Cancer.

Authors:  Sara Campora; Eleonora Campazzi; Silvia Zanardi; Matteo Puntoni; Marco Piccininno; Arnoldo Piccardo; Mehrdad Shoushtari Zadeh Naseri; Carlotta Defferrari; Nicoletta Provinciali; Marilena Petrera; Domenico Marra; Ennio Biscaldi; Gian Carlo Antonucci; Damiano Ricci; Matteo Clavarezza; Alessandra Gennari; Alberto Gozza; Mauro D'Amico; Marco Mori; Andrea DeCensi
Journal:  Transl Oncol       Date:  2016-12       Impact factor: 4.243

Review 7.  Impact of abiraterone on patient-related outcomes in metastatic castration-resistant prostate cancer: current perspectives.

Authors:  Joelle El-Amm; Rami Nassabein; Jeanny B Aragon-Ching
Journal:  Cancer Manag Res       Date:  2017-07-11       Impact factor: 3.989

8.  Abiraterone acetate and prednisone in the pre- and post-docetaxel setting for metastatic castration-resistant prostate cancer: a mono-institutional experience focused on cardiovascular events and their impact on clinical outcomes.

Authors:  Alessia Cavo; Alessandra Rubagotti; Elisa Zanardi; Chiara Fabbroni; Linda Zinoli; Antonio Di Meglio; Eleonora Arboscello; Andrea Bellodi; Paolo Spallarossa; Carlo Cattrini; Carlo Messina; Francesco Boccardo
Journal:  Ther Adv Med Oncol       Date:  2018-01-09       Impact factor: 8.168

Review 9.  Differential side effects profile in patients with mCRPC treated with abiraterone or enzalutamide: a meta-analysis of randomized controlled trials.

Authors:  Raphael B Moreira; Marcio Debiasi; Edoardo Francini; Pier V Nuzzo; Guillermo De Velasco; Fernando C Maluf; Andre P Fay; Joaquim Bellmunt; Toni K Choueiri; Fabio A Schutz
Journal:  Oncotarget       Date:  2017-08-08

10.  Effectiveness of abiraterone acetate plus prednisone in chemotherapy-naïve patients with metastatic castration-resistant prostate cancer in a large prospective real-world cohort: the ABItude study.

Authors:  Giuseppe Procopio; Vincenzo Emanuele Chiuri; Monica Giordano; Giovanna Mantini; Roberto Maisano; Roberto Bordonaro; Nicola Calvani; Gaetano Facchini; Sabino De Placido; Mario Airoldi; Andrea Sbrana; Donatello Gasparro; Giuseppe Mario Ludovico; Pamela Guglielmini; Emanuele Naglieri; Daniele Fagnani; Massimo Aglietta; Luigi Schips; Patrizia Beccaglia; Alessandro Sciarra; Lorenzo Livi; Daniele Santini
Journal:  Ther Adv Med Oncol       Date:  2020-10-29       Impact factor: 8.168

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