Literature DB >> 24050965

Evidence for cardiac safety and antiarrhythmic potential of chloroquine in systemic lupus erythematosus.

Ricardo Alkmim Teixeira1, Eduardo F Borba2, Anísio Pedrosa3, Silvana Nishioka3, Vilma S T Viana2, José A Ramires3, Roberto Kalil-Filho3, Eloísa Bonfá2, Martino Martinelli Filho3.   

Abstract

AIMS: To perform a comprehensive evaluation of heart rhythm disorders and the influence of disease/therapy factors in a large systemic lupus erythematosus (SLE) cohort. METHODS AND
RESULTS: Three hundred and seventeen consecutive patients of an ongoing electronic database protocol were evaluated by resting electrocardiogram and 142 were randomly selected for 24 h Holter monitoring for arrhythmia and conduction disturbances. The mean age was 40.2 ± 12.1 years and disease duration was 11.4 ± 8.1 years. Chloroquine (CQ) therapy was identified in 69.7% with a mean use of 8.5 ± 6.7 years. Electrocardiogram abnormalities were detected in 66 patients (20.8%): prolonged QTc/QTd (14.2%); bundle-branch block (2.5%); and atrioventricular block (AVB) (1.6%). Age was associated with AVB (P = 0.029) and prolonged QTc/QTd (P = 0.039) whereas anti-Ro/SS-A and Systemic Lupus Erythematosus Disease Activity Index (SLEDAI) scores were not (P > 0.05). Chloroquine was negatively associated with AVB (P = 0.01) as was its longer use (6.1 ± 6.9 vs. 1.0 ± 2.5 years, P = 0.018). Time of CQ use was related with the absence of AVB [odds ratio (OR) = 0.103; 95% confidence interval (CI) = 0.011-0.934, P = 0.043] in multiple logistic regression. Holter monitoring revealed abnormalities in 121 patients (85.2%): supraventricular ectopies (63.4%) and tachyarrhythmia (18.3%); ventricular ectopies (45.8%). Atrial tachycardia/fibrillation (AT/AF) were associated with shorter CQ duration (7.05 ± 7.99 vs. 3.63 ± 5.02 years, P = 0.043) with a trend to less CQ use (P = 0.054), and older age (P < 0.001). Predictors of AT/AF in multiple logistic regression were age (OR = 1.115; 95% CI = 1.059-1.174, P < 0.001) and anti-Ro/SS-A (OR = 0.172; 95% CI = 0.047-0.629, P = 0.008).
CONCLUSIONS: Chloroquine seems to play a protective role in the unexpected high rate of cardiac arrhythmias and conduction disturbances observed in SLE. Further studies are necessary to determine if this antiarrhythmic effect is due to the disease control or a direct effect of the drug. Published on behalf of the European Society of Cardiology. All rights reserved.
© The Author 2013. For permissions please email: journals.permissions@oup.com.

Entities:  

Keywords:  Antimalarial; Arrhythmia; Safety; Systemic lupus erythematosus; Treatment

Mesh:

Substances:

Year:  2013        PMID: 24050965     DOI: 10.1093/europace/eut290

Source DB:  PubMed          Journal:  Europace        ISSN: 1099-5129            Impact factor:   5.214


  12 in total

1.  Concentration-dependent mortality of chloroquine in overdose.

Authors:  James A Watson; Joel Tarning; Richard M Hoglund; Frederic J Baud; Bruno Megarbane; Jean-Luc Clemessy; Nicholas J White
Journal:  Elife       Date:  2020-07-08       Impact factor: 8.140

2.  Comparison of non-invasive assessment of arrhythmias, conduction disturbances and cardiac autonomic tone in systemic sclerosis and systemic lupus erythematosus.

Authors:  Piotr Bienias; Michał Ciurzyński; Bartłomiej Kisiel; Anna Chrzanowska; Katarzyna Ciesielska; Maria Siwicka; Agnieszka Kalińska-Bienias; Marek Saracyn; Monika Lisicka; Joanna Radochońska; Piotr Pruszczyk
Journal:  Rheumatol Int       Date:  2018-11-12       Impact factor: 2.631

3.  Prolonged Tpeak-Tend interval in anti-Ro52 antibody-positive connective tissue diseases.

Authors:  Ayse Nur Tufan; Saim Sag; Mustafa Ferhat Oksuz; Selime Ermurat; Belkis Nihan Coskun; Mustafa Gullulu; Ferah Budak; Ibrahim Baran; Yavuz Pehlivan; Ediz Dalkilic
Journal:  Rheumatol Int       Date:  2016-05-18       Impact factor: 2.631

Review 4.  Revisiting cardiac safety of hydroxychloroquine in rheumatological diseases during COVID-19 era: Facts and myths.

Authors:  Shivraj Padiyar; Debashish Danda
Journal:  Eur J Rheumatol       Date:  2020-10-08

5.  Assessment of inhomogeneities of repolarization in patients with systemic lupus erythematosus.

Authors:  Ahmet Avci; Kenan Demir; Bulent Behlul Altunkeser; Sema Yilmaz; Ahmet Yilmaz; Ahmet Ersecgin; Tarik Demir
Journal:  Ann Noninvasive Electrocardiol       Date:  2014-03-05       Impact factor: 1.468

Review 6.  Cardiac effects and toxicity of chloroquine: a short update.

Authors:  Kanigula Mubagwa
Journal:  Int J Antimicrob Agents       Date:  2020-06-19       Impact factor: 5.283

7.  Heart Involvement in Inflammatory Rheumatic Diseases: A Systematic Literature Review.

Authors:  Florina Buleu; Elena Sirbu; Alexandru Caraba; Simona Dragan
Journal:  Medicina (Kaunas)       Date:  2019-06-06       Impact factor: 2.430

8.  Chloroquine is grossly under dosed in young children with malaria: implications for drug resistance.

Authors:  Johan Ursing; Staffan Eksborg; Lars Rombo; Yngve Bergqvist; Daniel Blessborn; Amabelia Rodrigues; Poul-Erik Kofoed
Journal:  PLoS One       Date:  2014-01-23       Impact factor: 3.240

Review 9.  Long QT Syndrome: An Emerging Role for Inflammation and Immunity.

Authors:  Pietro Enea Lazzerini; Pier Leopoldo Capecchi; Franco Laghi-Pasini
Journal:  Front Cardiovasc Med       Date:  2015-05-27

10.  The Antimalarial Chloroquine Reduces the Burden of Persistent Atrial Fibrillation.

Authors:  Catalina Tobón; Laura C Palacio; Bojjibabu Chidipi; Diana P Slough; Thanh Tran; Nhi Tran; Michelle Reiser; Yu-Shan Lin; Bengt Herweg; Dany Sayad; Javier Saiz; Sami Noujaim
Journal:  Front Pharmacol       Date:  2019-11-27       Impact factor: 5.810

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