Warning: Undefined array key "mm" in /www/wwwroot/www.ai-bt.com/si.php on line 10 Deprecated: trim(): Passing null to parameter #1 ($string) of type string is deprecated in /www/wwwroot/www.ai-bt.com/si.php on line 10 N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases.

Literature DB >> 23975403

N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases.

N P Boltneva¹, O G Serebryakova, G F Makhaeva, I V Serkov, A N Proshin, S O Bachurin.

Abstract

Entities: Chemical

Mesh：

Substances：

Year: 2013 PMID： 23975403 DOI： 10.1134/S160767291304011X

Source DB: PubMed Journal: Dokl Biochem Biophys ISSN： 1607-6729 Impact factor: 0.788

Keyword Cloud
References

× No keyword cloud information.

12 in total

Review 1. Carboxylesterases--detoxifying enzymes and targets for drug therapy.

Authors: Philip M Potter; Randy M Wadkins
Journal: Curr Med Chem Date: 2006 Impact factor: 4.530

2. Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors.

Authors: Aldo Andreani; Silvia Burnelli; Massimiliano Granaiola; Massimo Guardigli; Alberto Leoni; Alessandra Locatelli; Rita Morigi; Mirella Rambaldi; Manuela Rizzoli; Lucilla Varoli; Aldo Roda
Journal: Eur J Med Chem Date: 2007-05-21 Impact factor: 6.514

3. Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols.

Authors: G F Makhaeva; O G Serebryakova; N P Boltneva; T G Galenko; A Yu Aksinenko; V B Sokolov; I V Martynov
Journal: Dokl Biochem Biophys Date: 2008 Nov-Dec Impact factor: 0.788

Review 4. Overview of the chemistry of 2-thiazolines.

Authors: Annie-Claude Gaumont; Mihaela Gulea; Jocelyne Levillain
Journal: Chem Rev Date: 2009-03-11 Impact factor: 60.622

5. Esterase profile of O-phosphorylated ethyltrifluorolactates in prediction of their therapeutic and toxic effects.

Authors: E V Rudakova; G F Makhaeva; T G Galenko; A Yu Aksinenko; V B Sokolov; R J Richardson; I V Martynov
Journal: Dokl Biochem Biophys Date: 2012-05-05 Impact factor: 0.788

6. A radiochemical assay method for carboxylesterase, and comparison of enzyme activity towards the substrates methyl [1-14C] butyrate and 4-nitrophenyl butyrate.

Authors: S H Sterri; B A Johnsen; F Fonnum
Journal: Biochem Pharmacol Date: 1985-08-01 Impact factor: 5.858

N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases.

Review 1. Carboxylesterases--detoxifying enzymes and targets for drug therapy.

2. Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors.

3. Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols.

Review 4. Overview of the chemistry of 2-thiazolines.

5. Esterase profile of O-phosphorylated ethyltrifluorolactates in prediction of their therapeutic and toxic effects.

6. A radiochemical assay method for carboxylesterase, and comparison of enzyme activity towards the substrates methyl [1-14C] butyrate and 4-nitrophenyl butyrate.

7. Competitive inhibition of acetylcholinesterase by several thiazolines and oxazolines.

8. Organophosphorus compound esterase profiles as predictors of therapeutic and toxic effects.

Review 9. Recent developments in cholinesterases inhibitors for Alzheimer's disease treatment.

Review 10. Cholinesterase inhibitors: new roles and therapeutic alternatives.