Literature DB >> 23937387

Efficacy and safety of oral tapentadol extended release in Japanese and Korean patients with moderate to severe, chronic malignant tumor-related pain.

Keiichiro Imanaka1, Yushin Tominaga, Mila Etropolski, Ilse van Hove, Masaki Ohsaka, Mikio Wanibe, Keiichiro Hirose, Taka Matsumura.   

Abstract

OBJECTIVE: This phase 3 study evaluated the efficacy and safety of tapentadol extended release (ER) compared with oxycodone controlled release (CR) for the management of moderate to severe, chronic malignant tumor-related cancer pain. RESEARCH DESIGN AND METHODS: This randomized, double-blind, active-controlled study included Japanese and Korean patients with moderate to severe, chronic malignant tumor-related pain. Patients were randomized (1:1) to receive oral tapentadol ER (25-200 mg bid) or oral oxycodone HCl CR (5-40 mg bid) for 4 weeks of double-blind treatment. ClinicalTrials.gov identifier: NCT01165281. MAIN OUTCOME MEASURES: This study was designed to evaluate the non-inferiority of the efficacy provided by tapentadol ER versus oxycodone CR, based on the mean change in average pain intensity (11 point numerical rating scale) from baseline to the last 3 days of study drug administration. Treatment-emergent adverse events (TEAEs) were recorded throughout the study.
RESULTS: Of the 374 patients who were screened, 343 were randomized and 236 completed treatment. The least-squares mean difference in the change in pain intensity from baseline to the last 3 days of study treatment between tapentadol ER and oxycodone CR was -0.06 (95% confidence interval [CI], -0.506 to 0.383). The upper limit of the 95% CI was <1 (the predefined threshold value for non-inferiority), indicating that tapentadol ER provided analgesic efficacy that was non-inferior to that of oxycodone CR. The percentage of patients reporting at least one TEAE was similar in the tapentadol ER (87.5% [147/168]) and oxycodone CR (90.1% [155/172]) treatment groups, but the incidence of gastrointestinal TEAEs was lower in the tapentadol ER group (55.4% [93/168]) than in the oxycodone CR group (67.4% [116/172]).
CONCLUSIONS: Tapentadol ER (25-200 mg bid) provides analgesic efficacy that is non-inferior to that provided by oxycodone HCl CR (5-40 mg bid) for the management of moderate to severe, chronic malignant tumor-related pain, and is well tolerated overall, with a better gastrointestinal tolerability profile than oxycodone CR.

Entities:  

Mesh:

Substances:

Year:  2013        PMID: 23937387     DOI: 10.1185/03007995.2013.831816

Source DB:  PubMed          Journal:  Curr Med Res Opin        ISSN: 0300-7995            Impact factor:   2.580


  27 in total

1.  Cancer pain physiology.

Authors:  Sarah Falk; Kirsty Bannister; Anthony H Dickenson
Journal:  Br J Pain       Date:  2014-11

2.  Efficacy and Safety of Fentanyl Citrate Patch, Including a Low-Dose 0.5 mg Formulation, in Opioid-Naïve Patients with Cancer Pain.

Authors:  Shigeki Yamaguchi; Eiji Uchida; Takaaki Terahara; Koji Okawa; Fumitaka Hashimoto; Yusuke Tanaka
Journal:  Clin Drug Investig       Date:  2020-11       Impact factor: 2.859

3.  Quantifying the Exposure of Tapentadol Extended Release in Japanese Patients with Cancer Pain and Bridging Tapentadol Pharmacokinetics Across Populations Using a Modeling Approach.

Authors:  Liping Zhang; Xiaoyu Yan; Sayori Nobe; Peter Zannikos; Mila Etropolski; Partha Nandy
Journal:  Clin Drug Investig       Date:  2017-03       Impact factor: 2.859

4.  NCCN Guidelines Insights: Survivorship, Version 2.2019.

Authors:  Tara Sanft; Crystal S Denlinger; Saro Armenian; K Scott Baker; Gregory Broderick; Wendy Demark-Wahnefried; Debra L Friedman; Mindy Goldman; Melissa Hudson; Nazanin Khakpour; Divya Koura; Robin M Lally; Terry S Langbaum; Allison L McDonough; Michelle Melisko; Kathi Mooney; Halle C F Moore; Javid J Moslehi; Tracey O'Connor; Linda Overholser; Electra D Paskett; Lindsay Peterson; William Pirl; M Alma Rodriguez; Kathryn J Ruddy; Sophia Smith; Karen L Syrjala; Amye Tevaarwerk; Susan G Urba; Phyllis Zee; Nicole R McMillian; Deborah A Freedman-Cass
Journal:  J Natl Compr Canc Netw       Date:  2019-07-01       Impact factor: 11.908

5.  To what extent are we confident that tapentadol induces less constipation and other side effects than the other opioids in chronic pain patients? a confidence evaluation in network meta-analysis.

Authors:  Patrice Forget; Mathieu Vermeersch
Journal:  Br J Pain       Date:  2020-08-03

Review 6.  Oxycodone for cancer-related pain.

Authors:  Mia Schmidt-Hansen; Michael I Bennett; Stephanie Arnold; Nathan Bromham; Jennifer S Hilgart; Andrew J Page; Yuan Chi
Journal:  Cochrane Database Syst Rev       Date:  2022-06-09

Review 7.  Multimechanistic Single-Entity Combinations for Chronic Pain Control: A Narrative Review.

Authors:  Joseph Pergolizzi; Peter Magnusson; Flaminia Coluzzi; Frank Breve; Jo Ann K LeQuang; Giustino Varrassi
Journal:  Cureus       Date:  2022-06-16

Review 8.  Oral tapentadol for cancer pain.

Authors:  Philip J Wiffen; Sheena Derry; Katrien Naessens; Rae F Bell
Journal:  Cochrane Database Syst Rev       Date:  2015-09-25

Review 9.  Oxycodone for cancer-related pain.

Authors:  Mia Schmidt-Hansen; Michael I Bennett; Stephanie Arnold; Nathan Bromham; Jennifer S Hilgart
Journal:  Cochrane Database Syst Rev       Date:  2017-08-22

10.  A pooled analysis evaluating the efficacy and tolerability of tapentadol extended release for chronic, painful diabetic peripheral neuropathy.

Authors:  Sherwyn Schwartz; Mila S Etropolski; Douglas Y Shapiro; Christine Rauschkolb; Aaron I Vinik; Bernd Lange; Kimberly Cooper; Ilse Van Hove; Juergen Haeussler
Journal:  Clin Drug Investig       Date:  2015-02       Impact factor: 2.859

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.