Literature DB >> 23826939

Suzuki-Miyaura cross-coupling of potassium trifluoro(N-methylheteroaryl)borates with aryl and heteroaryl halides.

Gary A Molander1, DaWeon Ryu, Mona Hosseini-Sarvari, Rammohan Devulapally, Dave G Seapy.   

Abstract

The synthesis of potassium trifluoro(N-methylheteroaryl)borates and their use in cross-coupling reactions with various aryl and heteroaryl halides to construct N-methyl heteroaryl-substituted aromatic and heteroaromatic compounds are reported.

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Year:  2013        PMID： 23826939      PMCID： PMC3752378          DOI： 10.1021/jo4009589

Source DB:  PubMed          Journal:  J Org Chem        ISSN： 0022-3263            Impact factor:   4.354


  16 in total

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6.  Scope of aminomethylations via Suzuki-Miyaura cross-coupling of organotrifluoroborates.

Authors:  Gary A Molander; Paul E Gormisky; Deidre L Sandrock
Journal:  J Org Chem       Date:  2008-02-20       Impact factor: 4.354

7.  Suzuki-Miyaura cross-coupling reactions of primary alkyltrifluoroborates with aryl chlorides.

Authors:  Spencer D Dreher; Siang-Ee Lim; Deidre L Sandrock; Gary A Molander
Journal:  J Org Chem       Date:  2009-05-15       Impact factor: 4.354

8.  Efficient cross-coupling of secondary alkyltrifluoroborates with aryl chlorides--reaction discovery using parallel microscale experimentation.

Authors:  Spencer D Dreher; Peter G Dormer; Deidre L Sandrock; Gary A Molander
Journal:  J Am Chem Soc       Date:  2008-06-27       Impact factor: 15.419

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Authors:  Shyama Sidique; Sergey A Shiryaev; Boris I Ratnikov; Ananda Herath; Ying Su; Alex Y Strongin; Nicholas D P Cosford
Journal:  Bioorg Med Chem Lett       Date:  2009-08-03       Impact factor: 2.823

10.  Aminomethylations via cross-coupling of potassium organotrifluoroborates with aryl bromides.

Authors:  Gary A Molander; Deidre L Sandrock
Journal:  Org Lett       Date:  2007-03-17       Impact factor: 6.005
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