Literature DB >> 23818141

α-Boryl isocyanides enable facile preparation of bioactive boropeptides.

Adam Zajdlik1, Zezhou Wang, Jennifer L Hickey, Ahmed Aman, Aaron D Schimmer, Andrei K Yudin.   

Abstract

Entities:  

Keywords:  boron; inhibitors; isocyanides; multicomponent reactions; peptides

Mesh：

Substances：

Year:  2013        PMID： 23818141     DOI： 10.1002/anie.201302818

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  16 in total

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2.  Facile construction of fused benzimidazole-isoquinolinones that induce cell-cycle arrest and apoptosis in colorectal cancer cells.

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3.  Facile synthesis of borofragments and their evaluation in activity-based protein profiling.

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Review 4.  The versatility of boron in biological target engagement.

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5.  From synthesis to function via iterative assembly of N-methyliminodiacetic acid boronate building blocks.

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6.  Toward Generalization of Iterative Small Molecule Synthesis.

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7.  A universal isocyanide for diverse heterocycle syntheses.

Authors:  Pravin Patil; Kareem Khoury; Eberhardt Herdtweck; Alexander Dömling
Journal:  Org Lett       Date:  2014-10-29       Impact factor: 6.005

8.  Multicomponent mapping of boron chemotypes furnishes selective enzyme inhibitors.

Authors:  Joanne Tan; Armand B Cognetta Iii; Diego B Diaz; Kenneth M Lum; Shinya Adachi; Soumajit Kundu; Benjamin F Cravatt; Andrei K Yudin
Journal:  Nat Commun       Date:  2017-11-24       Impact factor: 14.919

9.  Diversity-oriented synthesis of peptide-boronic acids by a versatile building-block approach.

Authors:  Stefan P A Hinkes; Severin Kämmerer; Christian D P Klein
Journal:  Chem Sci       Date:  2020-08-21       Impact factor: 9.825

10.  Synthesis of cyclic chiral α-amino boronates by copper-catalyzed asymmetric dearomative borylation of indoles.

Authors:  Lili Chen; Jun-Jian Shen; Qian Gao; Senmiao Xu
Journal:  Chem Sci       Date:  2018-06-12       Impact factor: 9.825
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