Literature DB >> 23805009

Microwave-assisted Heck Synthesis of Substituted 2,4-Diaminopyrimidine-based Antibiotics.

Baskar Nammalwar1, Richard A Bunce, K Darrell Berlin, Christina R Bourne, Philip C Bourne, Esther W Barrow, William W Barrow.   

Abstract

Entities:  

Year:  2012        PMID： 23805009      PMCID： PMC3691060          DOI： 10.1080/00304948.2012.676823

Source DB:  PubMed          Journal:  Org Prep Proced Int        ISSN： 0030-4948            Impact factor:   1.628


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  7 in total

Review 1.  Increasing rates of reaction: microwave-assisted organic synthesis for combinatorial chemistry.

Authors:  Amy Lew; Peter O Krutzik; Matthew E Hart; A Richard Chamberlin
Journal:  J Comb Chem       Date:  2002 Mar-Apr

Review 2.  Controlled microwave heating in modern organic synthesis.

Authors:  C Oliver Kappe
Journal:  Angew Chem Int Ed Engl       Date:  2004-11-26       Impact factor: 15.336

Review 3.  Controlled microwave heating in modern organic synthesis: highlights from the 2004-2008 literature.

Authors:  C Oliver Kappe; Doris Dallinger
Journal:  Mol Divers       Date:  2009-04-21       Impact factor: 2.943

4.  Towards the understanding of resistance mechanisms in clinically isolated trimethoprim-resistant, methicillin-resistant Staphylococcus aureus dihydrofolate reductase.

Authors:  Kathleen M Frey; Michael N Lombardo; Dennis L Wright; Amy C Anderson
Journal:  J Struct Biol       Date:  2009-12-21       Impact factor: 2.867

5.  In vitro efficacy of new antifolates against trimethoprim-resistant Bacillus anthracis.

Authors:  Esther W Barrow; Jürg Dreier; Stefan Reinelt; Philip C Bourne; William W Barrow
Journal:  Antimicrob Agents Chemother       Date:  2007-09-17       Impact factor: 5.191

6.  Microwave-assisted organic synthesis and transformations using benign reaction media.

Authors:  Vivek Polshettiwar; Rajender S Varma
Journal:  Acc Chem Res       Date:  2008-04-18       Impact factor: 22.384

7.  Crystal structure of Bacillus anthracis dihydrofolate reductase with the dihydrophthalazine-based trimethoprim derivative RAB1 provides a structural explanation of potency and selectivity.

Authors:  Christina R Bourne; Richard A Bunce; Philip C Bourne; K Darrell Berlin; Esther W Barrow; William W Barrow
Journal:  Antimicrob Agents Chemother       Date:  2009-04-13       Impact factor: 5.191
  7 in total
  4 in total

1.  Modified 2,4-diaminopyrimidine-based dihydrofolate reductase inhibitors as potential drug scaffolds against Bacillus anthracis.

Authors:  Baskar Nammalwar; Christina R Bourne; Nancy Wakeham; Philip C Bourne; Esther W Barrow; N Prasad Muddala; Richard A Bunce; K Darrell Berlin; William W Barrow
Journal:  Bioorg Med Chem       Date:  2014-11-11       Impact factor: 3.641

2.  Evaluation of New Dihydrophthalazine-Appended 2,4-Diaminopyrimidines against Bacillus anthracis: Improved Syntheses Using a New Pincer Complex.

Authors:  Nagendra Prasad Muddala; Baskar Nammalwar; Subhashini Selvaraju; Christina R Bourne; Mary Henry; Richard A Bunce; K Darrell Berlin; Esther W Barrow; William W Barrow
Journal:  Molecules       Date:  2015-04-21       Impact factor: 4.411

3.  Dual and selective inhibitors of pteridine reductase 1 (PTR1) and dihydrofolate reductase-thymidylate synthase (DHFR-TS) from Leishmania chagasi.

Authors:  Bárbara Velame Ferreira Teixeira; André Lacerda Braga Teles; Suellen Gonçalves da Silva; Camila Carane Bitencourt Brito; Humberto Fonseca de Freitas; Acássia Benjamim Leal Pires; Thamires Quadros Froes; Marcelo Santos Castilho
Journal:  J Enzyme Inhib Med Chem       Date:  2019-12       Impact factor: 5.051

4.  Synthesis and biological evaluation of 2,4-diaminopyrimidine-based antifolate drugs against Bacillus anthracis.

Authors:  Baskar Nammalwar; N Prasad Muddala; Christina R Bourne; Mary Henry; Philip C Bourne; Richard A Bunce; Esther W Barrow; K Darrell Berlin; William W Barrow
Journal:  Molecules       Date:  2014-03-17       Impact factor: 4.411
  4 in total

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