Literature DB >> 23453884

Qualitative and quantitative measures of various compounded formulations of 17-alpha hydroxyprogesterone caproate.

Steve N Caritis1, Yang Zhao, Joseph Bettinger, Raman Venkataramanan.   

Abstract

OBJECTIVE: 17-alpha hydroxyprogesterone caproate (17-OHPC) is available both as an Food and Drug Administration (FDA)-approved medication and as a product prepared for individual patients by compounding pharmacies. Compounding pharmacies may omit the preservative that is used in the FDA-approved formulation or use an alternate preservative and may dispense 17-OHPC in containers that differ from the FDA-approved product. The objective of this study was to assess the stability and the microbiologic and pyrogen status of 17-OHPC formulations under various compounding and dispensing conditions. STUDY
DESIGN: 17-OHPC was prepared by a local compounding pharmacy. The formulations that were prepared included 1 identical to the FDA-approved product with benzyl alcohol as a preservative, 1 with benzalkonium chloride as a preservative, and 1 without a preservative. These various formulations were dispensed into either single-dose 1-mL plastic syringes or glass vials or 10-mL glass vials. The concentration of 17-OHPC and microbial and pyrogen status were evaluated at various time intervals over the ensuing 19 weeks.
RESULTS: The concentration of 17-OHPC did not change over the duration of study, regardless of the dispensing medium that was used or the absence or presence of any preservatives. The preparations remained microbe- and pyrogen-free during the study period, regardless of the dispensing medium that was used or the absence of presence of any preservatives.
CONCLUSION: Products that contained 17-OHPC tested in this study were quite stable over the 19-week period of study in different dispensing containers and in the absence or presence of a different preservative. The compounded products remained sterile and pyrogen-free during the period of observation.
Copyright © 2013 Mosby, Inc. All rights reserved.

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Year:  2013        PMID: 23453884      PMCID: PMC3672260          DOI: 10.1016/j.ajog.2013.02.028

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  9 in total

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5.  Pharmacology and placental transport of 17-hydroxyprogesterone caproate in singleton gestation.

Authors:  Steve N Caritis; Shringi Sharma; Raman Venkataramanan; Gary D Hankins; Menachem Miodovnik; Mary F Hebert; Jason G Umans; Thomas Benedetti; Donald Mattison; Anne Zajicek; Dawn Fischer; Aimee Jackson
Journal:  Am J Obstet Gynecol       Date:  2012-08-16       Impact factor: 8.661

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Journal:  Obstet Gynecol       Date:  2003-11       Impact factor: 7.661

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8.  Relationship between 17-hydroxyprogesterone caproate concentrations and gestational age at delivery in twin gestation.

Authors:  Steve N Caritis; Hyagriv N Simhan; Yuan Zhao; Dwight J Rouse; Alan M Peaceman; Anthony Sciscione; Catherine Y Spong; Michael W Varner; Fergal D Malone; Jay D Iams; Brian M Mercer; John M Thorp; Yoram Sorokin; Marshall Carpenter; Julie Lo; Susan M Ramin; Margaret Harper
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Journal:  N Engl J Med       Date:  2003-06-12       Impact factor: 91.245

  9 in total
  1 in total

1.  Quality assessment of compounded 17-hydroxyprogesterone caproate.

Authors:  Justine Chang; Yang Zhao; Wenchen Zhao; Raman Venkataramanan; Steve N Caritis
Journal:  Am J Obstet Gynecol       Date:  2013-11-04       Impact factor: 8.661

  1 in total

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