Literature DB >> 23425436

Design and synthesis of 2-acylbenzothiazoles via in situ cross-trapping strategy from benzothiazoles with aryl ketones.

Qinghe Gao1, Xia Wu, Fengcheng Jia, Meicai Liu, Yanping Zhu, Qun Cai, Anxin Wu.   

Abstract

An I2/KOH synergistically promoted direct ring-opening aroylation of benzothiazoles with aryl ketones has been discovered. Aryl ketones were seen to act as carbonyl sources to construct 2-acylbenzothiazoles. This reaction could provide an example for the convergent integration of self-labor domino sequences based on an in situ cross-trapping strategy.

Entities:  

Year:  2013        PMID: 23425436     DOI: 10.1021/jo302754c

Source DB:  PubMed          Journal:  J Org Chem        ISSN: 0022-3263            Impact factor:   4.354


  1 in total

1.  New synthesis of 2-aroylbenzothiazoles via metal-free domino transformations of anilines, acetophenones, and elemental sulfur.

Authors:  Tien V Huynh; Khang V Doan; Ngoc T K Luong; Duyen T P Nguyen; Son H Doan; Tung T Nguyen; Nam T S Phan
Journal:  RSC Adv       Date:  2020-05-14       Impact factor: 3.361

  1 in total

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