Literature DB >> 23228172

Abiraterone in metastatic prostate cancer without previous chemotherapy.

Charles J Ryan1, Matthew R Smith, Johann S de Bono, Arturo Molina, Christopher J Logothetis, Paul de Souza, Karim Fizazi, Paul Mainwaring, Josep M Piulats, Siobhan Ng, Joan Carles, Peter F A Mulders, Ethan Basch, Eric J Small, Fred Saad, Dirk Schrijvers, Hendrik Van Poppel, Som D Mukherjee, Henrik Suttmann, Winald R Gerritsen, Thomas W Flaig, Daniel J George, Evan Y Yu, Eleni Efstathiou, Allan Pantuck, Eric Winquist, Celestia S Higano, Mary-Ellen Taplin, Youn Park, Thian Kheoh, Thomas Griffin, Howard I Scher, Dana E Rathkopf.   

Abstract

BACKGROUND: Abiraterone acetate, an androgen biosynthesis inhibitor, improves overall survival in patients with metastatic castration-resistant prostate cancer after chemotherapy. We evaluated this agent in patients who had not received previous chemotherapy.
METHODS: In this double-blind study, we randomly assigned 1088 patients to receive abiraterone acetate (1000 mg) plus prednisone (5 mg twice daily) or placebo plus prednisone. The coprimary end points were radiographic progression-free survival and overall survival.
RESULTS: The study was unblinded after a planned interim analysis that was performed after 43% of the expected deaths had occurred. The median radiographic progression-free survival was 16.5 months with abiraterone-prednisone and 8.3 months with prednisone alone (hazard ratio for abiraterone-prednisone vs. prednisone alone, 0.53; 95% confidence interval [CI], 0.45 to 0.62; P<0.001). Over a median follow-up period of 22.2 months, overall survival was improved with abiraterone-prednisone (median not reached, vs. 27.2 months for prednisone alone; hazard ratio, 0.75; 95% CI, 0.61 to 0.93; P=0.01) but did not cross the efficacy boundary. Abiraterone-prednisone showed superiority over prednisone alone with respect to time to initiation of cytotoxic chemotherapy, opiate use for cancer-related pain, prostate-specific antigen progression, and decline in performance status. Grade 3 or 4 mineralocorticoid-related adverse events and abnormalities on liver-function testing were more common with abiraterone-prednisone.
CONCLUSIONS: Abiraterone improved radiographic progression-free survival, showed a trend toward improved overall survival, and significantly delayed clinical decline and initiation of chemotherapy in patients with metastatic castration-resistant prostate cancer. (Funded by Janssen Research and Development, formerly Cougar Biotechnology; ClinicalTrials.gov number, NCT00887198.).

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Year:  2012        PMID: 23228172      PMCID: PMC3683570          DOI: 10.1056/NEJMoa1209096

Source DB:  PubMed          Journal:  N Engl J Med        ISSN: 0028-4793            Impact factor:   91.245


  26 in total

Review 1.  Novel therapeutic strategies for castration resistant prostate cancer: inhibition of persistent androgen production and androgen receptor mediated signaling.

Authors:  Arturo Molina; Arie Belldegrun
Journal:  J Urol       Date:  2011-01-15       Impact factor: 7.450

2.  Effects of abiraterone acetate on androgen signaling in castrate-resistant prostate cancer in bone.

Authors:  Eleni Efstathiou; Mark Titus; Dimitra Tsavachidou; Vassiliki Tzelepi; Sijin Wen; Anh Hoang; Arturo Molina; Nicole Chieffo; Lisa A Smith; Maria Karlou; Patricia Troncoso; Christopher J Logothetis
Journal:  J Clin Oncol       Date:  2011-12-19       Impact factor: 44.544

3.  Prognostic model for predicting survival in men with hormone-refractory metastatic prostate cancer.

Authors:  Susan Halabi; Eric J Small; Philip W Kantoff; Michael W Kattan; Ellen B Kaplan; Nancy A Dawson; Ellis G Levine; Brent A Blumenstein; Nicholas J Vogelzang
Journal:  J Clin Oncol       Date:  2003-04-01       Impact factor: 44.544

Review 4.  Second-line hormonal therapy for advanced prostate cancer: a shifting paradigm.

Authors:  E J Small; N J Vogelzang
Journal:  J Clin Oncol       Date:  1997-01       Impact factor: 44.544

5.  Docetaxel and estramustine compared with mitoxantrone and prednisone for advanced refractory prostate cancer.

Authors:  Daniel P Petrylak; Catherine M Tangen; Maha H A Hussain; Primo N Lara; Jeffrey A Jones; Mary Ellen Taplin; Patrick A Burch; Donna Berry; Carol Moinpour; Manish Kohli; Mitchell C Benson; Eric J Small; Derek Raghavan; E David Crawford
Journal:  N Engl J Med       Date:  2004-10-07       Impact factor: 91.245

6.  Docetaxel plus prednisone or mitoxantrone plus prednisone for advanced prostate cancer.

Authors:  Ian F Tannock; Ronald de Wit; William R Berry; Jozsef Horti; Anna Pluzanska; Kim N Chi; Stephane Oudard; Christine Théodore; Nicholas D James; Ingela Turesson; Mark A Rosenthal; Mario A Eisenberger
Journal:  N Engl J Med       Date:  2004-10-07       Impact factor: 91.245

7.  The 16,17-double bond is needed for irreversible inhibition of human cytochrome p45017alpha by abiraterone (17-(3-pyridyl)androsta-5, 16-dien-3beta-ol) and related steroidal inhibitors.

Authors:  M Jarman; S E Barrie; J M Llera
Journal:  J Med Chem       Date:  1998-12-31       Impact factor: 7.446

8.  A randomized, placebo-controlled trial of zoledronic acid in patients with hormone-refractory metastatic prostate carcinoma.

Authors:  Fred Saad; Donald M Gleason; Robin Murray; Simon Tchekmedyian; Peter Venner; Louis Lacombe; Joseph L Chin; Jeferson J Vinholes; J Allen Goas; Bee Chen
Journal:  J Natl Cancer Inst       Date:  2002-10-02       Impact factor: 13.506

9.  Design and end points of clinical trials for patients with progressive prostate cancer and castrate levels of testosterone: recommendations of the Prostate Cancer Clinical Trials Working Group.

Authors:  Howard I Scher; Susan Halabi; Ian Tannock; Michael Morris; Cora N Sternberg; Michael A Carducci; Mario A Eisenberger; Celestia Higano; Glenn J Bubley; Robert Dreicer; Daniel Petrylak; Philip Kantoff; Ethan Basch; William Kevin Kelly; William D Figg; Eric J Small; Tomasz M Beer; George Wilding; Alison Martin; Maha Hussain
Journal:  J Clin Oncol       Date:  2008-03-01       Impact factor: 44.544

10.  Multinational, double-blind, phase III study of prednisone and either satraplatin or placebo in patients with castrate-refractory prostate cancer progressing after prior chemotherapy: the SPARC trial.

Authors:  Cora N Sternberg; Daniel P Petrylak; Oliver Sartor; J Alfred Witjes; Tomasz Demkow; Jean-Marc Ferrero; Jean-Christophe Eymard; Silvia Falcon; Fabio Calabrò; Nicholas James; Istvan Bodrogi; Peter Harper; Manfred Wirth; William Berry; Michael E Petrone; Thomas J McKearn; Mojtaba Noursalehi; Martine George; Marcel Rozencweig
Journal:  J Clin Oncol       Date:  2009-10-05       Impact factor: 44.544

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  827 in total

Review 1.  Use of prednisone with abiraterone acetate in metastatic castration-resistant prostate cancer.

Authors:  Richard J Auchus; Margaret K Yu; Suzanne Nguyen; Suneel D Mundle
Journal:  Oncologist       Date:  2014-10-31

2.  Clinical significance of D4A in prostate cancer therapy with abiraterone.

Authors:  Hamid Emamekhoo; Zhenfei Li; Nima Sharifi
Journal:  Cell Cycle       Date:  2015       Impact factor: 4.534

3.  [Chemotherapy of prostate cancer].

Authors:  C-H Ohlmann
Journal:  Urologe A       Date:  2015-10       Impact factor: 0.639

Review 4.  Practical guide to the use of abiraterone in castration resistant prostate cancer.

Authors:  Elahe A Mostaghel; Daniel W Lin
Journal:  Can J Urol       Date:  2014-04       Impact factor: 1.344

5.  Gene Expression Analysis of Immunomagnetically Enriched Circulating Tumor Cell Fraction in Castration-Resistant Prostate Cancer.

Authors:  Markéta Škereňová; Veronika Mikulová; Otakar Čapoun; David Švec; Katarína Kološtová; Viktor Soukup; Hana Honová; Tomáš Hanuš; Tomáš Zima
Journal:  Mol Diagn Ther       Date:  2018-06       Impact factor: 4.074

6.  Docetaxel and dasatinib or placebo in men with metastatic castration-resistant prostate cancer (READY): a randomised, double-blind phase 3 trial.

Authors:  John C Araujo; Géralyn C Trudel; Fred Saad; Andrew J Armstrong; Evan Y Yu; Joaquim Bellmunt; George Wilding; John McCaffrey; Sergio V Serrano; Vsevolod B Matveev; Eleni Efstathiou; Stephane Oudard; Michael J Morris; Bruce Sizer; Peter J Goebell; Axel Heidenreich; Johann S de Bono; Stephen Begbie; Jun H Hong; Eduardo Richardet; Enrique Gallardo; Prashni Paliwal; Susan Durham; Shinta Cheng; Christopher J Logothetis
Journal:  Lancet Oncol       Date:  2013-11-08       Impact factor: 41.316

7.  Predicting Time From Metastasis to Overall Survival in Castration-Resistant Prostate Cancer: Results From SEARCH.

Authors:  Daniel M Moreira; Lauren E Howard; Katharine N Sourbeer; Hiruni S Amarasekara; Lydia C Chow; Dillon C Cockrell; Connor L Pratson; Brian T Hanyok; William J Aronson; Christopher J Kane; Martha K Terris; Christopher L Amling; Matthew R Cooperberg; Stephen J Freedland
Journal:  Clin Genitourin Cancer       Date:  2016-08-31       Impact factor: 2.872

8.  Lysine-specific demethylase 1 has dual functions as a major regulator of androgen receptor transcriptional activity.

Authors:  Changmeng Cai; Housheng Hansen He; Shuai Gao; Sen Chen; Ziyang Yu; Yanfei Gao; Shaoyong Chen; Mei Wei Chen; Jesse Zhang; Musaddeque Ahmed; Yang Wang; Eric Metzger; Roland Schüle; X Shirley Liu; Myles Brown; Steven P Balk
Journal:  Cell Rep       Date:  2014-12-04       Impact factor: 9.423

Review 9.  The evolving role of cytotoxic chemotherapy in the management of patients with metastatic prostate cancer.

Authors:  Elan Diamond; María del Carmen Garcias; Beerinder Karir; Scott T Tagawa
Journal:  Curr Treat Options Oncol       Date:  2015-02

10.  An imaging agent to detect androgen receptor and its active splice variants in prostate cancer.

Authors:  Yusuke Imamura; Amy H Tien; Jinhe Pan; Jacky K Leung; Carmen A Banuelos; Kunzhong Jian; Jun Wang; Nasrin R Mawji; Javier Garcia Fernandez; Kuo-Shyan Lin; Raymond J Andersen; Marianne D Sadar
Journal:  JCI Insight       Date:  2016-07-21
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