Literature DB >> 23170990

A multicentre, multinational, randomized, placebo-controlled, double-blind, phase 3 trial to evaluate the efficacy and safety of gemigliptin (LC15-0444) in patients with type 2 diabetes.

S J Yang1, K W Min, S K Gupta, J Y Park, V K Shivane, S U Pitale, P K Agarwal, A Sosale, P Gandhi, M Dharmalingam, V Mohan, U Mahesh, D M Kim, Y S Kim, J A Kim, P K Kim, S H Baik.   

Abstract

AIM: This study was designed to assess the efficacy and safety of the dipeptidyl peptidase IV inhibitor gemigliptin (LC15-0444) 50 mg versus placebo in patients with type 2 diabetes.
METHODS: We conducted a 24-week, randomized, double-blind, placebo-controlled phase III trial in 182 patients (74 from Korea and 108 from India) with type 2 diabetes. After an initial 2 weeks of a diet and exercise programme followed by 2 weeks of a single-blind placebo run-in period, eligible patients were randomized to gemigliptin 50 mg or placebo, receiving the assigned treatment for 24 weeks. HbA1c and fasting plasma glucose (FPG) were measured periodically, and oral glucose tolerance test was performed at baseline and weeks 12 and 24.
RESULTS: At week 24, gemigliptin treatment led to significant reductions in HbA1c measurements compared to placebo (adjust mean after subtracting the placebo effect size: -0.71%, 95% confidence interval: -1.04 to -0.37%). A significantly greater proportion of patients achieved an HbA1c <7% with gemigliptin than with placebo. The placebo-subtracted FPG change from baseline at week 24 was -19.80 mg/dl. The overall incidence rates for adverse events were similar in the gemigliptin and placebo groups.
CONCLUSIONS: This study showed the efficacy and safety of gemigliptin 50 mg administered once daily as a monotherapy for type 2 diabetes patients.
© 2012 Blackwell Publishing Ltd.

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Year:  2012        PMID: 23170990     DOI: 10.1111/dom.12042

Source DB:  PubMed          Journal:  Diabetes Obes Metab        ISSN: 1462-8902            Impact factor:   6.577


  23 in total

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4.  Pharmacokinetic and pharmacodynamic interaction between gemigliptin and metformin in healthy subjects.

Authors:  Dongseong Shin; Young Min Cho; SeungHwan Lee; Kyoung Soo Lim; Jeong-Ae Kim; Ji-Yung Ahn; Joo-Youn Cho; Howard Lee; In-Jin Jang; Kyung-Sang Yu
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Review 6.  Gemigliptin: An Update of Its Clinical Use in the Management of Type 2 Diabetes Mellitus.

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Journal:  Drug Des Devel Ther       Date:  2014-06-03       Impact factor: 4.162

10.  Evaluation of pharmacokinetic drug interactions between gemigliptin (dipeptidylpeptidase-4 inhibitor) and glimepiride (sulfonylurea) in healthy volunteers.

Authors:  Hee Youn Choi; Yo Han Kim; Mi Jo Kim; Shi Hyang Lee; Keunsu Bang; Song Han; Hyeong-Seok Lim; Kyun-Seop Bae
Journal:  Drugs R D       Date:  2014-09
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