Literature DB >> 23153913

Selective factor XIIa inhibition attenuates silent brain ischemia: application of molecular imaging targeting coagulation pathway.

John W Chen1, Jose-Luiz Figueiredo, Gregory R Wojtkiewicz, Cory Siegel, Yoshiko Iwamoto, Dong-Eog Kim, Marc W Nolte, Gerhard Dickneite, Ralph Weissleder, Matthias Nahrendorf.   

Abstract

OBJECTIVES: The purpose of this study was use molecular imaging targeting coagulation pathway and inflammation to better understand the pathophysiology of silent brain ischemia (SBI) and monitor the effects of factor XIIa inhibition.
BACKGROUND: SBI can be observed in patients who undergo invasive vascular procedures. Unlike acute stroke, the diffuse nature of SBI and its less tangible clinical symptoms make this disease difficult to diagnose and treat.
METHODS: We induced SBI in mice by intra-arterial injection of fluorescently labeled microbeads or fractionated clot into the carotid artery. After SBI induction, diffusion-weighted magnetic resonance imaging was performed to confirm the presence of microinfarcts in asymptomatic mice. Molecular imaging targeting the downstream factor XIII activity (single-photon emission computed tomography/computed tomography) at 3 h and myeloperoxidase activity (magnetic resonance imaging) on day 3 after SBI induction were performed, without and with the intravenous administration of a recombinant selective factor XIIa inhibitor derived from the hematophagous insect Triatoma infestans (rHA-Infestin-4). Statistical comparisons between 2 groups were evaluated by the Student t test or Mann-Whitney U test.
RESULTS: In SBI-induced mice, we found abnormal activation of the coagulation cascade (factor XIII activity) and increased inflammation (myeloperoxidase activity) close to where emboli lodge in the brain. rHA-Infestin-4 administration significantly reduced ischemic damage (53% to 85% reduction of infarct volume, p < 0.05) and pathological coagulation (35% to 39% reduction of factor XIII activity, p < 0.05) without increasing hemorrhagic frequency. Myeloperoxidase activity, when normalized to the infarct volume, did not significantly change with rHA-Infestin-4 treatment, suggesting that this treatment does not further decrease inflammation other than that resulting from the reduction in infarct volume.
CONCLUSIONS: Focal intracerebral clotting and inflammatory activity are part of the pathophysiology underlying SBI. Inhibiting factor XIIa with rHA-Infestin-4 may present a safe and effective treatment to decrease the morbidity of SBI.
Copyright © 2012 American College of Cardiology Foundation. Published by Elsevier Inc. All rights reserved.

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Year:  2012        PMID: 23153913      PMCID: PMC3502014          DOI: 10.1016/j.jcmg.2012.01.025

Source DB:  PubMed          Journal:  JACC Cardiovasc Imaging        ISSN: 1876-7591


  29 in total

1.  Factor XIII deficiency causes cardiac rupture, impairs wound healing, and aggravates cardiac remodeling in mice with myocardial infarction.

Authors:  Matthias Nahrendorf; Kai Hu; Stefan Frantz; Farouc A Jaffer; Ching-Hsuan Tung; Karl-Heinz Hiller; Sabine Voll; Peter Nordbeck; David Sosnovik; Stefan Gattenlöhner; Mikhail Novikov; Gerhard Dickneite; Guy L Reed; Peter Jakob; Anthony Rosenzweig; Wolfgang R Bauer; Ralph Weissleder; Georg Ertl
Journal:  Circulation       Date:  2006-02-27       Impact factor: 29.690

2.  Factor XIIa inhibitor recombinant human albumin Infestin-4 abolishes occlusive arterial thrombus formation without affecting bleeding.

Authors:  Ina Hagedorn; Stefan Schmidbauer; Irina Pleines; Christoph Kleinschnitz; Ulrich Kronthaler; Guido Stoll; Gerhard Dickneite; Bernhard Nieswandt
Journal:  Circulation       Date:  2010-03-22       Impact factor: 29.690

3.  Imaging of myeloperoxidase in mice by using novel amplifiable paramagnetic substrates.

Authors:  John W Chen; Manel Querol Sans; Alexei Bogdanov; Ralph Weissleder
Journal:  Radiology       Date:  2006-08       Impact factor: 11.105

4.  Modulation of the human monocyte binding site for monomeric immunoglobulin G by activated Hageman factor.

Authors:  P Chien; R A Pixley; L G Stumpo; R W Colman; A D Schreiber
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5.  Protease imaging of human atheromata captures molecular information of atherosclerosis, complementing anatomic imaging.

Authors:  Dong-Eog Kim; Jeong-Yeon Kim; Dawid Schellingerhout; Eo-Jin Kim; Hyang Kyoung Kim; Seulki Lee; Kwangmeyung Kim; Ick Chan Kwon; Soo-Min Shon; Sang-Wuk Jeong; So-Hyang Im; Dong Kun Lee; Myoung Mook Lee; Geun-Eun Kim
Journal:  Arterioscler Thromb Vasc Biol       Date:  2010-01-07       Impact factor: 8.311

6.  A rapid, reliable, and valid method for measuring infarct and brain compartment volumes from computed tomographic scans.

Authors:  P D Lyden; R Zweifler; Z Mahdavi; L Lonzo
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Review 7.  Silent cerebral ischaemia: hidden fingerprints of invasive medical procedures.

Authors:  Martin Bendszus; Guido Stoll
Journal:  Lancet Neurol       Date:  2006-04       Impact factor: 44.182

8.  Tracking the inflammatory response in stroke in vivo by sensing the enzyme myeloperoxidase.

Authors:  Michael O Breckwoldt; John W Chen; Lars Stangenberg; Elena Aikawa; Elisenda Rodriguez; Shumei Qiu; Michael A Moskowitz; Ralph Weissleder
Journal:  Proc Natl Acad Sci U S A       Date:  2008-11-14       Impact factor: 11.205

9.  Activatable magnetic resonance imaging agent reports myeloperoxidase activity in healing infarcts and noninvasively detects the antiinflammatory effects of atorvastatin on ischemia-reperfusion injury.

Authors:  Matthias Nahrendorf; David Sosnovik; John W Chen; Peter Panizzi; Jose-Luiz Figueiredo; Elena Aikawa; Peter Libby; Filip K Swirski; Ralph Weissleder
Journal:  Circulation       Date:  2008-02-11       Impact factor: 29.690

10.  Defective thrombus formation in mice lacking coagulation factor XII.

Authors:  Thomas Renné; Miroslava Pozgajová; Sabine Grüner; Kai Schuh; Hans-Ulrich Pauer; Peter Burfeind; David Gailani; Bernhard Nieswandt
Journal:  J Exp Med       Date:  2005-07-11       Impact factor: 14.307

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  9 in total

1.  Factor XII inhibition reduces thrombus formation in a primate thrombosis model.

Authors:  Anton Matafonov; Philberta Y Leung; Adam E Gailani; Stephanie L Grach; Cristina Puy; Qiufang Cheng; Mao-Fu Sun; Owen J T McCarty; Erik I Tucker; Hiroaki Kataoka; Thomas Renné; James H Morrissey; Andras Gruber; David Gailani
Journal:  Blood       Date:  2014-01-09       Impact factor: 22.113

2.  Novel contact-kinin inhibitor sylvestin targets thromboinflammation and ameliorates ischemic stroke.

Authors:  Zhiye Zhang; Chuanbin Shen; Mingqian Fang; Yajun Han; Chengbo Long; Weihui Liu; Min Yang; Ming Liu; Dengdeng Zhang; Qiqi Cao; Xue Chen; Yaqun Fang; Qiumin Lu; Zongliu Hou; Yaxiong Li; Zhenze Liu; Xi Lei; Heyu Ni; Ren Lai
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3.  Radionuclide Imaging of Atherothrombotic Diseases.

Authors:  Mitchel R Stacy
Journal:  Curr Cardiovasc Imaging Rep       Date:  2019-03-27

4.  Imaging Neuroinflammation - from Bench to Bedside.

Authors:  Benjamin Pulli; John W Chen
Journal:  J Clin Cell Immunol       Date:  2014

Review 5.  Recent advances on plasmin inhibitors for the treatment of fibrinolysis-related disorders.

Authors:  Rami A Al-Horani; Umesh R Desai
Journal:  Med Res Rev       Date:  2014-03-21       Impact factor: 12.944

Review 6.  Hypercoagulability Is a Stronger Risk Factor for Ischaemic Stroke than for Myocardial Infarction: A Systematic Review.

Authors:  Alberto Maino; Frits R Rosendaal; Ale Algra; Flora Peyvandi; Bob Siegerink
Journal:  PLoS One       Date:  2015-08-07       Impact factor: 3.240

7.  Targeting coagulation factor XII as a novel therapeutic option in brain trauma.

Authors:  Sarah Hopp; Christiane Albert-Weissenberger; Stine Mencl; Michael Bieber; Michael K Schuhmann; Christian Stetter; Bernhard Nieswandt; Peter M Schmidt; Camelia-Maria Monoranu; Irina Alafuzoff; Niklas Marklund; Marc W Nolte; Anna-Leena Sirén; Christoph Kleinschnitz
Journal:  Ann Neurol       Date:  2016-04-28       Impact factor: 10.422

8.  The Coagulation Factor XIIa Inhibitor rHA-Infestin-4 Improves Outcome after Cerebral Ischemia/Reperfusion Injury in Rats.

Authors:  Jennifer Krupka; Frauke May; Thomas Weimer; Ingo Pragst; Christoph Kleinschnitz; Guido Stoll; Con Panousis; Gerhard Dickneite; Marc W Nolte
Journal:  PLoS One       Date:  2016-01-27       Impact factor: 3.240

9.  Factor XII as a Risk Marker for Hemorrhagic Stroke: A Prospective Cohort Study.

Authors:  Kristina Johansson; Jan-Håkan Jansson; Lars Johansson; Ingemar Bylesjö; Torbjörn K Nilsson; Mats Eliasson; Stefan Söderberg; Marcus Lind
Journal:  Cerebrovasc Dis Extra       Date:  2017-04-21
  9 in total

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