Literature DB >> 23053328

Dosimetry of 223Ra-chloride: dose to normal organs and tissues.

Michael Lassmann1, Dietmar Nosske.   

Abstract

PURPOSE: (223)Ra-Chloride (also called Alpharadin®) targets bone metastases with short range alpha particles. In recent years several clinical trials have been carried out showing, in particular, the safety and efficacy of palliation of painful bone metastases in patients with castration-resistant prostate cancer using (223)Ra-chloride. The purpose of this work was to provide a comprehensive dosimetric calculation of organ doses after intravenous administration of (223)Ra-chloride according to the present International Commission on Radiological Protection (ICRP) model for radium.
METHODS: Absorbed doses were calculated for 25 organs or tissues.
RESULTS: Bone endosteum and red bone marrow show the highest dose coefficients followed by liver, colon and intestines. After a treatment schedule of six intravenous injections with 0.05 MBq/kg of (223)Ra-chloride each, corresponding to 21 MBq for a 70 kg patient, the absorbed alpha dose to the bone endosteal cells is about 16 Gy and the corresponding absorbed dose to the red bone marrow is approximately 1.5 Gy.
CONCLUSION: The comprehensive list of dose coefficients presented in this work will assist in comparing and evaluating organ doses from various therapy modalities used in nuclear medicine and will provide a base for further development of patient-specific dosimetry.

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Year:  2012        PMID: 23053328     DOI: 10.1007/s00259-012-2265-y

Source DB:  PubMed          Journal:  Eur J Nucl Med Mol Imaging        ISSN: 1619-7070            Impact factor:   9.236


  14 in total

1.  Age-dependent doses to members of the public from intake of radionuclides: Part 4. Inhalation dose coefficients. A report of a task group of Committee 2 of the International Commission on Radiological Protection.

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Journal:  Ann ICRP       Date:  1995

Review 2.  High-linear energy transfer irradiation targeted to skeletal metastases by the alpha-emitter 223Ra: adjuvant or alternative to conventional modalities?

Authors:  Øyvind S Bruland; Sten Nilsson; Darrell R Fisher; Roy H Larsen
Journal:  Clin Cancer Res       Date:  2006-10-15       Impact factor: 12.531

Review 3.  A randomized, dose-response, multicenter phase II study of radium-223 chloride for the palliation of painful bone metastases in patients with castration-resistant prostate cancer.

Authors:  S Nilsson; P Strang; A K Aksnes; L Franzèn; P Olivier; A Pecking; J Staffurth; S Vasanthan; C Andersson; Ø S Bruland
Journal:  Eur J Cancer       Date:  2012-02-15       Impact factor: 9.162

4.  First clinical experience with alpha-emitting radium-223 in the treatment of skeletal metastases.

Authors:  Sten Nilsson; Roy H Larsen; Sophie D Fosså; Lise Balteskard; Kari W Borch; Jan-Erik Westlin; Gro Salberg; Oyvind S Bruland
Journal:  Clin Cancer Res       Date:  2005-06-15       Impact factor: 12.531

5.  Age-dependent doses to members of the public from intake of radionuclides: Part 2. Ingestion dose coefficients. A report of a Task Group of Committee 2 of the International Commission on Radiological Protection.

Authors: 
Journal:  Ann ICRP       Date:  1993

6.  Radiotoxicity of gadolinium-148 and radium-223 in mouse testes: relative biological effectiveness of alpha-particle emitters in vivo.

Authors:  R W Howell; S M Goddu; V R Narra; D R Fisher; R E Schenter; D V Rao
Journal:  Radiat Res       Date:  1997-03       Impact factor: 2.841

7.  Human alimentary tract model for radiological protection. ICRP Publication 100. A report of The International Commission on Radiological Protection.

Authors: 
Journal:  Ann ICRP       Date:  2006

8.  Therapy of ankylosing spondylitis with 224Ra-radium chloride: dosimetry and risk considerations.

Authors:  Michael Lassmann; Dietmar Nosske; Christoph Reiners
Journal:  Radiat Environ Biophys       Date:  2002-09-07       Impact factor: 1.925

9.  A bone marrow toxicity model for ²²³Ra alpha-emitter radiopharmaceutical therapy.

Authors:  Robert F Hobbs; Hong Song; Christopher J Watchman; Wesley E Bolch; Anne-Kirsti Aksnes; Thomas Ramdahl; Glenn D Flux; George Sgouros
Journal:  Phys Med Biol       Date:  2012-05-01       Impact factor: 3.609

10.  Bone-targeted radium-223 in symptomatic, hormone-refractory prostate cancer: a randomised, multicentre, placebo-controlled phase II study.

Authors:  Sten Nilsson; Lars Franzén; Christopher Parker; Christopher Tyrrell; René Blom; Jan Tennvall; Bo Lennernäs; Ulf Petersson; Dag C Johannessen; Michael Sokal; Katharine Pigott; Jeffrey Yachnin; Michael Garkavij; Peter Strang; Johan Harmenberg; Bjørg Bolstad; Oyvind S Bruland
Journal:  Lancet Oncol       Date:  2007-07       Impact factor: 41.316

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  33 in total

Review 1.  Clinical experience with radium-223 in the treatment of patients with advanced castrate-resistant prostate cancer and symptomatic bone metastases.

Authors:  Christina Hague; John P Logue
Journal:  Ther Adv Urol       Date:  2016-02-25

Review 2.  Treatment of Bone Metastasis with Bone-Targeting Radiopharmaceuticals.

Authors:  Joon Young Choi
Journal:  Nucl Med Mol Imaging       Date:  2018-01-12

3.  Alpha Particle Radium 223 Dichloride in High-risk Osteosarcoma: A Phase I Dose Escalation Trial.

Authors:  Vivek Subbiah; Pete M Anderson; Kalevi Kairemo; Kenneth Hess; Winston W Huh; Vinod Ravi; Najat C Daw; Neeta Somaiah; Joseph A Ludwig; Robert S Benjamin; Sant Chawla; David S Hong; Funda Meric-Bernstam; Gregory Ravizzini; Eugenie Kleinerman; Homer Macapinlac; Eric Rohren
Journal:  Clin Cancer Res       Date:  2019-02-07       Impact factor: 12.531

Review 4.  From palliative therapy to prolongation of survival: (223)RaCl2 in the treatment of bone metastases.

Authors:  Knut Liepe; Ajit Shinto
Journal:  Ther Adv Med Oncol       Date:  2016-04-25       Impact factor: 8.168

Review 5.  [Alpha emitter radium-223 dichloride: new therapy in castration-resistant prostate cancer with symptomatic bone metastases].

Authors:  H Heinzer; F König; S Klutmann
Journal:  Urologe A       Date:  2014-04       Impact factor: 0.639

Review 6.  Radium-223 dichloride: a review of its use in patients with castration-resistant prostate cancer with symptomatic bone metastases.

Authors:  Matt Shirley; Paul L McCormack
Journal:  Drugs       Date:  2014-04       Impact factor: 9.546

7.  EANM guideline for radionuclide therapy with radium-223 of metastatic castration-resistant prostate cancer.

Authors:  Thorsten D Poeppel; Daria Handkiewicz-Junak; Michael Andreeff; Alexander Becherer; Andreas Bockisch; Eva Fricke; Lilli Geworski; Alexander Heinzel; Bernd J Krause; Thomas Krause; Markus Mitterhauser; Wilfried Sonnenschein; Lisa Bodei; Roberto C Delgado-Bolton; Michael Gabriel
Journal:  Eur J Nucl Med Mol Imaging       Date:  2017-12-12       Impact factor: 9.236

8.  Dose-Dependent Growth Delay of Breast Cancer Xenografts in the Bone Marrow of Mice Treated with 223Ra: The Role of Bystander Effects and Their Potential for Therapy.

Authors:  Calvin N Leung; Brian S Canter; Didier Rajon; Tom A Bäck; J Christopher Fritton; Edouard I Azzam; Roger W Howell
Journal:  J Nucl Med       Date:  2019-09-13       Impact factor: 10.057

Review 9.  Targeted α-particle therapy of bone metastases in prostate cancer.

Authors:  Hossein Jadvar; David I Quinn
Journal:  Clin Nucl Med       Date:  2013-12       Impact factor: 7.794

Review 10.  Radium-223 dichloride in clinical practice: a review.

Authors:  Luigia Florimonte; Luca Dellavedova; Lorenzo Stefano Maffioli
Journal:  Eur J Nucl Med Mol Imaging       Date:  2016-04-28       Impact factor: 9.236

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