Literature DB >> 22909146

Cognitive effects of oxybutynin chloride topical gel in older healthy subjects: a 1-week, randomized, double-blind, placebo- and active-controlled study.

Gary G Kay1, David R Staskin, Scott MacDiarmid, Marilyn McIlwain, Naomi V Dahl.   

Abstract

BACKGROUND AND
OBJECTIVE: Oxybutynin is a common antimuscarinic therapy for overactive bladder. Transdermally administered oxybutynin chloride topical gel 10% (OTG) has a low propensity for anticholinergic adverse effects and possibly also a low risk of cognitive impairment. A randomized, double-blind, placebo- and active-controlled study evaluated the effects of OTG on cognitive and psychomotor functions in older healthy adults.
METHODS: Healthy adults aged 60-79 years were assigned randomly (1:1:1) to 1-week's treatment with OTG (1 g [100 mg oxybutynin] applied once daily on rotating sites of upper arms/shoulders, abdomen or thighs) plus oral placebo, immediate-release oxybutynin (OXB-IR; 5 mg capsule three times/day) plus placebo gel, or double placebo. Delayed recall Name-Face Association Test (NFAT) score was the primary end point. Treatments were compared by analysis of covariance.
RESULTS: Of 152 participants (mean age, 68 years), 49 received OTG, 52 OXB-IR and 51 placebo. NFAT Delayed Recall tests revealed no significant treatment differences (overall, p = 0.2733; OTG vs placebo, p = 0.1551; OXB-IR vs placebo, p = 0.1767). However, a significant effect (p = 0.0294) was noted for the Misplaced Objects Test, with scores declining only for OXB-IR. Approximately twice as many participants receiving OXB-IR (n = 10) as those receiving OTG (n = 5) or placebo (n = 6) showed a significant decline (≥6 points) in Total Recall score for the Hopkins Verbal Learning Test-Revised. No significant effects on psychomotor reaction time were observed. The most common adverse event, dry mouth, occurred in 6.1%, 73.1% and 7.8% of participants receiving OTG, OXB-IR and placebo, respectively.
CONCLUSIONS: OTG applied for 1 week had no clinically meaningful effect on recent memory or other cognitive functions in healthy, older adults. CLINICAL TRIAL REGISTRATION: Registered as NCT00752141 at www.clinicaltrials.gov.

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Year:  2012        PMID: 22909146     DOI: 10.1007/BF03261924

Source DB:  PubMed          Journal:  Clin Drug Investig        ISSN: 1173-2563            Impact factor:   2.859


  19 in total

Review 1.  Pharmacotherapy for overactive bladder: an evidence-based approach to selecting an antimuscarinic agent.

Authors:  Rodney A Appell
Journal:  Drugs       Date:  2006       Impact factor: 9.546

2.  A short-term, multicenter, randomized double-blind dose titration study of the efficacy and anticholinergic side effects of transdermal compared to immediate release oral oxybutynin treatment of patients with urge urinary incontinence.

Authors:  G W Davila; C A Daugherty; S W Sanders
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3.  Comparison of oxybutynin and its active metabolite, N-desethyl-oxybutynin, in the human detrusor and parotid gland.

Authors:  K Waldeck; B Larsson; K E Andersson
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4.  Differential effects of the antimuscarinic agents darifenacin and oxybutynin ER on memory in older subjects.

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5.  Empirical methods for assessing meaningful neuropsychological change following epilepsy surgery.

Authors:  S M Sawrie; G J Chelune; R I Naugle; H O Lüders
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Review 6.  Oxybutynin chloride topical gel: a new formulation of an established antimuscarinic therapy for overactive bladder.

Authors:  David R Staskin; Dudley Robinson
Journal:  Expert Opin Pharmacother       Date:  2009-12       Impact factor: 3.889

Review 7.  Preserving cognitive function for patients with overactive bladder: evidence for a differential effect with darifenacin.

Authors:  G G Kay; U Ebinger
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8.  Efficacy and safety of transdermal oxybutynin in patients with urge and mixed urinary incontinence.

Authors:  Roger R Dmochowski; G Willy Davila; Norman R Zinner; Marc C Gittelman; Daniel R Saltzstein; Sydney Lyttle; Steven W Sanders
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10.  Measurement of oxybutynin and its N-desethyl metabolite in plasma, and its application to pharmacokinetic studies in young, elderly and frail elderly volunteers.

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Authors:  Scott C McFerren; Alex Gomelsky
Journal:  Drugs Aging       Date:  2015-10       Impact factor: 3.923

4.  Differential Prescribing of Antimuscarinic Agents in Older Adults with Cognitive Impairment.

Authors:  Scott Martin Vouri; Mario Schootman; Seth A Strope; Stanley J Birge; Margaret A Olsen
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Review 5.  An update on the use of transdermal oxybutynin in the management of overactive bladder disorder.

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Review 6.  Pharmacotherapy of overactive bladder in adults: a review of efficacy, tolerability, and quality of life.

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Review 7.  Overactive bladder - 18 years - Part II.

Authors:  Jose Carlos Truzzi; Cristiano Mendes Gomes; Carlos A Bezerra; Ivan Mauricio Plata; Jose Campos; Gustavo Luis Garrido; Fernando G Almeida; Marcio Augusto Averbeck; Alexandre Fornari; Anibal Salazar; Arturo Dell'Oro; Caio Cintra; Carlos Alberto Ricetto Sacomani; Juan Pablo Tapia; Eduardo Brambila; Emilio Miguel Longo; Flavio Trigo Rocha; Francisco Coutinho; Gabriel Favre; Jose Antonio Garcia; Juan Castano; Miguel Reyes; Rodrigo Eugenio Leyton; Ruiter Silva Ferreira; Sergio Duran; Vanda Lopez; Ricardo Reges
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Review 8.  A Guide to Medications Inducing Salivary Gland Dysfunction, Xerostomia, and Subjective Sialorrhea: A Systematic Review Sponsored by the World Workshop on Oral Medicine VI.

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Review 9.  Clinical utility of transdermal delivery of oxybutynin gel via a metered-dose pump in the management of overactive bladder.

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