Literature DB >> 22855172

Intraperitoneal bevacizumab combined with cytoreductive surgery: a pre-clinical study of tolerance and pharmacokinetics in an animal model.

Guillaume Passot1, Aurélien Dupré, Michel Rivoire, Faheez Mohamed, Naoual Bakrin, Olivier Glehen.   

Abstract

INTRODUCTION: Cytoreductive Surgery (CRS) combined with Hyperthermic Intraperitoneal Chemotherapy (HIPEC) is currently the only potentially curative treatment for peritoneal carcinomatosis (PC). Systemic administration of bevacizumab improves survival in patients with metastatic colorectal or ovarian cancer. Intraperitoneal administration of bevacizumab has been shown to be safe and effective in treating malignant ascites. The combination of CRS with intraperitoneal (IP) bevacizumab could maximize local control and survival from PC, but the associated morbidity from this is unknown. The aim of this study was to evaluate the safety of the combination of CRS with IP bevacizumab and to determine the pharmacokinetics of the drug in a rabbit model.
METHODS: Twenty healthy rabbits underwent a standardized procedure of debulking surgery, including peritonectomy and gastrointestinal anastomosis and were randomized to receive IP bevacizumab (25 mg/kg) or placebo. Another group of three rabbits underwent an instillation of IP bevacizumab (25 mg/kg) without surgery.
RESULTS: One rabbit that received IP bevacizumab died with no complication associated with the use of bevacizumab at autopsy. There was no significant difference between IP bevacizumab and placebo in weight loss, length of surgery or morbidity. The plasma concentration of bevacizumab increased to a peak at 24 h post IP administration. Bevacizumab was not detected in the plasma of animals without surgery.
CONCLUSION: This study suggests that IP bevacizumab does not increase morbidity and mortality of debulking surgery in an animal model. When surgery is performed, the pharmacokinetics of IP bevacizumab are modified in plasma.

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Year:  2012        PMID: 22855172     DOI: 10.1007/s12094-012-0888-x

Source DB:  PubMed          Journal:  Clin Transl Oncol        ISSN: 1699-048X            Impact factor:   3.405


  41 in total

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2.  Surgical wound healing complications in metastatic colorectal cancer patients treated with bevacizumab.

Authors:  Frank A Scappaticci; Louis Fehrenbacher; Thomas Cartwright; John D Hainsworth; William Heim; Jordan Berlin; Fairooz Kabbinavar; William Novotny; Somnath Sarkar; Herbert Hurwitz
Journal:  J Surg Oncol       Date:  2005-09-01       Impact factor: 3.454

3.  Preoperative serum vascular endothelial growth factor as a prognostic parameter in ovarian cancer.

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Journal:  Gynecol Oncol       Date:  2006-06-05       Impact factor: 5.482

4.  Pharmacology and pharmacodynamics of bevacizumab as monotherapy or in combination with cytotoxic therapy in preclinical studies.

Authors:  Hans-Peter Gerber; Napoleone Ferrara
Journal:  Cancer Res       Date:  2005-02-01       Impact factor: 12.701

5.  Peritoneal VEGF burden as a predictor of cytoreductive surgery outcome in women with epithelial ovarian cancer.

Authors:  Solange Maria Diniz Bizzo; Débora Dummer Meira; José Marinaldo Lima; Jânio da Silva Mororó; José Cláudio Casali-da-Rocha; Maria Helena Faria Ornellas
Journal:  Int J Gynaecol Obstet       Date:  2010-02-18       Impact factor: 3.561

Review 6.  Systemic chemotherapy in the management of malignant peritoneal mesothelioma.

Authors:  R Garcia-Carbonero; L Paz-Ares
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7.  Phase II trial of bevacizumab in persistent or recurrent epithelial ovarian cancer or primary peritoneal cancer: a Gynecologic Oncology Group Study.

Authors:  Robert A Burger; Michael W Sill; Bradley J Monk; Benjamin E Greer; Joel I Sorosky
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8.  Suppressive effect of bevacizumab on peritoneal dissemination from gastric cancer in a peritoneal metastasis model.

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Journal:  Surg Today       Date:  2010-08-26       Impact factor: 2.549

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Journal:  N Engl J Med       Date:  2004-06-03       Impact factor: 91.245

10.  Direct evidence that the VEGF-specific antibody bevacizumab has antivascular effects in human rectal cancer.

Authors:  Christopher G Willett; Yves Boucher; Emmanuelle di Tomaso; Dan G Duda; Lance L Munn; Ricky T Tong; Daniel C Chung; Dushyant V Sahani; Sanjeeva P Kalva; Sergey V Kozin; Mari Mino; Kenneth S Cohen; David T Scadden; Alan C Hartford; Alan J Fischman; Jeffrey W Clark; David P Ryan; Andrew X Zhu; Lawrence S Blaszkowsky; Helen X Chen; Paul C Shellito; Gregory Y Lauwers; Rakesh K Jain
Journal:  Nat Med       Date:  2004-01-25       Impact factor: 53.440

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  5 in total

1.  The effects of bevacizumab on intestinal anastomotic healing in rabbits.

Authors:  Hayato Nakamura; Yukihiro Yokoyama; Keisuke Uehara; Toshio Kokuryo; Junpei Yamaguchi; Toyonori Tsuzuki; Masato Nagino
Journal:  Surg Today       Date:  2016-05-12       Impact factor: 2.549

Review 2.  Peritoneal metastases of colorectal origin treated by cytoreduction and HIPEC: An overview.

Authors:  Alvaro Arjona-Sánchez; Francisco Javier Medina-Fernández; Francisco Cristobal Muñoz-Casares; Angela Casado-Adam; Juan Manuel Sánchez-Hidalgo; Sebastián Rufián-Peña
Journal:  World J Gastrointest Oncol       Date:  2014-10-15

3.  Cytoreductive surgery (SRC) and hyperthermic intraperitoneal chemotherapy (HIPEC) for treatment of peritoneal carcinomatosis: Our initial experience and technical details.

Authors:  Koray Topgül; Mehmet Bilge Çetinkaya; N Çiğdem Arslan; Mustafa Kemal Gül; Murat Çan; Mahmut Fikret Gürsel; Dilek Erdem; Zafer Malazgirt
Journal:  Ulus Cerrahi Derg       Date:  2015-09-01

Review 4.  Cytoreductive surgery with intraperitoneal chemotherapy in the management of peritoneal surface malignancy: a pharmacist's perspective.

Authors:  Priya Mistry; Faheez Mohamed; Sanjeev Dayal; Tom D Cecil; Brendan J Moran
Journal:  Eur J Hosp Pharm       Date:  2016-04-05

5.  Angiogenesis-Related Markers and Prognosis After Cytoreductive Surgery and Hyperthermic Intraperitoneal Chemotherapy for Metastatic Colorectal Cancer.

Authors:  E M V de Cuba; I H J T de Hingh; N R Sluiter; R Kwakman; V M H Coupé; J A M Beliën; V J Verwaal; W J H J Meijerink; P M Delis-van Diemen; H J Bonjer; G A Meijer; E A Te Velde
Journal:  Ann Surg Oncol       Date:  2016-01-04       Impact factor: 5.344

  5 in total

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