Literature DB >> 22854885

I2 promoted domino oxidative cyclization for one-pot synthesis of 2-acylbenzothiazoles via metal-free sp3 C-H functionalization.

Yan-Ping Zhu1, Mi Lian, Feng-Cheng Jia, Mei-Cai Liu, Jing-Jing Yuan, Qing-He Gao, An-Xin Wu.   

Abstract

An I(2) promoted domino protocol was developed to construct 2-acylbenzothiazoles from simple and readily available aromatic ketones/unsaturated methyl ketones and o-aminobenzenethiols. The reaction proceeded smoothly under metal-free and peroxide-free conditions.

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Year:  2012        PMID： 22854885     DOI： 10.1039/c2cc34561g

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  3 in total

1.  Reagent-controlled regiodivergent intermolecular cyclization of 2-aminobenzothiazoles with β-ketoesters and β-ketoamides.

Authors:  Irwan Iskandar Roslan; Kian-Hong Ng; Gaik-Khuan Chuah; Stephan Jaenicke
Journal:  Beilstein J Org Chem       Date:  2017-12-18       Impact factor: 2.883

2.  S8-Catalyzed triple cleavage of bromodifluoro compounds for the assembly of N-containing heterocycles.

Authors:  Shuilin Deng; Haohua Chen; Xingxing Ma; Yao Zhou; Kai Yang; Yu Lan; Qiuling Song
Journal:  Chem Sci       Date:  2019-06-05       Impact factor: 9.825

3.  Chalcones and Five-Membered Heterocyclic Isosteres Bind to Alpha Synuclein Fibrils in Vitro.

Authors:  Chia-Ju Hsieh; Kuiying Xu; Iljung Lee; Thomas J A Graham; Zhude Tu; Dhruva Dhavale; Paul Kotzbauer; Robert H Mach
Journal:  ACS Omega       Date:  2018-04-24
  3 in total

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