Literature DB >> 22809630

Continuous glucose profiles with vildagliptin versus sitagliptin in add-on to metformin: results from the randomized Optima study.

B Guerci1, L Monnier, P Serusclat, C Petit, P Valensi, D Huet, D Raccah, C Colette, S Quéré, S Dejager.   

Abstract

AIM: To compare continuous glucose monitoring (CGM) profiles on vildagliptin versus sitagliptin in addition to metformin, in patients with inadequately controlled type 2 diabetes mellitus (HbA(1c) 6.5-8.0%).
METHODS: A multicenter, prospective, randomised, open-label study with blinded endpoint analysis. CGM data acquired over three days--firstly on metformin alone and then 8 weeks after the addition of either vildagliptin (n=14) or sitagliptin (n=16)--were blinded and analyzed centrally.
RESULTS: In comparable populations with a mean baseline HbA1c of 7.1%, 24-hour glucose variability--measured by mean amplitude of glucose excursions and standard deviation of mean glucose concentration--showed similar improvement on both drugs versus metformin alone. In contrast, a series of predefined parameters reflecting daily glycaemic control--mean 24-hour blood glucose concentration, and the times spent in the optimal glycaemic range (70-140 mg/dL) and above the hyperglycaemic thresholds of 140 and 180 mg/dL together with the corresponding AUC values--were significantly improved from baseline only in the vildagliptin arm. In addition, overall hyperglycaemia (AUC[24 h] > 100 mg/dL) significantly dropped from baseline on vildagliptin [-37%] but not on sitagliptin [-9%], while postprandial hyperglycaemia (AUC[0-4 h] × 3) was significantly reduced on both, and basal hyperglycaemia (overall--postprandial hyperglycaemia was reduced only on vildagliptin [-41%; P = 0.04]).
CONCLUSIONS: The addition of a DPP-4 inhibitor significantly reduced glycaemic variability with no difference between the two drugs. However, vildagliptin induced better circadian glycaemic control than sitagliptin with a significant decrease on overall hyperglycemia, mainly driven by reduction on basal hyperglycaemia.
Copyright © 2012 Elsevier Masson SAS. All rights reserved.

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Year:  2012        PMID: 22809630     DOI: 10.1016/j.diabet.2012.06.001

Source DB:  PubMed          Journal:  Diabetes Metab        ISSN: 1262-3636            Impact factor:   6.041


  24 in total

Review 1.  Near normal HbA1c with stable glucose homeostasis: the ultimate target/aim of diabetes therapy.

Authors:  L Monnier; C Colette; S Dejager; D R Owens
Journal:  Rev Endocr Metab Disord       Date:  2016-03       Impact factor: 6.514

Review 2.  Vildagliptin: a review of its use in type 2 diabetes mellitus.

Authors:  Gillian M Keating
Journal:  Drugs       Date:  2014-04       Impact factor: 9.546

3.  The renoprotective effect and safety of a DPP-4 inhibitor, sitagliptin, at a small dose in type 2 diabetic patients with a renal dysfunction when changed from other DPP-4 inhibitors: REAL trial.

Authors:  Koichi Kanozawa; Yuichi Noguchi; Souichi Sugahara; Satoko Nakamura; Hirohisa Yamamoto; Keiko Kaneko; Rika Kono; Saeko Sato; Tomonari Ogawa; Hajime Hasegawa; Shigehiro Katayama
Journal:  Clin Exp Nephrol       Date:  2017-12-23       Impact factor: 2.801

4.  Exercise at lunchtime: effect on glycemic control and oxidative stress in middle-aged men with type 2 diabetes.

Authors:  Jonida Haxhi; Gaetano Leto; Alessandro Scotto di Palumbo; Paola Sbriccoli; Laura Guidetti; Cristina Fantini; Raffaella Buzzetti; Daniela Caporossi; Luigi Di Luigi; Massimo Sacchetti
Journal:  Eur J Appl Physiol       Date:  2015-12-28       Impact factor: 3.078

Review 5.  Glycemic Variability: Risk Factors, Assessment, and Control.

Authors:  Boris Kovatchev
Journal:  J Diabetes Sci Technol       Date:  2019-01-29

Review 6.  Metrics for glycaemic control - from HbA1c to continuous glucose monitoring.

Authors:  Boris P Kovatchev
Journal:  Nat Rev Endocrinol       Date:  2017-03-17       Impact factor: 43.330

7.  Dipeptidyl peptidase-4 inhibitors and the risk of heart failure: a systematic review and meta-analysis.

Authors:  Subodh Verma; Ronald M Goldenberg; Deepak L Bhatt; Michael E Farkouh; Adrian Quan; Hwee Teoh; Kim A Connelly; Lawrence A Leiter; Jan O Friedrich
Journal:  CMAJ Open       Date:  2017-02-24

8.  Recommendations for Practical Use of Metformin, a Central Pharmacological Therapy in Type 2 Diabetes.

Authors:  Inês H Vieira; Luísa M Barros; Carla F Baptista; Dírcea M Rodrigues; Isabel M Paiva
Journal:  Clin Diabetes       Date:  2022-01

Review 9.  Glycemic variability and acute ischemic stroke: the missing link?

Authors:  Emmanuel I González-Moreno; Carlos R Cámara-Lemarroy; José G González-González; Fernando Góngora-Rivera
Journal:  Transl Stroke Res       Date:  2014-08-03       Impact factor: 6.829

10.  Dipeptidyl peptidase-4 inhibitor improves glycemic variability in multiple daily insulin-treated type 2 diabetes: a prospective randomized-controlled trial.

Authors:  Fukumi Yoshikawa; Tomoko Nagashima; Hiroshi Uchino; Shuki Usui; Masahiko Miyagi; Yasuyo Ando; Takahisa Hirose
Journal:  Diabetol Int       Date:  2021-06-05
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