| Literature DB >> 22749869 |
Tetsuyoshi Matsufuji1, Mika Ikeda, Asuka Naito, Masakazu Hirouchi, Hideo Takakusa, Shoichi Kanda, Masanori Izumi, Jun Harada, Tsuyoshi Shinozuka.
Abstract
The discovery, optimization and structure-activity relationship of novel FATP1 inhibitors have been described. The detailed SAR studies of each moiety of the inhibitors combined with metabolite analysis led to the identification of the potent inhibitors 11p and 11q with improved blood stability.Entities:
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Year: 2012 PMID： 22749869 DOI： 10.1016/j.bmcl.2012.05.130
Source DB: PubMed Journal: Bioorg Med Chem Lett ISSN： 0960-894X Impact factor: 2.823