Literature DB >> 22727346

Pharmacokinetics and ovarian suppression during use of a contraceptive vaginal ring in normal-weight and obese women.

Carolyn L Westhoff1, Anupama H Torgal, Elizabeth Rose Mayeda, Kelsey Petrie, Tiffany Thomas, Monica Dragoman, Serge Cremers.   

Abstract

OBJECTIVE: Many observational studies indicate higher oral contraceptive failure among obese women, but most clinical trials and physiologic studies do not support these differences. Limited data indicate higher failure rates among obese contraceptive patch users. Data regarding contraceptive vaginal ring performance in obese women are needed. STUDY
DESIGN: Twenty normal weight (body mass index [BMI] 19.0-24.9; median, 21.65) and 20 obese (BMI 30.0-39.9; median, 33.7) women enrolled in a prospective study of ethinyl estradiol (EE(2)) and etonorgestrel pharmacokinetics and of ovarian follicle development, endometrial thickness, and bleeding patterns, all measured biweekly during the second cycle of contraceptive vaginal ring use.
RESULTS: Thirty-seven women completed follow-up. Mean day 0-21 EE(2) concentrations were lower among obese vs normal weight women (15.0 vs 22.0 pg/mL, respectively, P = .004), whereas etonorgestrel concentrations were similar (1138 vs 1256 pg/mL, respectively, P = .39). Follicular development was minimal in both groups, with only 5 women achieving a maximum follicle diameter >13 mm at any time during 3 weeks follow-up (3 normal weight and 2 obese women); these women had serum progesterone levels <1.0. Obese women reported more bleeding or spotting than normal weight women (3.6 vs 1.4 days, respectively, P = .01).
CONCLUSION: Although obese women had lower EE(2) levels during contraceptive vaginal ring use, they had excellent suppression of ovarian follicle development, similar to normal weight women. This predicts that contraceptive vaginal ring effectiveness will be similar in women with a BMI up to 39.9. The lower serum EE(2) levels in the obese women may explain the greater reported bleeding or spotting days.
Copyright © 2012 Mosby, Inc. All rights reserved.

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Year:  2012        PMID: 22727346      PMCID: PMC3403702          DOI: 10.1016/j.ajog.2012.04.022

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  26 in total

1.  Use of the novel combined contraceptive vaginal ring NuvaRing for ovulation inhibition.

Authors:  T M Mulders; T O Dieben
Journal:  Fertil Steril       Date:  2001-05       Impact factor: 7.329

2.  Pharmacokinetics of etonogestrel and ethinylestradiol released from a combined contraceptive vaginal ring.

Authors:  C J Timmer; T M Mulders
Journal:  Clin Pharmacokinet       Date:  2000-09       Impact factor: 6.447

3.  Contraceptive efficacy and cycle control with the Ortho Evra/Evra transdermal system: the analysis of pooled data.

Authors:  Miriam Zieman; John Guillebaud; Edith Weisberg; Gary A Shangold; Alan C Fisher; George W Creasy
Journal:  Fertil Steril       Date:  2002-02       Impact factor: 7.329

4.  Ultrasound evaluation of ovarian activity under oral contraceptives.

Authors:  H J Hoogland; S O Skouby
Journal:  Contraception       Date:  1993-06       Impact factor: 3.375

5.  Body weight and risk of oral contraceptive failure.

Authors:  Victoria L Holt; Kara L Cushing-Haugen; Janet R Daling
Journal:  Obstet Gynecol       Date:  2002-05       Impact factor: 7.661

6.  The analysis of vaginal bleeding patterns induced by fertility regulating methods. World Health Organization Special Programme of Research, Development and Research Training in Human Reproduction.

Authors:  E M Belsey; D Machin; C d'Arcangues
Journal:  Contraception       Date:  1986-09       Impact factor: 3.375

7.  Serum steroid binding protein concentrations, distribution of progestogens, and bioavailability of testosterone during treatment with contraceptives containing desogestrel or levonorgestrel.

Authors:  G L Hammond; M S Langley; P A Robinson; S Nummi; L Lund
Journal:  Fertil Steril       Date:  1984-07       Impact factor: 7.329

8.  Manipulation of the pill-free interval in oral contraceptive pill users: the effect on follicular suppression.

Authors:  William D Schlaff; Anne M Lynch; Heather D Hughes; Marcelle I Cedars; Deborah L Smith
Journal:  Am J Obstet Gynecol       Date:  2004-04       Impact factor: 8.661

9.  Protein binding of the contraceptive steroids gestodene, 3-keto-desogestrel and ethinylestradiol in human serum.

Authors:  W Kuhnz; M Pfeffer; G al-Yacoub
Journal:  J Steroid Biochem       Date:  1990-02       Impact factor: 4.292

10.  Derivatization of ethinylestradiol with dansyl chloride to enhance electrospray ionization: application in trace analysis of ethinylestradiol in rhesus monkey plasma.

Authors:  M Reza Anari; Ray Bakhtiar; Bing Zhu; Su Huskey; Ronald B Franklin; David C Evans
Journal:  Anal Chem       Date:  2002-08-15       Impact factor: 6.986

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  11 in total

1.  Prolonged use of the etonogestrel implant and levonorgestrel intrauterine device: 2 years beyond Food and Drug Administration-approved duration.

Authors:  Colleen McNicholas; Erin Swor; Leping Wan; Jeffrey F Peipert
Journal:  Am J Obstet Gynecol       Date:  2017-01-29       Impact factor: 8.661

Review 2. 

Authors:  Sabrina Lorico; Blaine Colton
Journal:  Can Fam Physician       Date:  2020-06       Impact factor: 3.275

Review 3.  Obesity and hormonal contraceptive efficacy.

Authors:  Jennifer A Robinson; Anne E Burke
Journal:  Womens Health (Lond)       Date:  2013-09

4.  Pharmacokinetics of Hormonal Contraception in Individuals with Obesity: a Review.

Authors:  Shaalini Ramanadhan; William J Jusko; Alison Edelman
Journal:  Curr Obstet Gynecol Rep       Date:  2020-05-04

5.  Contraceptive vaginal ring effectiveness is maintained during 6 weeks of use: a prospective study of normal BMI and obese women.

Authors:  Monica Dragoman; Kelsey Petrie; Anupama Torgal; Tiffany Thomas; Serge Cremers; Carolyn L Westhoff
Journal:  Contraception       Date:  2012-12-10       Impact factor: 3.375

Review 6.  Clarification of contraceptive drug pharmacokinetics in obesity.

Authors:  William J Jusko
Journal:  Contraception       Date:  2016-08-16       Impact factor: 3.375

7.  A UPLC-MS/MS method for therapeutic drug monitoring of etonogestrel.

Authors:  Tiffany Thomas; Kelsey Petrie; Joonho Shim; Kirsten M Abildskov; Carolyn L Westhoff; Serge Cremers
Journal:  Ther Drug Monit       Date:  2013-12       Impact factor: 3.681

Review 8.  Medication management and pharmacokinetic changes after bariatric surgery.

Authors:  Sabrina Lorico; Blaine Colton
Journal:  Can Fam Physician       Date:  2020-06       Impact factor: 3.275

Review 9.  Hormonal contraceptives for contraception in overweight or obese women.

Authors:  Laureen M Lopez; Alissa Bernholc; Mario Chen; Thomas W Grey; Conrad Otterness; Carolyn Westhoff; Alison Edelman; Frans M Helmerhorst
Journal:  Cochrane Database Syst Rev       Date:  2016-08-18

Review 10.  Pharmacokinetics, metabolism and serum concentrations of progestins used in contraception.

Authors:  Alexis J Bick; Renate Louw-du Toit; Salndave B Skosana; Donita Africander; Janet P Hapgood
Journal:  Pharmacol Ther       Date:  2020-12-13       Impact factor: 13.400

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