Literature DB >> 22672501

Effects of a vildagliptin/metformin combination on markers of atherosclerosis, thrombosis, and inflammation in diabetic patients with coronary artery disease.

Robert Klempfner1, Jonathan Leor, Alexander Tenenbaum, Enrique Z Fisman, Ilan Goldenberg.   

Abstract

BACKGROUND: Diabetic patients present with an accelerated atherosclerotic process and an increased risk for future cardiovascular events. In addition to the risk imposed by the disease itself, pharmacological treatment adds also a sizable risk, especially if certain classes of antidiabetic drugs are employed. Animal evidence indicates that dipeptidyl peptidase-4 inhibitors have anti-atherosclerotic effects, yet clinical data are scarcely available.
DESIGN: We plan to prospectively investigate the effects of dipeptidyl peptidase-4 inhibition with vildagliptin on a number of atherothrombotic markers and adipokines in patients with proven atherosclerosis and type 2 diabetes. The selected markers are: interleukin-6, high sensitivity C reactive protein, interleukin 1-beta, total adiponectin levels, matrix metallo-proteinase 9 and platelet reactivity testing. Sixty eligible patients will be randomized in a 2:1 ratio to vildagliptin/metformin or metformin only treatment, for a 3-month duration treatment. Blood sampling for the proposed investigations will be taken at enrollment and immediately after completion of the study period. DISCUSSION: Demonstrating antiatherothrombotic properties of dipeptidyl peptidase-4 inhibitors on proven markers is of substantial clinical significance. Coupled with their proven good safety profile these findings could translate into a significant clinical benefit.

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Year:  2012        PMID: 22672501      PMCID: PMC3403890          DOI: 10.1186/1475-2840-11-60

Source DB:  PubMed          Journal:  Cardiovasc Diabetol        ISSN: 1475-2840            Impact factor:   9.951


  31 in total

1.  Using clinical guidelines designed for older adults with diabetes mellitus and complex health status.

Authors:  Samuel C Durso
Journal:  JAMA       Date:  2006-04-26       Impact factor: 56.272

2.  American Association of Clinical Endocrinologists Medical Guidelines for Clinical Practice for developing a diabetes mellitus comprehensive care plan.

Authors:  Yehuda Handelsman; Jeffrey I Mechanick; Lawrence Blonde; George Grunberger; Zachary T Bloomgarden; George A Bray; Samuel Dagogo-Jack; Jaime A Davidson; Daniel Einhorn; Om Ganda; Alan J Garber; Irl B Hirsch; Edward S Horton; Faramarz Ismail-Beigi; Paul S Jellinger; Kenneth L Jones; Lois Jovanovič; Harold Lebovitz; Philip Levy; Etie S Moghissi; Eric A Orzeck; Aaron I Vinik; Kathleen L Wyne
Journal:  Endocr Pract       Date:  2011 Mar-Apr       Impact factor: 3.443

3.  Adiposopathy is "sick fat" a cardiovascular disease?

Authors:  Harold E Bays
Journal:  J Am Coll Cardiol       Date:  2011-06-21       Impact factor: 24.094

4.  Increased levels of platelet activation markers are positively associated with carotid wall thickness and other atherosclerotic risk factors in obese patients.

Authors:  Éva Csongrádi; Béla Nagy; Tibor Fulop; Zsuzsa Varga; Zsolt Karányi; Mária T Magyar; László Oláh; Mária Papp; Andrea Facskó; János Kappelmayer; György Paragh; Miklós Káplár
Journal:  Thromb Haemost       Date:  2011-08-25       Impact factor: 5.249

5.  Statins and cardiovascular diseases: the multiple effects of lipid-lowering therapy by statins.

Authors:  U Rauch; J I Osende; J H Chesebro; V Fuster; D A Vorchheimer; K Harris; P Harris; D A Sandler; J T Fallon; S Jayaraman; J J Badimon
Journal:  Atherosclerosis       Date:  2000-11       Impact factor: 5.162

6.  Effects of one year treatment of vildagliptin added to pioglitazone or glimepiride in poorly controlled type 2 diabetic patients.

Authors:  G Derosa; P Maffioli; I Ferrari; R Mereu; P D Ragonesi; F Querci; I G Franzetti; G Gadaleta; L Ciccarelli; M N Piccinni; A D'Angelo; S A T Salvadeo
Journal:  Horm Metab Res       Date:  2010-06-17       Impact factor: 2.936

7.  Pleiotropic effects of statins in atherosclerosis and diabetes.

Authors:  S Bellosta; N Ferri; L Arnaboldi; F Bernini; R Paoletti; A Corsini
Journal:  Diabetes Care       Date:  2000-04       Impact factor: 19.112

8.  Metalloproteases 2 and 9, Lp-PLA(2) and lipoprotein profile in coronary patients.

Authors:  Maria Luz Muzzio; Veronica Miksztowicz; Fernando Brites; Daniel Aguilar; Esteban Martin Repetto; Regina Wikinski; Marcelo Tavella; Laura Schreier; Gabriela Alicia Berg
Journal:  Arch Med Res       Date:  2009-01       Impact factor: 2.235

9.  Matrix metalloproteinases and inflammatory markers in coronary artery ectasia: their relationship to severity of coronary artery ectasia.

Authors:  Abdullah Dogan; Nurullah Tuzun; Yasin Turker; Selahattin Akcay; Selcuk Kaya; Mehmet Ozaydin
Journal:  Coron Artery Dis       Date:  2008-12       Impact factor: 1.439

10.  Cardiovascular safety with linagliptin in patients with type 2 diabetes mellitus: a pre-specified, prospective, and adjudicated meta-analysis of a phase 3 programme.

Authors:  Odd Erik Johansen; Dietmar Neubacher; Maximilian von Eynatten; Sanjay Patel; Hans-Juergen Woerle
Journal:  Cardiovasc Diabetol       Date:  2012-01-10       Impact factor: 9.951

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  9 in total

1.  Effects of dapagliflozin vs vildagliptin on cardiometabolic parameters in diabetic patients with coronary artery disease: a randomised study.

Authors:  Arintaya Phrommintikul; Wanwarang Wongcharoen; Sirinart Kumfu; Thidarat Jaiwongkam; Siriluck Gunaparn; Siriporn Chattipakorn; Nipon Chattipakorn
Journal:  Br J Clin Pharmacol       Date:  2019-04-13       Impact factor: 4.335

2.  The addition of vildagliptin to metformin prevents the elevation of interleukin 1ß in patients with type 2 diabetes and coronary artery disease: a prospective, randomized, open-label study.

Authors:  Arwa Younis; Dana Eskenazi; Ronen Goldkorn; Jonathan Leor; Nili Naftali-Shani; Enrique Z Fisman; Alexander Tenenbaum; Ilan Goldenberg; Robert Klempfner
Journal:  Cardiovasc Diabetol       Date:  2017-05-22       Impact factor: 9.951

Review 3.  Cardiovascular effects of gliptins.

Authors:  André J Scheen
Journal:  Nat Rev Cardiol       Date:  2013-01-08       Impact factor: 32.419

Review 4.  Cardiovascular safety profile of currently available diabetic drugs.

Authors:  Komola Azimova; Zinnia San Juan; Debabrata Mukherjee
Journal:  Ochsner J       Date:  2014

5.  Change in levels of C-reactive protein (CRP) and serum cortisol in morbidly obese patients after laparoscopic sleeve gastrectomy.

Authors:  Jaime Ruiz-Tovar; Inmaculada Oller; Isabel Galindo; Carolina Llavero; Antonio Arroyo; Alicia Calero; María Diez; Lorea Zubiaga; Rafael Calpena
Journal:  Obes Surg       Date:  2013-06       Impact factor: 4.129

6.  Liquiritin attenuates advanced glycation end products-induced endothelial dysfunction via RAGE/NF-κB pathway in human umbilical vein endothelial cells.

Authors:  Xiaoyi Zhang; Yu Song; Xiaolin Han; Liang Feng; Rushang Wang; Minghua Zhang; Maomao Zhu; Xiaobin Jia; Shaoying Hu
Journal:  Mol Cell Biochem       Date:  2012-11-15       Impact factor: 3.396

7.  Adiponectin and IL-6: Mediators of inflammation in progression of healthy to type 2 diabetes in Indian population.

Authors:  Smitha Upadhyaya; Vinitha Kadamkode; Rafi Mahammed; Chandraprabha Doraiswami; Gautam Banerjee
Journal:  Adipocyte       Date:  2013-10-08       Impact factor: 4.534

8.  Association of metformin with lower atrial fibrillation risk among patients with type 2 diabetes mellitus: a population-based dynamic cohort and in vitro studies.

Authors:  Shang-Hung Chang; Lung-Sheng Wu; Meng-Jiun Chiou; Jia-Rou Liu; Kuang-Hui Yu; Chang-Fu Kuo; Ming-Shien Wen; Wei-Jan Chen; Yung-Hsin Yeh; Lai-Chu See
Journal:  Cardiovasc Diabetol       Date:  2014-08-10       Impact factor: 9.951

Review 9.  Hypoglycemic agents and potential anti-inflammatory activity.

Authors:  Vishal Kothari; John A Galdo; Suresh T Mathews
Journal:  J Inflamm Res       Date:  2016-04-11
  9 in total

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