Literature DB >> 22654150

SYNTHESIS OF N-SUBSTITUTED CARBONYLAMINO-1,2,3,6-TETRAHYDROPYRIDINES AS POTENTIAL ANTI-INFLAMMATORY AGENTS.

Mohammad A Ghaffari1, Tiffany W Ardley, Madhavi Gangapuram, Kinfe K Redda.   

Abstract

Several N-substituted carbonyl/sulfonylamino-1,2,3,6-tetrahydropyridines (5a-i and 9a, b) were synthesized via sodium borohydride reduction of the corresponding N-substitutedimino-pyridinium ylides (4a-i and 8a, b) in absolute ethanol.

Entities:  

Year:  2011        PMID： 22654150      PMCID： PMC3361725          DOI： 10.1080/00397911.2010.515335

Source DB:  PubMed          Journal:  Synth Commun        ISSN： 0039-7911            Impact factor:   2.007


  9 in total

1.  Synthesis and anti-inflammatory activities of N-benzoylamino-1,2,3,6-tetrahydropyridine analogs.

Authors:  B Mochona; T Wilson; K Redda
Journal:  Drugs Exp Clin Res       Date:  2003

2.  Synthesis and anti-inflammatory activities of some N-[pyridyl(phenyl)carbonylamino]-tert-butyl/phenyl-1,2,3,6- tetrahydropyridines.

Authors:  K K Redda; K N Rao; A S Heiman; F Y Onayemi; J B Clark
Journal:  Chem Pharm Bull (Tokyo)       Date:  1991-03       Impact factor: 1.645

3.  Aspirin selectively inhibits prostaglandin production in human platelets.

Authors:  J B Smith; A L Willis
Journal:  Nat New Biol       Date:  1971-06-23

4.  Inhibition of prostaglandin synthesis as a mechanism of action for aspirin-like drugs.

Authors:  J R Vane
Journal:  Nat New Biol       Date:  1971-06-23

Review 5.  The chemistry and pharmacology of tetrahydropyridines.

Authors:  N N Mateeva; L L Winfield; K K Redda
Journal:  Curr Med Chem       Date:  2005       Impact factor: 4.530

6.  Syntheses of N-substituted 2(3,4)-pyridylcarboxylic acid hydrazides with analgesic and antiinflammatory activity.

Authors:  K Redda; L A Corleto; E E Knaus
Journal:  J Med Chem       Date:  1979-09       Impact factor: 7.446

7.  Conformational analysis and molecular properties of N-(substituted phenyl-carbonylamino)-4-(1-hydroxymethylphenyl)-1,2,3,6-tetrahydropyridines.

Authors:  Cosmas O Okoroa; Tiffany L Wilsonb; Kinfe K Redda
Journal:  Curr Med Chem       Date:  2003-02       Impact factor: 4.530

8.  Inhibitory effects of N-(substituted benzoylamino)-4-ethyl-1,2,3,6-tetrahydropyridines on nitric oxide generation in stimulated raw 264.7 macrophages.

Authors:  K Yoon; K Soliman; K Redda
Journal:  Drugs Exp Clin Res       Date:  2002

9.  Synthesis and pharmacological evaluation of some N-[pyridyl(phenyl)carbonylamino]methyl-1,2,3,6-tetrahydropyrid ines.

Authors:  K K Redda; K N Rao; A S Heiman; H Melles
Journal:  J Pharm Sci       Date:  1992-05       Impact factor: 3.534
  9 in total
  1 in total

1.  Design, Synthesis and Evaluation of Novel N-Substituted-[Benzoylamino]-5-Ethyl-1,2,3,6-Tetrahydropyridines as Potential Anti-Cancer Agents.

Authors:  Elizabeth D Henderson; Madhavi Gangapuram; Suresh Kumar Vk Eyunni; Kinfe K Redda; Tiffany Wilson-Ardley
Journal:  Madridge J Pharm Res       Date:  2019-03-04
  1 in total

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