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17 in total

1. Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 Inhibitors.

Authors: Yonghua Lei; Tianhan Hu; Xingsen Wu; Yue Wu; Qichao Bao; Lianshan Zhang; Hua Xia; Haopeng Sun; Qidong You; Xiaojin Zhang
Journal: ACS Med Chem Lett Date: 2015-11-09 Impact factor: 4.345

2. Reporter ligand NMR screening method for 2-oxoglutarate oxygenase inhibitors.

Authors: Ivanhoe K H Leung; Marina Demetriades; Adam P Hardy; Clarisse Lejeune; Tristan J Smart; Andrea Szöllössi; Akane Kawamura; Christopher J Schofield; Timothy D W Claridge
Journal: J Med Chem Date: 2013-01-04 Impact factor: 7.446

3. Reversible linkage of two distinct small molecule inhibitors of Myc generates a dimeric inhibitor with improved potency that is active in myc over-expressing cancer cell lines.

Authors: Jutta Wanner; Darlene Romashko; Douglas S Werner; Earl W May; Yue Peng; Ryan Schulz; Kenneth W Foreman; Suzanne Russo; Lee D Arnold; Maneesh Pingle; Donald E Bergstrom; Francis Barany; Stuart Thomson
Journal: PLoS One Date: 2015-04-15 Impact factor: 3.240

4. trans-Symmetric Dynamic Covalent Systems: Connected Transamination and Transimination Reactions.

Authors: Fredrik Schaufelberger; Lei Hu; Olof Ramström
Journal: Chemistry Date: 2015-06-03 Impact factor: 5.236

5. Dynamic covalent organocatalysts discovered from catalytic systems through rapid deconvolution screening.

Authors: Fredrik Schaufelberger; Olof Ramström
Journal: Chemistry Date: 2015-07-14 Impact factor: 5.236

6. Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry.

Authors: Milon Mondal; Nedyalka Radeva; Hugo Fanlo-Virgós; Sijbren Otto; Gerhard Klebe; Anna K H Hirsch
Journal: Angew Chem Int Ed Engl Date: 2016-07-12 Impact factor: 15.336

Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors.

1. Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 Inhibitors.

2. Reporter ligand NMR screening method for 2-oxoglutarate oxygenase inhibitors.

3. Reversible linkage of two distinct small molecule inhibitors of Myc generates a dimeric inhibitor with improved potency that is active in myc over-expressing cancer cell lines.

4. trans-Symmetric Dynamic Covalent Systems: Connected Transamination and Transimination Reactions.

5. Dynamic covalent organocatalysts discovered from catalytic systems through rapid deconvolution screening.

6. Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry.

7. Design, preparation, and selection of DNA-encoded dynamic libraries.

8. NMR-filtered virtual screening leads to non-metal chelating metallo-β-lactamase inhibitors.

Review 9. Protein-Directed Dynamic Combinatorial Chemistry: A Guide to Protein Ligand and Inhibitor Discovery.

10. Dynamic Covalent Chemistry of Aldehyde Enamines: Bi^III - and Sc^III -Catalysis of Amine-Enamine Exchange.