Literature DB >> 22517399

A safety run-in and randomized phase 2 study of cilengitide combined with chemoradiation for newly diagnosed glioblastoma (NABTT 0306).

L Burt Nabors1, Thomas Mikkelsen, Monika E Hegi, Xiaubu Ye, Tracy Batchelor, Glenn Lesser, David Peereboom, Myrna R Rosenfeld, Jeff Olsen, Steve Brem, Joy D Fisher, Stuart A Grossman.   

Abstract

BACKGROUND: Cilengitide is a selective integrin inhibitor that is well tolerated and has demonstrated biologic activity in patients with recurrent malignant glioma. The primary objectives of this randomized phase 2 trial were to determine the safety and efficacy of cilengitide when combined with radiation and temozolomide for patients with newly diagnosed glioblastoma multiforme and to select a dose for comparative clinical testing.
METHODS: In total, 112 patients were accrued. Eighteen patients received standard radiation and temozolomide with cilengitide in a safety run-in phase followed by a randomized phase 2 trial with 94 patients assigned to either a 500 mg dose group or 2000 mg dose group. The trial was designed to estimate overall survival benefit compared with a New Approaches to Brain Tumor Therapy (NABTT) Consortium internal historic control and data from the published European Organization for Research and Treatment of Cancer (EORTC) trial EORTC 26981.
RESULTS: Cilengitide at all doses studied was well tolerated with radiation and temozolomide. The median survival was 19.7 months for all patients, 17.4 months for the patients in the 500 mg dose group, 20.8 months for patients in the 2000 mg dose group, 30 months for patients who had methylated O6-methylguanine-DNA methyltransferase (MGMT) status, and 17.4 months for patients who had unmethylated MGMT status. For patients aged ≤70 years, the median survival and survival at 24 months was superior to what was observed in the EORTC trial (20.7 months vs 14.6 months and 41% vs 27%, respectively; P = .008).
CONCLUSIONS: Cilengitide was well tolerated when combined with standard chemoradiation and may improve survival for patients newly diagnosed with glioblastoma multiforme regardless of MGMT methylation status. The authors concluded that, from an efficacy and safety standpoint, future trials of this agent in this population should use the 2000 mg dose.
Copyright © 2012 American Cancer Society.

Entities:  

Mesh:

Substances:

Year:  2012        PMID: 22517399      PMCID: PMC3423527          DOI: 10.1002/cncr.27585

Source DB:  PubMed          Journal:  Cancer        ISSN: 0008-543X            Impact factor:   6.860


  14 in total

1.  alphav beta 3 and alphav beta 5 integrin antagonists inhibit angiogenesis in vitro.

Authors:  Riccardo E Nisato; Jean-Christophe Tille; Alfred Jonczyk; Simon L Goodman; Michael S Pepper
Journal:  Angiogenesis       Date:  2003       Impact factor: 9.596

2.  Effect of the angiogenesis inhibitor Cilengitide (EMD 121974) on glioblastoma growth in nude mice.

Authors:  Shinya Yamada; Xing-Yao Bu; Vazgen Khankaldyyan; Ignacio Gonzales-Gomez; J Gordon McComb; Walter E Laug
Journal:  Neurosurgery       Date:  2006-12       Impact factor: 4.654

3.  Preferential susceptibility of brain tumors to the antiangiogenic effects of an alpha(v) integrin antagonist.

Authors:  T J MacDonald; T Taga; H Shimada; P Tabrizi; B V Zlokovic; D A Cheresh; W E Laug
Journal:  Neurosurgery       Date:  2001-01       Impact factor: 4.654

4.  Phase II study of bevacizumab plus temozolomide during and after radiation therapy for patients with newly diagnosed glioblastoma multiforme.

Authors:  Albert Lai; Anh Tran; Phioanh L Nghiemphu; Whitney B Pope; Orestes E Solis; Michael Selch; Emese Filka; William H Yong; Paul S Mischel; Linda M Liau; Surasak Phuphanich; Keith Black; Scott Peak; Richard M Green; Cynthia E Spier; Tatjana Kolevska; Jonathan Polikoff; Louis Fehrenbacher; Robert Elashoff; Timothy Cloughesy
Journal:  J Clin Oncol       Date:  2010-12-06       Impact factor: 44.544

5.  Human malignant glioma therapy using anti-alpha(v)beta3 integrin agents.

Authors:  S Chatterjee; A Matsumura; J Schradermeier; G Y Gillespie
Journal:  J Neurooncol       Date:  2000       Impact factor: 4.130

6.  Nanomolar small molecule inhibitors for alphav(beta)6, alphav(beta)5, and alphav(beta)3 integrins.

Authors:  Simon L Goodman; Günter Hölzemann; Gábor A G Sulyok; Horst Kessler
Journal:  J Med Chem       Date:  2002-02-28       Impact factor: 7.446

7.  Radiotherapy plus concomitant and adjuvant temozolomide for glioblastoma.

Authors:  Roger Stupp; Warren P Mason; Martin J van den Bent; Michael Weller; Barbara Fisher; Martin J B Taphoorn; Karl Belanger; Alba A Brandes; Christine Marosi; Ulrich Bogdahn; Jürgen Curschmann; Robert C Janzer; Samuel K Ludwin; Thierry Gorlia; Anouk Allgeier; Denis Lacombe; J Gregory Cairncross; Elizabeth Eisenhauer; René O Mirimanoff
Journal:  N Engl J Med       Date:  2005-03-10       Impact factor: 91.245

8.  Phase I and correlative biology study of cilengitide in patients with recurrent malignant glioma.

Authors:  L Burt Nabors; Tom Mikkelsen; Steven S Rosenfeld; Fred Hochberg; Narasimha S Akella; Joy D Fisher; Gretchen A Cloud; Yu Zhang; Kathryn Carson; Sabine M Wittemer; A Dimitrios Colevas; Stuart A Grossman
Journal:  J Clin Oncol       Date:  2007-05-01       Impact factor: 44.544

9.  Kinetic analysis of integrin-dependent cell adhesion on vitronectin--the inhibitory potential of plasminogen activator inhibitor-1 and RGD peptides.

Authors:  M Germer; S M Kanse; T Kirkegaard; L Kjøller; B Felding-Habermann; S Goodman; K T Preissner
Journal:  Eur J Biochem       Date:  1998-05-01

10.  Validation of real-time methylation-specific PCR to determine O6-methylguanine-DNA methyltransferase gene promoter methylation in glioma.

Authors:  Ilse Vlassenbroeck; Stéphane Califice; Annie-Claire Diserens; Eugenia Migliavacca; Josef Straub; Ivano Di Stefano; Fabrice Moreau; Marie-France Hamou; Isabelle Renard; Mauro Delorenzi; Bruno Flamion; James DiGuiseppi; Katja Bierau; Monika E Hegi
Journal:  J Mol Diagn       Date:  2008-06-13       Impact factor: 5.568

View more
  45 in total

1.  MGMT promoter methylation is not correlated with integrin expression in malignant gliomas: clarifying recent clinical trial results.

Authors:  Oliver Schnell; Valerie Albrecht; David Pfirrmann; Sabina Eigenbrod; Bjarne Krebs; Alexander Romagna; Sebastian Siller; Armin Giese; Jörg-Christian Tonn; Christian Schichor
Journal:  Med Oncol       Date:  2018-06-07       Impact factor: 3.064

2.  End of the road: confounding results of the CORE trial terminate the arduous journey of cilengitide for glioblastoma.

Authors:  Warren P Mason
Journal:  Neuro Oncol       Date:  2015-02-13       Impact factor: 12.300

3.  To randomize, or not to randomize, that is the question: using data from prior clinical trials to guide future designs.

Authors:  Alyssa M Vanderbeek; Steffen Ventz; Rifaquat Rahman; Geoffrey Fell; Timothy F Cloughesy; Patrick Y Wen; Lorenzo Trippa; Brian M Alexander
Journal:  Neuro Oncol       Date:  2019-10-09       Impact factor: 12.300

4.  Phase II study of cilengitide in the treatment of refractory or relapsed high-grade gliomas in children: a report from the Children's Oncology Group.

Authors:  Tobey J MacDonald; Gilbert Vezina; Clinton F Stewart; David Turner; Christopher R Pierson; Lu Chen; Ian F Pollack; Amar Gajjar; Mark W Kieran
Journal:  Neuro Oncol       Date:  2013-09-05       Impact factor: 12.300

5.  The effect of cilengitide in combination with irradiation and chemotherapy in head and neck squamous cell carcinoma cell lines.

Authors:  G Heiduschka; C Lill; S Schneider; R Seemann; G Kornek; R Schmid; U Kotowski; D Thurnher
Journal:  Strahlenther Onkol       Date:  2014-02-21       Impact factor: 3.621

6.  Antitumor activity of 7-O-succinyl macrolactin A tromethamine salt in the mouse glioma model.

Authors:  Jun Jin; Suh Hee Choi; Jung Eun Lee; Jin-Deok Joo; Jung Ho Han; Su-Young Park; Chae-Yong Kim
Journal:  Oncol Lett       Date:  2017-03-27       Impact factor: 2.967

7.  Tumor cohesion and glioblastoma cell dispersal.

Authors:  Ramsey A Foty
Journal:  Future Oncol       Date:  2013-08       Impact factor: 3.404

8.  The integrin inhibitor cilengitide enhances the anti-glioma efficacy of vasculostatin-expressing oncolytic virus.

Authors:  K Fujii; K Kurozumi; T Ichikawa; M Onishi; Y Shimazu; J Ishida; E A Chiocca; B Kaur; I Date
Journal:  Cancer Gene Ther       Date:  2013-07-05       Impact factor: 5.987

9.  Two cilengitide regimens in combination with standard treatment for patients with newly diagnosed glioblastoma and unmethylated MGMT gene promoter: results of the open-label, controlled, randomized phase II CORE study.

Authors:  L Burt Nabors; Karen L Fink; Tom Mikkelsen; Danica Grujicic; Rafal Tarnawski; Do Hyun Nam; Maria Mazurkiewicz; Michael Salacz; Lynn Ashby; Vittorina Zagonel; Roberta Depenni; James R Perry; Christine Hicking; Martin Picard; Monika E Hegi; Benoit Lhermitte; David A Reardon
Journal:  Neuro Oncol       Date:  2015-03-11       Impact factor: 12.300

Review 10.  Tumor stroma as targets for cancer therapy.

Authors:  Jing Zhang; Jinsong Liu
Journal:  Pharmacol Ther       Date:  2012-10-12       Impact factor: 12.310

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.