Literature DB >> 22506260

Review of boceprevir and telaprevir for the treatment of chronic hepatitis C.

Kyle John Wilby1, Nilufar Partovi, Jo-Ann E Ford, Erica Greanya, Eric M Yoshida.   

Abstract

OBJECTIVE: To summarize and evaluate the published literature pertaining to boceprevir and telaprevir, and to provide clinicians with suggestions for use in patients with chronic hepatitis C infection.
METHODS: A standardized search strategy was performed using the MEDLINE, EMBASE, Google Scholar and International Pharmaceuticals Abstracts databases using the search terms "boceprevir", "telaprevir", "boceprevir and hepatitis C", and "telaprevir and hepatitis C". A manual search of references was performed to identify articles missed by the electronic search. Studies were included in the review if they assessed either boceprevir or telaprevir in comparison with standard of care in chronic hepatitis C patients.
RESULTS: The studies identified assessed boceprevir and telaprevir in genotype-1 hepatitis C patients. In both treatment-naive and treatment-experienced patients, sustained virological response rates were achieved more often with boceprevir or telaprevir in combination with pegylated interferon and ribavirin compared with pegylated interferon and ribavirin alone. Both medications were well tolerated, with anemia presenting as the most treatment-limiting adverse effect.
CONCLUSIONS: Boceprevir and telaprevir will revolutionize the management of hepatitis C genotype 1 patients and will most likely decrease the burden of end-stage disease worldwide. However, current clinical limitations include establishing appropriate and cost-effective treatment durations, and use in special populations such as transplant patients and patients coinfected with HIV. Future research will need to clarify these clinical obstacles to clearly define the role of these agents in hepatitis C management.

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Year:  2012        PMID: 22506260      PMCID: PMC3354889          DOI: 10.1155/2012/751057

Source DB:  PubMed          Journal:  Can J Gastroenterol        ISSN: 0835-7900            Impact factor:   3.522


  26 in total

1.  Telaprevir is effective given every 8 or 12 hours with ribavirin and peginterferon alfa-2a or -2b to patients with chronic hepatitis C.

Authors:  Patrick Marcellin; Xavier Forns; Tobias Goeser; Peter Ferenci; Frederik Nevens; Giampiero Carosi; Joost P Drenth; Lawrence Serfaty; Koen De Backer; Rolf Van Heeswijk; Donghan Luo; Gaston Picchio; Maria Beumont
Journal:  Gastroenterology       Date:  2010-10-26       Impact factor: 22.682

2.  Direct-acting antiviral medications for chronic hepatitis C virus infection.

Authors:  Alison B Jazwinski; Andrew J Muir
Journal:  Gastroenterol Hepatol (N Y)       Date:  2011-03

3.  Telaprevir for previously treated chronic HCV infection.

Authors:  John G McHutchison; Michael P Manns; Andrew J Muir; Norah A Terrault; Ira M Jacobson; Nezam H Afdhal; E Jenny Heathcote; Stefan Zeuzem; Hendrik W Reesink; Jyotsna Garg; Mohammad Bsharat; Shelley George; Robert S Kauffman; Nathalie Adda; Adrian M Di Bisceglie
Journal:  N Engl J Med       Date:  2010-04-08       Impact factor: 91.245

4.  Peginterferon alfa-2b plus ribavirin compared with interferon alfa-2b plus ribavirin for initial treatment of chronic hepatitis C: a randomised trial.

Authors:  M P Manns; J G McHutchison; S C Gordon; V K Rustgi; M Shiffman; R Reindollar; Z D Goodman; K Koury; M Ling; J K Albrecht
Journal:  Lancet       Date:  2001-09-22       Impact factor: 79.321

5.  Efficacy of boceprevir, an NS3 protease inhibitor, in combination with peginterferon alfa-2b and ribavirin in treatment-naive patients with genotype 1 hepatitis C infection (SPRINT-1): an open-label, randomised, multicentre phase 2 trial.

Authors:  Paul Y Kwo; Eric J Lawitz; Jonathan McCone; Eugene R Schiff; John M Vierling; David Pound; Mitchell N Davis; Joseph S Galati; Stuart C Gordon; Natarajan Ravendhran; Lorenzo Rossaro; Frank H Anderson; Ira M Jacobson; Raymond Rubin; Kenneth Koury; Lisa D Pedicone; Clifford A Brass; Eirum Chaudhri; Janice K Albrecht
Journal:  Lancet       Date:  2010-08-06       Impact factor: 79.321

6.  Antiviral activity of telaprevir (VX-950) and peginterferon alfa-2a in patients with hepatitis C.

Authors:  Nicole Forestier; Hendrik W Reesink; Christine J Weegink; Lindsay McNair; Tara L Kieffer; Hui-May Chu; Susan Purdy; Peter L M Jansen; Stefan Zeuzem
Journal:  Hepatology       Date:  2007-09       Impact factor: 17.425

7.  Telaprevir with peginterferon and ribavirin for chronic HCV genotype 1 infection.

Authors:  John G McHutchison; Gregory T Everson; Stuart C Gordon; Ira M Jacobson; Mark Sulkowski; Robert Kauffman; Lindsay McNair; John Alam; Andrew J Muir
Journal:  N Engl J Med       Date:  2009-04-30       Impact factor: 91.245

8.  Telaprevir and peginterferon with or without ribavirin for chronic HCV infection.

Authors:  Christophe Hézode; Nicole Forestier; Geoffrey Dusheiko; Peter Ferenci; Stanislas Pol; Tobias Goeser; Jean-Pierre Bronowicki; Marc Bourlière; Shahin Gharakhanian; Leif Bengtsson; Lindsay McNair; Shelley George; Tara Kieffer; Ann Kwong; Robert S Kauffman; John Alam; Jean-Michel Pawlotsky; Stefan Zeuzem
Journal:  N Engl J Med       Date:  2009-04-30       Impact factor: 91.245

9.  Peginterferon-alpha2a and ribavirin combination therapy in chronic hepatitis C: a randomized study of treatment duration and ribavirin dose.

Authors:  Stephanos J Hadziyannis; Hoel Sette; Timothy R Morgan; Vijayan Balan; Moises Diago; Patrick Marcellin; Giuliano Ramadori; Henry Bodenheimer; David Bernstein; Mario Rizzetto; Stefan Zeuzem; Paul J Pockros; Amy Lin; Andrew M Ackrill
Journal:  Ann Intern Med       Date:  2004-03-02       Impact factor: 25.391

10.  Re-treatment with peginterferon alfa-2a and ribavirin in patients with chronic hepatitis C who have relapsed or not responded to a first course of pegylated interferon-based therapy.

Authors:  E M Yoshida; M Sherman; V G Bain; C L Cooper; M Deschênes; P J Marotta; S S Lee; M Krajden; H Witt-Sullivan; R J Bailey; C Usaty; K Peltekian
Journal:  Can J Gastroenterol       Date:  2009-03       Impact factor: 3.522

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  18 in total

1.  HIV and HCV Medications in End-Stage Renal Disease.

Authors:  Keiko I Greenberg; Mark A Perazella; Mohamed G Atta
Journal:  Semin Dial       Date:  2015-04-06       Impact factor: 3.455

2.  Advanced Hepatitis C Virus Replication PDE Models within a Realistic Intracellular Geometric Environment.

Authors:  Markus M Knodel; Paul Targett-Adams; Alfio Grillo; Eva Herrmann; Gabriel Wittum
Journal:  Int J Environ Res Public Health       Date:  2019-02-12       Impact factor: 3.390

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5.  3D Spatially Resolved Models of the Intracellular Dynamics of the Hepatitis C Genome Replication Cycle.

Authors:  Markus M Knodel; Sebastian Reiter; Paul Targett-Adams; Alfio Grillo; Eva Herrmann; Gabriel Wittum
Journal:  Viruses       Date:  2017-09-30       Impact factor: 5.048

Review 6.  Taming a beast: lessons from the domestication of hepatitis C virus.

Authors:  Joseph M Luna; Mohsan Saeed; Charles M Rice
Journal:  Curr Opin Virol       Date:  2019-03-12       Impact factor: 7.090

Review 7.  Unboxing the molecular modalities of mutagens in cancer.

Authors:  Smita Kumari; Sudhanshu Sharma; Dia Advani; Akanksha Khosla; Pravir Kumar; Rashmi K Ambasta
Journal:  Environ Sci Pollut Res Int       Date:  2021-10-05       Impact factor: 5.190

8.  Follow-up testing for hepatitis C virus infection: an analysis of Massachusetts surveillance data, 2007-2010.

Authors:  Kerri Barton; Dan Church; Shauna Onofrey; Noelle Cocoros; Alfred DeMaria
Journal:  Public Health Rep       Date:  2014 Sep-Oct       Impact factor: 2.792

9.  Basic concepts in population modeling, simulation, and model-based drug development: part 3-introduction to pharmacodynamic modeling methods.

Authors:  R N Upton; D R Mould
Journal:  CPT Pharmacometrics Syst Pharmacol       Date:  2014-01-02

10.  Identification of a resveratrol tetramer as a potent inhibitor of hepatitis C virus helicase.

Authors:  Sungjin Lee; Kee Dong Yoon; Myungeun Lee; Yoojin Cho; Gahee Choi; Hongje Jang; BeomSeok Kim; Da-Hee Jung; Jin-Gyo Oh; Geon-Woo Kim; Jong-Won Oh; Yong-Joo Jeong; Ho Jeong Kwon; Soo Kyung Bae; Dal-Hee Min; Marc P Windisch; Tae-Hwe Heo; Choongho Lee
Journal:  Br J Pharmacol       Date:  2015-11-25       Impact factor: 8.739

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