Literature DB >> 22495744

Transmembrane estrogen receptor GPR30 is more frequently expressed in malignant than benign ovarian endometriotic cysts and correlates with MMP-9 expression.

Li Long1, Yi Cao, Liang-Dan Tang.   

Abstract

OBJECTIVE: Molecular studies supporting the idea of malignant transformation of endometriosis are sparse and not well substantiated. The aims of this study were to detect expression levels of the novel estrogen-responsive receptor G protein-coupled estrogen receptor 1 GPER, also termed GPR30, and to determine its correlation with matrix metalloproteinase-9 (MMP-9) in benign and malignant ovarian endometriotic cysts and to explore the significance of GPR30.
METHODS: Immunohistochemical staining with the streptavidin-peroxidase method was conducted to determine the expression of GPR30 and MMP-9 in 24 cases of endometriosis-associated ovarian carcinoma (EAOC) and 32 specimens of ovarian endometriosis without malignant transformation. Reverse transcriptase polymerase chain reaction was performed to determine messenger RNA expression of GPR30 and MMP-9 in benign and malignant ovarian endometriotic cysts. We also investigated their associations with known clinic pathological parameters and the interrelationship between the expressions of the 2 proteins.
RESULTS: The positive staining ratio of GPR30 was 95.8% (23/24) in EAOC cases, and the HScore was 268; whereas the positive ratio was 25% (8/32) in benign endometriotic cysts, and the Hscore was 95. Matrix metalloproteinase-9 was expressed in all 24 EAOC cases and 87.5% (28/32) of the benign samples, and the Hscores were 280 and 260, respectively (P > 0.05). The receptor GPR30 was significantly higher in EAOCs than in benign endometriotic cysts (P < 0.05). The expression of GPR30 messenger RNA was also significantly higher in malignant ovarian endometriotic cysts than in the benign group. The receptor GPR30 was positively related to tumor size, tumor stage, and lymph node metastasis. A positive relationship between GPR30 and MMP-9 was found (P = 0.002).
CONCLUSIONS: The results suggest that the abnormal expression of GPR30 may be involved in malignant transformation, invasion, and metastasis of EAOCs. Testing of GPR30 expression levels may present both diagnostic and therapeutic options for the treatment of ovarian malignancies.

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Year:  2012        PMID: 22495744     DOI: 10.1097/IGC.0b013e318247323d

Source DB:  PubMed          Journal:  Int J Gynecol Cancer        ISSN: 1048-891X            Impact factor:   3.437


  9 in total

Review 1.  Estrogen signaling crosstalk: Implications for endocrine resistance in ovarian cancer.

Authors:  Jennifer R Ribeiro; Richard N Freiman
Journal:  J Steroid Biochem Mol Biol       Date:  2014-02-22       Impact factor: 4.292

2.  Activation of G protein coupled estrogen receptor (GPER) promotes the migration of renal cell carcinoma via the PI3K/AKT/MMP-9 signals.

Authors:  Bao-Zhang Guan; Rui-Ling Yan; Jian-Wei Huang; Fo-Lan Li; Ying-Xue Zhong; Yu Chen; Fan-Na Liu; Bo Hu; Si-Bo Huang; Liang-Hong Yin
Journal:  Cell Adh Migr       Date:  2018-01-29       Impact factor: 3.405

3.  Baicalein, unlike 4-hydroxytamoxifen but similar to G15, suppresses 17β-estradiol-induced cell invasion, and matrix metalloproteinase-9 expression and activation in MCF-7 human breast cancer cells.

Authors:  Yan Chen; Duan-Yang Hong; Jing Wang; Jun Ling-Hu; Yan-Yan Zhang; Di Pan; Yi-Ni Xu; Ling Tao; Hong Luo; Xiang-Chun Shen
Journal:  Oncol Lett       Date:  2017-06-02       Impact factor: 2.967

4.  Correlation between matrix metalloproteinase-9 and endometriosis.

Authors:  Haiping Liu; Jianye Wang; Haiyu Wang; Ning Tang; Yunfei Li; Yan Zhang; Tianyu Hao
Journal:  Int J Clin Exp Pathol       Date:  2015-10-01

Review 5.  International Union of Basic and Clinical Pharmacology. XCVII. G Protein-Coupled Estrogen Receptor and Its Pharmacologic Modulators.

Authors:  Eric R Prossnitz; Jeffrey B Arterburn
Journal:  Pharmacol Rev       Date:  2015-07       Impact factor: 25.468

6.  Decreased Expression of GPER1 Gene and Protein in Goiter.

Authors:  Raquel Weber; Ana Paula Santin Bertoni; Laura Walter Bessestil; Ilma Simoni Brum; Tania Weber Furlanetto
Journal:  Int J Endocrinol       Date:  2015-03-12       Impact factor: 3.257

Review 7.  Local estrogen formation and its regulation in endometriosis.

Authors:  Taisuke Mori; Fumitake Ito; Akemi Koshiba; Hisashi Kataoka; Osamu Takaoka; Hiroyuki Okimura; Khaleque N Khan; Jo Kitawaki
Journal:  Reprod Med Biol       Date:  2019-06-18

8.  The Expression of GPR30 in Iron-Overloaded Atypical Ovarian Epithelium and Ectopic Endometrium Is Closely Correlated with Transferrin Receptor and Pi3K.

Authors:  Li Long; Zhaoning Duan
Journal:  Biomed Res Int       Date:  2022-09-12       Impact factor: 3.246

Review 9.  The Role of Endocrine G Protein-Coupled Receptors in Ovarian Cancer Progression.

Authors:  Qingyu Zhang; Nadine Ellen Madden; Alice Sze Tsai Wong; Billy Kwok Chong Chow; Leo Tsz On Lee
Journal:  Front Endocrinol (Lausanne)       Date:  2017-04-07       Impact factor: 5.555

  9 in total

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