Literature DB >> 22492508

Bicyclic peptides with optimized ring size inhibit human plasma kallikrein and its orthologues while sparing paralogous proteases.

Vanessa Baeriswyl1, Helen Rapley, Lisa Pollaro, Catherine Stace, Dan Teufel, Edward Walker, Shiyu Chen, Greg Winter, John Tite, Christian Heinis.   

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Year:  2012        PMID： 22492508     DOI： 10.1002/cmdc.201200071

Source DB:  PubMed          Journal:  ChemMedChem        ISSN： 1860-7179            Impact factor:   3.466


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  13 in total

1.  Highly Constrained Bicyclic Scaffolds for the Discovery of Protease-Stable Peptides via mRNA Display.

Authors:  David E Hacker; Jan Hoinka; Emil S Iqbal; Teresa M Przytycka; Matthew C T Hartman
Journal:  ACS Chem Biol       Date:  2017-02-01       Impact factor: 5.100

2.  Development of Potent and Selective S. aureus Sortase A Inhibitors Based on Peptide Macrocycles.

Authors:  Inmaculada Rentero Rebollo; Shawna McCallin; Davide Bertoldo; José Manuel Entenza; Philippe Moreillon; Christian Heinis
Journal:  ACS Med Chem Lett       Date:  2016-04-14       Impact factor: 4.345

3.  Identification of target-binding peptide motifs by high-throughput sequencing of phage-selected peptides.

Authors:  Inmaculada Rentero Rebollo; Michal Sabisz; Vanessa Baeriswyl; Christian Heinis
Journal:  Nucleic Acids Res       Date:  2014-10-27       Impact factor: 16.971

4.  Small cyclic agonists of iron regulatory hormone hepcidin.

Authors:  Kristine Chua; Eileen Fung; Ewa D Micewicz; Tomas Ganz; Elizabeta Nemeth; Piotr Ruchala
Journal:  Bioorg Med Chem Lett       Date:  2015-03-12       Impact factor: 2.823

Review 5.  A Genetically Encoded, Phage-Displayed Cyclic-Peptide Library.

Authors:  Xiaoshan Shayna Wang; Peng-Hsun Chase Chen; J Trae Hampton; Jeffery M Tharp; Catrina A Reed; Sukant K Das; Duen-Shian Wang; Hamed S Hayatshahi; Yang Shen; Jin Liu; Wenshe Ray Liu
Journal:  Angew Chem Int Ed Engl       Date:  2019-09-09       Impact factor: 15.336

6.  Synthesis of a large library of macrocyclic peptides containing multiple and diverse N-alkylated residues.

Authors:  Jumpei Morimoto; Thomas Kodadek
Journal:  Mol Biosyst       Date:  2015-10

7.  Bridged Analogues for p53-Dependent Cancer Therapy Obtained by S-Alkylation.

Authors:  Ewa D Micewicz; Shantanu Sharma; Alan J Waring; Hai T Luong; William H McBride; Piotr Ruchala
Journal:  Int J Pept Res Ther       Date:  2015-08-19       Impact factor: 1.931

8.  Side-chain-to-tail cyclization of ribosomally derived peptides promoted by aryl and alkyl amino-functionalized unnatural amino acids.

Authors:  John R Frost; Zhijie Wu; Yick Chong Lam; Andrew E Owens; Rudi Fasan
Journal:  Org Biomol Chem       Date:  2016-04-11       Impact factor: 3.876

9.  Design of Specific Serine Protease Inhibitors Based on a Versatile Peptide Scaffold: Conversion of a Urokinase Inhibitor to a Plasma Kallikrein Inhibitor.

Authors:  Peng Xu; Mingming Xu; Longguang Jiang; Qinglan Yang; Zhipu Luo; Zbigniew Dauter; Mingdong Huang; Peter A Andreasen
Journal:  J Med Chem       Date:  2015-11-12       Impact factor: 7.446

10.  Genetically encoded libraries of nonstandard peptides.

Authors:  Takashi Kawakami; Hiroshi Murakami
Journal:  J Nucleic Acids       Date:  2012-10-14
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