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19 in total

1. Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.

Authors: Dilip K Tosh; Kenneth A Jacobson
Journal: Medchemcomm Date: 2013-12-17 Impact factor: 3.597

Review 2. A₃ Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.

Authors: Kenneth A Jacobson; Stefania Merighi; Katia Varani; Pier Andrea Borea; Stefania Baraldi; Mojgan Aghazadeh Tabrizi; Romeo Romagnoli; Pier Giovanni Baraldi; Antonella Ciancetta; Dilip K Tosh; Zhan-Guo Gao; Stefania Gessi
Journal: Med Res Rev Date: 2017-07-06 Impact factor: 12.944

3. N⁶-Substituted 5'-N-Methylcarbamoyl-4'-selenoadenosines as Potent and Selective A₃ Adenosine Receptor Agonists with Unusual Sugar Puckering and Nucleobase Orientation.

Authors: Jinha Yu; Long Xuan Zhao; Jongmi Park; Hyuk Woo Lee; Pramod K Sahu; Minghua Cui; Steven M Moss; Eva Hammes; Eugene Warnick; Zhan-Guo Gao; Minsoo Noh; Sun Choi; Hee-Chul Ahn; Jungwon Choi; Kenneth A Jacobson; Lak Shin Jeong
Journal: J Med Chem Date: 2017-04-19 Impact factor: 7.446

4. Machine Learning for Discovery of New ADORA Modulators.

Authors: Ana C Puhl; Zhan-Guo Gao; Kenneth A Jacobson; Sean Ekins
Journal: Front Pharmacol Date: 2022-06-22 Impact factor: 5.988

Review 5. Adenosine receptors as drug targets--what are the challenges?

Authors: Jiang-Fan Chen; Holger K Eltzschig; Bertil B Fredholm
Journal: Nat Rev Drug Discov Date: 2013-04 Impact factor: 84.694

6. Extended N(6) substitution of rigid C2-arylethynyl nucleosides for exploring the role of extracellular loops in ligand recognition at the A3 adenosine receptor.

Authors: Dilip K Tosh; Silvia Paoletta; Zhoumou Chen; Steven M Moss; Zhan-Guo Gao; Daniela Salvemini; Kenneth A Jacobson
Journal: Bioorg Med Chem Lett Date: 2014-06-11 Impact factor: 2.823

Review 7. Structure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.

Authors: Kenneth A Jacobson
Journal: J Med Chem Date: 2013-05-09 Impact factor: 7.446

Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications.

1. Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.

Review 2. A₃ Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.

3. N⁶-Substituted 5'-N-Methylcarbamoyl-4'-selenoadenosines as Potent and Selective A₃ Adenosine Receptor Agonists with Unusual Sugar Puckering and Nucleobase Orientation.

4. Machine Learning for Discovery of New ADORA Modulators.

Review 5. Adenosine receptors as drug targets--what are the challenges?

6. Extended N(6) substitution of rigid C2-arylethynyl nucleosides for exploring the role of extracellular loops in ligand recognition at the A3 adenosine receptor.

Review 7. Structure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.

8. Probing structure-activity relationship in β-arrestin2 recruitment of diversely substituted adenosine derivatives.

Review 9. Molecular Simulations and Drug Discovery of Adenosine Receptors.

10. Limits of ligand selectivity from docking to models: in silico screening for A(1) adenosine receptor antagonists.

Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications.

1. Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.

Review 2. A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.

3. N6-Substituted 5'-N-Methylcarbamoyl-4'-selenoadenosines as Potent and Selective A3 Adenosine Receptor Agonists with Unusual Sugar Puckering and Nucleobase Orientation.

4. Machine Learning for Discovery of New ADORA Modulators.

Review 5. Adenosine receptors as drug targets--what are the challenges?

6. Extended N(6) substitution of rigid C2-arylethynyl nucleosides for exploring the role of extracellular loops in ligand recognition at the A3 adenosine receptor.

Review 7. Structure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.

8. Probing structure-activity relationship in β-arrestin2 recruitment of diversely substituted adenosine derivatives.

Review 9. Molecular Simulations and Drug Discovery of Adenosine Receptors.

10. Limits of ligand selectivity from docking to models: in silico screening for A(1) adenosine receptor antagonists.

Review 2. A₃ Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.

3. N⁶-Substituted 5'-N-Methylcarbamoyl-4'-selenoadenosines as Potent and Selective A₃ Adenosine Receptor Agonists with Unusual Sugar Puckering and Nucleobase Orientation.