Literature DB >> 22370318

Vandetanib Versus placebo in patients with advanced non-small-cell lung cancer after prior therapy with an epidermal growth factor receptor tyrosine kinase inhibitor: a randomized, double-blind phase III trial (ZEPHYR).

Jin Soo Lee1, Vera Hirsh, Keunchil Park, Shukui Qin, Cesar R Blajman, Reury-Perng Perng, Yuh-Min Chen, Laura Emerson, Peter Langmuir, Christian Manegold.   

Abstract

PURPOSE: Vandetanib is a once-daily oral inhibitor of vascular endothelial growth factor receptor, epidermal growth factor receptor (EGFR), and RET signaling. This placebo-controlled trial assessed whether vandetanib conferred an overall survival benefit in patients with advanced non-small-cell lung cancer (NSCLC) after prior treatment with an EGFR tyrosine kinase inhibitor and one or two chemotherapy regimens. PATIENTS AND METHODS: Eligible patients were randomly assigned 2:1 to receive vandetanib 300 mg/d or placebo until disease progression or unacceptable toxicity. The primary objective was to compare the outcomes between the two arms with respect to overall survival.
RESULTS: Overall, 924 patients received vandetanib (n = 617) or placebo (n = 307). No significant increase in overall survival was detected in the vandetanib cohort compared with placebo (hazard ratio = 0.95; 95.2% CI, 0.81 to 1.11; P = .527); median overall survival was 8.5 months versus 7.8 months for vandetanib and placebo patients, respectively. Statistically significant advantages favoring vandetanib were observed for progression-free survival (hazard ratio = 0.63; P < .001) and objective response rate (2.6% v 0.7%; P = .028). Postprogression therapy was balanced across the cohorts in both number and type. Adverse events were generally consistent with previous NSCLC studies of vandetanib 300 mg; common events occurring with a greater frequency in the vandetanib arm versus placebo included diarrhea (46% v 11%), rash (42% v 11%), and hypertension (26% v 3%).
CONCLUSION: The study did not demonstrate an overall survival benefit for vandetanib versus placebo. There was a higher incidence of some adverse events with vandetanib.

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Year:  2012        PMID: 22370318     DOI: 10.1200/JCO.2011.36.1709

Source DB:  PubMed          Journal:  J Clin Oncol        ISSN: 0732-183X            Impact factor:   44.544


  104 in total

Review 1.  Risk of gastrointestinal events with newly approved (after 2011) vascular endothelial growth factor receptor tyrosine kinase inhibitors in cancer patients: a meta-analysis of randomized controlled trials.

Authors:  Jing Li; Jian Gu
Journal:  Eur J Clin Pharmacol       Date:  2017-07-15       Impact factor: 2.953

Review 2.  Strategies for overcoming resistance to EGFR family tyrosine kinase inhibitors.

Authors:  Giuseppe Giaccone; Yisong Wang
Journal:  Cancer Treat Rev       Date:  2011-03-01       Impact factor: 12.111

3.  Review of the treatment of metastatic non small cell lung carcinoma: A practical approach.

Authors:  Vera Hirsh
Journal:  World J Clin Oncol       Date:  2011-06-10

4.  Vandetanib in advanced non small cell lung cancer: a promise unfulfilled.

Authors:  Richard H de Boer
Journal:  Transl Lung Cancer Res       Date:  2013-02

5.  ZEPHYR: failure of a "spring wind" in lung cancer.

Authors:  Alessandro Morabito
Journal:  Transl Lung Cancer Res       Date:  2013-02

Review 6.  Targeting angiogenesis in lung cancer - Pitfalls in drug development.

Authors:  Wolfgang Hilbe; Christian Manegold; Andreas Pircher
Journal:  Transl Lung Cancer Res       Date:  2012-06

7.  Fatigue associated with newly approved vascular endothelial growth factor receptor tyrosine kinase inhibitors in cancer patients: an up-to-date meta-analysis.

Authors:  Jing Li; Jian Gu
Journal:  Int J Clin Oncol       Date:  2017-07-21       Impact factor: 3.402

8.  Apatinib for EGFR-TKI and chemotherapy refractory in an advanced lung cancer patient: a case report.

Authors:  Ying Chen; Junping Gong; Huiming Zhou; Xiujuan Qu; Yuee Teng; Yunpeng Liu; Bo Jin
Journal:  J Thorac Dis       Date:  2018-07       Impact factor: 2.895

Review 9.  Clinical meta-analyses of targeted therapies in adenocarcinoma.

Authors:  Emilio Bria; Maria Bonomi; Sara Pilotto; Francesco Massari; Silvia Novello; Matteo Giaj Levra; Giampaolo Tortora; Giorgio Scagliotti
Journal:  Target Oncol       Date:  2013-01-25       Impact factor: 4.493

Review 10.  Radiation therapy for early stage lung cancer.

Authors:  Bhupesh Parashar; Shruthi Arora; A Gabriella Wernicke
Journal:  Semin Intervent Radiol       Date:  2013-06       Impact factor: 1.513

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