Literature DB >> 22222600

Phase I and pharmacokinetic study of elacytarabine, a novel 5'-elaidic acid derivative of cytarabine, in adults with refractory hematological malignancies.

F J Giles, N Vey, D Rizzieri, F Ravandi, T Prebet, G Borthakur, T F Jacobsen, S Hagen, B Nilsson, S O'Brien.   

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Year:  2012        PMID: 22222600     DOI: 10.1038/leu.2012.1

Source DB:  PubMed          Journal:  Leukemia        ISSN: 0887-6924            Impact factor:   11.528


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  6 in total

1.  Elacytarabine has single-agent activity in patients with advanced acute myeloid leukaemia.

Authors:  Susan O'Brien; David A Rizzieri; Norbert Vey; Farhad Ravandi; Utz O Krug; Mikkael A Sekeres; Mike Dennis; Adriano Venditti; Donald A Berry; Tove Flem Jacobsen; Karin Staudacher; Trygve Bergeland; Francis J Giles
Journal:  Br J Haematol       Date:  2012-06-15       Impact factor: 6.998

Review 2.  Novel therapeutics in acute myeloid leukemia.

Authors:  Kendra Sweet; Jeffrey E Lancet
Journal:  Curr Hematol Malig Rep       Date:  2014-06       Impact factor: 3.952

3.  Elacytarabine, a novel 5'-elaidic acid derivative of cytarabine, and idarubicin combination is active in refractory acute myeloid leukemia.

Authors:  Francis Giles; David Rizzieri; Farhad Ravandi; Ronan Swords; Tove Flem Jacobsen; Susan O'Brien
Journal:  Leuk Res       Date:  2012-01-09       Impact factor: 3.156

Review 4.  Clinical potential of elacytarabine in patients with acute myeloid leukemia.

Authors:  Lindsay A M Rein; David A Rizzieri
Journal:  Ther Adv Hematol       Date:  2014-12

Review 5.  Developmental therapeutics in acute myelogenous leukemia: are there any new effective cytotoxic chemotherapeutic agents out there?

Authors:  Alice Mims; Robert K Stuart
Journal:  Curr Hematol Malig Rep       Date:  2013-06       Impact factor: 3.952

Review 6.  Improving nucleoside analogs via lipid conjugation: Is fatter any better?

Authors:  Peter Alexander; Gregory Kucera; Timothy S Pardee
Journal:  Crit Rev Oncol Hematol       Date:  2016-01-21       Impact factor: 6.312

  6 in total

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