Literature DB >> 22217678

Kinetics of nevirapine and its impact on HIV-1 RNA levels in maternal plasma and breast milk over time after perinatal single-dose nevirapine.

Jim Aizire1, Michelle S McConnell, Peter Mudiope, Michael Mubiru, Flavia Matovu, Teresa L Parsons, Ali Elbireer, Monica Nolan, Edward N Janoff, Mary Glenn Fowler.   

Abstract

OBJECTIVE: To determine kinetics after single-dose nevirapine and the impact on HIV RNA [viral load (VL)] in maternal plasma and breast milk (BM).
METHODS: Cohort of 120 HIV-1-infected pregnant Ugandan women received perinatal single-dose nevirapine alone and followed up with their infants through 24 weeks postdelivery. We assessed the relationship of nevirapine concentration (tandem mass spectroscopy) and HIV-1 VL (Roche AMPLICOR HIV-1 Kit, version 1.5) in maternal plasma and BM over time.
RESULTS: At week 1 postpartum, NVP (≥10 ng/mL) was detected in all 53 plasma and 47 of 51 (92.2%) BM samples with median (interquartile ranges) of, respectively, 171 (78-214) ng/mL and 112 (64-158) ng/mL, P = 0.075, which decreased subsequently with traces persisting through week 4 in plasma. Plasma and BM VL dropped by week 1 and were highly correlated at delivery (R = 0.71, P < 0.001) and week 1 (R = 0.69, P < 0.001) but not thereafter. At week 1, VL correlated inversely with NVP concentration in plasma (R = 0.39, P = 0.004) and BM (R = 0.48, P = 0.013). There was a VL rebound in both compartments, which peaked at week 4 to levels greater than those at week 1 [significantly in plasma (P < 0.001) but not in BM] and remained stable thereafter. Median VL was consistently greater (11- to 50-fold) in plasma than BM at all time points (all P < 0.001).
CONCLUSIONS: After single-dose nevirapine, NVP concentration was comparably high through week 1, accompanied by suppression of plasma and BM VL. A longer "tail" (>1 week) of potent postnatal antiretroviral drugs is warranted to minimize the observed VL rebound and potential for NVP resistance as a result of persistent NVP traces.

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Year:  2012        PMID: 22217678     DOI: 10.1097/QAI.0b013e318246bf9e

Source DB:  PubMed          Journal:  J Acquir Immune Defic Syndr        ISSN: 1525-4135            Impact factor:   3.731


  7 in total

1.  Dynamics of breast milk HIV-1 RNA with unilateral mastitis or abscess.

Authors:  Katherine Semrau; Louise Kuhn; Daniel R Brooks; Howard Cabral; Moses Sinkala; Chipepo Kankasa; Donald M Thea; Grace M Aldrovandi
Journal:  J Acquir Immune Defic Syndr       Date:  2013-03-01       Impact factor: 3.731

2.  Clinical and genetic determinants of plasma nevirapine exposure following an intrapartum dose to prevent mother-to-child HIV transmission.

Authors:  Saran Vardhanabhuti; Edward P Acosta; Heather J Ribaudo; Patrice Severe; Umesh Lalloo; Nagalingeshwaran Kumarasamy; Frank Taulo; Joseph Kabanda; Olola Oneko; Prudence Ive; Pradeep Sambarey; Ellen S Chan; Jane Hitti; Francis Hong; Deborah McMahon; David W Haas
Journal:  J Infect Dis       Date:  2013-05-17       Impact factor: 5.226

Review 3.  Impact of antiretroviral drugs in pregnant women and their children in Africa: HIV resistance and treatment outcomes.

Authors:  Roger Paredes; Vincent C Marconi; Shahin Lockman; Elaine J Abrams; Louise Kuhn
Journal:  J Infect Dis       Date:  2013-06-15       Impact factor: 5.226

Review 4.  Is infant exposure to antiretroviral drugs during breastfeeding quantitatively important? A systematic review and meta-analysis of pharmacokinetic studies.

Authors:  Catriona John Waitt; Paul Garner; Laura Jayne Bonnett; Saye Hock Khoo; Laura Jayne Else
Journal:  J Antimicrob Chemother       Date:  2015-04-08       Impact factor: 5.790

5.  Mother-to-Child HIV-1 Transmission Events Are Differentially Impacted by Breast Milk and Its Components from HIV-1-Infected Women.

Authors:  Ruizhong Shen; Jenna Achenbach; Yue Shen; Jana Palaia; Jeremy T Rahkola; Heidi J Nick; Lesley E Smythies; Michelle McConnell; Mary G Fowler; Phillip D Smith; Edward N Janoff
Journal:  PLoS One       Date:  2015-12-17       Impact factor: 3.240

6.  Nevirapine, sodium concentration and HIV-1 RNA in breast milk and plasma among HIV-infected women receiving short-course antiretroviral prophylaxis.

Authors:  Kirsten Salado-Rasmussen; Zahra P Theilgaard; Mercy G Chiduo; Ib C Bygbjerg; Jan Gerstoft; Margrethe Lüneborg-Nielsen; Martha Lemnge; Terese L Katzenstein
Journal:  PLoS One       Date:  2015-03-26       Impact factor: 3.240

7.  Postnatally-transmitted HIV-1 Envelope variants have similar neutralization-sensitivity and function to that of nontransmitted breast milk variants.

Authors:  Genevieve G Fouda; Tatenda Mahlokozera; Jesus F Salazar-Gonzalez; Maria G Salazar; Gerald Learn; Surender B Kumar; S Moses Dennison; Elizabeth Russell; Katherine Rizzolo; Frederick Jaeger; Fangping Cai; Nathan A Vandergrift; Feng Gao; Beatrice Hahn; George M Shaw; Christina Ochsenbauer; Ronald Swanstrom; Steve Meshnick; Victor Mwapasa; Linda Kalilani; Susan Fiscus; David Montefiori; Barton Haynes; Jesse Kwiek; S Munir Alam; Sallie R Permar
Journal:  Retrovirology       Date:  2013-01-10       Impact factor: 4.602

  7 in total

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