Literature DB >> 22173279

The mast cell stabilizer ketotifen reduces joint capsule fibrosis in a rabbit model of post-traumatic joint contractures.

Michael J Monument1, David A Hart, A Dean Befus, Paul T Salo, Mei Zhang, Kevin A Hildebrand.   

Abstract

OBJECTIVES: Using a rabbit model of post-traumatic joint contractures, we investigated whether treatment with a mast cell stabilizer after joint injury would lessen the molecular manifestations of joint capsule fibrosis.
METHODS: Surgical joint injury was used to create stable post-traumatic contractures of the knee in skeletally mature New Zealand white rabbits. Four groups of animals were studied: a non-operated control group (n = 8), an operated contracture group (n = 13) and two operated groups treated with the mast cell stabilizer, ketotifen, at doses of 0.5 mg/kg (n = 9) and 1.0 mg/kg (n = 9) twice daily. Joint capsule fibrosis was assessed by quantifying the mRNA and protein levels of α-SMA, tryptase, TGF-β1, collagen I and collagen III. Significance was tested using an ANOVA analysis of variance.
RESULTS: The protein and mRNA levels of α-SMA, TGF-β1, tryptase and collagen I and III were significantly elevated in the operated contracture group compared to control (p < 0.01). In both ketotifen-treated groups, protein and mRNA levels of α-SMA, TGF-β1 and collagen I were significantly reduced compared to the operated contracture group (p < 0.01).
CONCLUSIONS: These data suggest an inflammatory pathway mediated by mast cell activation is involved in joint capsule fibrosis after traumatic injury.

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Year:  2011        PMID: 22173279      PMCID: PMC3710138          DOI: 10.1007/s00011-011-0409-3

Source DB:  PubMed          Journal:  Inflamm Res        ISSN: 1023-3830            Impact factor:   4.575


  38 in total

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Authors:  R Lindholm; S Lindholm; P Liukko; J Paasimäki; S Isokääntä; R Rossi; E Autio; E Tamminen
Journal:  J Bone Joint Surg Br       Date:  1969-02-01

Review 6.  Ketotifen. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic use in asthma and allergic disorders.

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Journal:  Drugs       Date:  1990-09       Impact factor: 9.546

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Journal:  Arzneimittelforschung       Date:  1989-10

10.  Ketotifen: current views on its mechanism of action and their therapeutic implications.

Authors:  L P Craps; U M Ney
Journal:  Respiration       Date:  1984       Impact factor: 3.580

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