Literature DB >> 22170412

Small bowel injury induced by selective cyclooxygenase-2 inhibitors: a prospective, double-blind, randomized clinical trial comparing celecoxib and meloxicam.

Yuji Maehata1, Motohiro Esaki, Toshibumi Morishita, Shuji Kochi, Shingo Endo, Kentaro Shikata, Hiroyuki Kobayashi, Takayuki Matsumoto.   

Abstract

BACKGROUND: Selective cyclooxygenase (COX)-2 inhibitors are less harmful to the small bowel mucosa than non-selective anti-inflammatory drugs. We aimed to compare the severity of small bowel mucosal injury in healthy volunteers induced by two selective COX-2 inhibitors, celecoxib and meloxicam, in a randomized, double-blind trial, using capsule endoscopy (CE).
METHODS: Twenty-nine healthy subjects were randomized to take either celecoxib (200 mg twice daily) or meloxicam (10 mg once daily) for 2 weeks. The incidence and the number of small bowel mucosal injuries (bleeding, ulcers, and erosions) observed by CE were compared between the two groups.
RESULTS: The overall incidence of small bowel mucosal injury was not different between the celecoxib group (6 of 14 subjects, 42.9%) and the meloxicam group (4 of 15 subjects, 26.7%, P = 0.45). In subjects with positive CE findings, the number of ulcers was greater in the meloxicam group than in the celecoxib group (P = 0.02), while such a trend was not found with regard to erosions (P = 0.52). The distribution of mucosal lesions within the small bowel was similar in the two groups.
CONCLUSIONS: Selective COX-2 inhibitors are not completely safe for the small bowel. The mucosal lesions may be less severe with celecoxib than with meloxicam.

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Year:  2011        PMID: 22170412     DOI: 10.1007/s00535-011-0501-z

Source DB:  PubMed          Journal:  J Gastroenterol        ISSN: 0944-1174            Impact factor:   7.527


  40 in total

1.  Distribution of small intestinal mucosal injuries as a result of NSAID administration.

Authors:  Shunji Fujimori; Katya Gudis; Yoko Takahashi; Tsuguhiko Seo; Yukie Yamada; Akihito Ehara; Tsuyoshi Kobayashi; Keigo Mitsui; Masaoki Yonezawa; Shu Tanaka; Atsushi Tatsuguchi; Choitsu Sakamoto
Journal:  Eur J Clin Invest       Date:  2010-04-14       Impact factor: 4.686

2.  Prevention of NSAID-induced gastric ulcer with misoprostol: multicentre, double-blind, placebo-controlled trial.

Authors:  D Y Graham; N M Agrawal; S H Roth
Journal:  Lancet       Date:  1988-12-03       Impact factor: 79.321

3.  Clinical and endoscopic features of nonsteroidal anti-inflammatory drug-induced colonic ulcerations.

Authors:  K Kurahara; T Matsumoto; M Iida; K Honda; T Yao; M Fujishima
Journal:  Am J Gastroenterol       Date:  2001-02       Impact factor: 10.864

4.  Cyclooxygenase selectivity of non-steroid anti-inflammatory drugs in humans: ex vivo evaluation.

Authors:  F Giuliano; J G Ferraz; R Pereira; G de Nucci; T D Warner
Journal:  Eur J Pharmacol       Date:  2001-08-24       Impact factor: 4.432

5.  Gastrointestinal toxicity with celecoxib vs nonsteroidal anti-inflammatory drugs for osteoarthritis and rheumatoid arthritis: the CLASS study: A randomized controlled trial. Celecoxib Long-term Arthritis Safety Study.

Authors:  F E Silverstein; G Faich; J L Goldstein; L S Simon; T Pincus; A Whelton; R Makuch; G Eisen; N M Agrawal; W F Stenson; A M Burr; W W Zhao; J D Kent; J B Lefkowith; K M Verburg; G S Geis
Journal:  JAMA       Date:  2000-09-13       Impact factor: 56.272

6.  Nonsteroidal anti-inflammatory drug enteropathy in rats: role of permeability, bacteria, and enterohepatic circulation.

Authors:  B K Reuter; N M Davies; J L Wallace
Journal:  Gastroenterology       Date:  1997-01       Impact factor: 22.682

7.  Gastrointestinal tolerability of meloxicam compared to diclofenac in osteoarthritis patients. International MELISSA Study Group. Meloxicam Large-scale International Study Safety Assessment.

Authors:  C Hawkey; A Kahan; K Steinbrück; C Alegre; E Baumelou; B Bégaud; J Dequeker; H Isomäki; G Littlejohn; J Mau; S Papazoglou
Journal:  Br J Rheumatol       Date:  1998-09

8.  Improvement in gastrointestinal tolerability of the selective cyclooxygenase (COX)-2 inhibitor, meloxicam, compared with piroxicam: results of the Safety and Efficacy Large-scale Evaluation of COX-inhibiting Therapies (SELECT) trial in osteoarthritis.

Authors:  J Dequeker; C Hawkey; A Kahan; K Steinbrück; C Alegre; E Baumelou; B Bégaud; H Isomäki; G Littlejohn; J Mau; S Papazoglou
Journal:  Br J Rheumatol       Date:  1998-09

9.  Long-term effects of nonsteroidal anti-inflammatory drugs and cyclooxygenase-2 selective agents on the small bowel: a cross-sectional capsule enteroscopy study.

Authors:  Laurence Maiden; Bjarni Thjodleifsson; Anna Seigal; Ingvar Iain Bjarnason; David Scott; Sigurbjorn Birgisson; Ingvar Bjarnason
Journal:  Clin Gastroenterol Hepatol       Date:  2007-07-10       Impact factor: 11.382

10.  Gastrointestinal damage associated with the use of nonsteroidal antiinflammatory drugs.

Authors:  M C Allison; A G Howatson; C J Torrance; F D Lee; R I Russell
Journal:  N Engl J Med       Date:  1992-09-10       Impact factor: 91.245

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  5 in total

Review 1.  Multiple NSAID-induced hits injure the small intestine: underlying mechanisms and novel strategies.

Authors:  Urs A Boelsterli; Matthew R Redinbo; Kyle S Saitta
Journal:  Toxicol Sci       Date:  2012-10-22       Impact factor: 4.849

2.  Capsule endoscopy findings for the diagnosis of Crohn's disease: a nationwide case-control study.

Authors:  Motohiro Esaki; Takayuki Matsumoto; Naoki Ohmiya; Ema Washio; Toshifumi Morishita; Kei Sakamoto; Hiroo Abe; Shojiro Yamamoto; Tetsu Kinjo; Kazutomo Togashi; Kenji Watanabe; Fumihito Hirai; Masanao Nakamura; Sadaharu Nouda; Shinya Ashizuka; Teppei Omori; Shuji Kochi; Shunichi Yanai; Yuta Fuyuno; Atsushi Hirano; Junji Umeno; Takanari Kitazono; Fukunori Kinjo; Mamoru Watanabe; Toshiyuki Matsui; Yasuo Suzuki
Journal:  J Gastroenterol       Date:  2018-09-15       Impact factor: 7.527

3.  Emu oil reduces small intestinal inflammation in the absence of clinical improvement in a rat model of indomethacin-induced enteropathy.

Authors:  Suzanne M Abimosleh; Cuong D Tran; Gordon S Howarth
Journal:  Evid Based Complement Alternat Med       Date:  2013-03-14       Impact factor: 2.629

4.  Non-steroidal anti-inflammatory drug-induced enteropathy as a major risk factor for small bowel bleeding: a retrospective study.

Authors:  Doo-Ho Lim; Kyoungwon Jung; Seung Bum Lee; In Kyu Park; Hee Jeong Cha; Jae Ho Park; Byung Gyu Kim; Seok Won Jung; Jae Hyun Kim; Sung Eun Kim; Won Moon; Moo In Park; Seun Ja Park
Journal:  BMC Gastroenterol       Date:  2020-06-08       Impact factor: 3.067

Review 5.  Current knowledge on non-steroidal anti-inflammatory drug-induced small-bowel damage: a comprehensive review.

Authors:  Toshio Watanabe; Yasuhiro Fujiwara; Francis K L Chan
Journal:  J Gastroenterol       Date:  2019-12-21       Impact factor: 7.527

  5 in total

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