Literature DB >> 22111917

Expanding the azaspiro[3.3]heptane family: synthesis of novel highly functionalized building blocks.

Johannes A Burkhard1, Carine Guérot, Henner Knust, Erick M Carreira.   

Abstract

The preparation of versatile azaspiro[3.3]heptanes carrying multiple exit vectors is disclosed. Expedient synthetic routes enable the straightforward access to these novel modules that are expected to have significance in drug discovery and design.
© 2011 American Chemical Society

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Year:  2011        PMID： 22111917     DOI： 10.1021/ol2028459

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  11 in total

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