Literature DB >> 22025154

Preliminary efficacy of the anti-insulin-like growth factor type 1 receptor antibody figitumumab in patients with refractory Ewing sarcoma.

Heribert Juergens1, Najat C Daw, Birgit Geoerger, Stefano Ferrari, Milena Villarroel, Isabelle Aerts, Jeremy Whelan, Uta Dirksen, Mary L Hixon, Donghua Yin, Tao Wang, Stephanie Green, Luisa Paccagnella, Antonio Gualberto.   

Abstract

PURPOSE: Patients with Ewing sarcoma (ES) with metastases and those who relapse fare poorly and receive therapies that carry significant toxicity. This phase 1/2 study was conducted to evaluate the efficacy of figitumumab in advanced ES. PATIENTS AND METHODS: Patients with sarcoma 10 to 18 years old were enrolled in two dose escalation cohorts (20 and 30 mg/Kg intravenously every 4 weeks) in the phase 1 portion of the study. Patients with ES 10 years old or older were enrolled in the phase 2 portion of the study. The primary phase 2 objective was objective response rate (ORR).
RESULTS: Thirty-one patients with ES (n = 16), osteosarcoma (n = 11), or other sarcomas (n = 4) were enrolled in the phase 1 portion of the study. Dose escalation proceeded to 30 mg/kg every 4 weeks with no dose-limiting toxicity identified. In the phase 2 portion of the study, 107 patients with ES received figitumumab at 30 mg/kg every 4 weeks for a median of 2 cycles (range, 1 to 16). Sixty three percent of phase 2 patients had received at least three prior treatment regimens. Of 106 evaluable patients, 15 had a partial response (ORR, 14.2%) and 25 had stable disease. Median overall survival was 8.9 months. Importantly, patients with a pretreatment circulating free insulin-like growth factor (IGF) -1 lower than 0.65 ng/mL (n = 14) had a median OS of 3.6 months, whereas those with a baseline free IGF-1 ≥ 0.65 ng/mL (n = 84) had a median OS of 10.4 months (P < .001).
CONCLUSION: Figitumumab had modest activity as single agent in advanced ES. A strong association between pretreatment serum IGF-1 and survival benefit was identified.

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Year:  2011        PMID: 22025154      PMCID: PMC3236653          DOI: 10.1200/JCO.2010.33.0670

Source DB:  PubMed          Journal:  J Clin Oncol        ISSN: 0732-183X            Impact factor:   44.544


  20 in total

Review 1.  Figitumumab (CP-751,871) for cancer therapy.

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4.  Insulin-like growth factor-I and cancer mortality in older men.

Authors:  Jacqueline M Major; Gail A Laughlin; Donna Kritz-Silverstein; Deborah L Wingard; Elizabeth Barrett-Connor
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5.  The insulin-like growth factor-1 receptor-targeting antibody, CP-751,871, suppresses tumor-derived VEGF and synergizes with rapamycin in models of childhood sarcoma.

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Journal:  Cancer Res       Date:  2009-09-29       Impact factor: 12.701

Review 6.  Emerging role of insulin-like growth factor receptor inhibitors in oncology: early clinical trial results and future directions.

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Review 7.  Insulin and insulin-like growth factor signalling in neoplasia.

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8.  Safety, pharmacokinetics, and preliminary activity of the anti-IGF-1R antibody figitumumab (CP-751,871) in patients with sarcoma and Ewing's sarcoma: a phase 1 expansion cohort study.

Authors:  David Olmos; Sophie Postel-Vinay; L Rhoda Molife; Scott H Okuno; Scott M Schuetze; M Luisa Paccagnella; Gretchen N Batzel; Donghua Yin; Kathryn Pritchard-Jones; Ian Judson; Francis P Worden; Antonio Gualberto; Michelle Scurr; Johann S de Bono; Paul Haluska
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9.  Insulin-like growth factor 1 (IGF1), IGF binding protein 3 (IGFBP3), and breast cancer risk: pooled individual data analysis of 17 prospective studies.

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  93 in total

1.  Targeting of insulin-like growth factor type 1 receptor in Ewing sarcoma: unfulfilled promise or a promising beginning?

Authors:  Alan L Ho; Gary K Schwartz
Journal:  J Clin Oncol       Date:  2011-10-24       Impact factor: 44.544

Review 2.  Molecular Pathways: Clinical Applications and Future Direction of Insulin-like Growth Factor-1 Receptor Pathway Blockade.

Authors:  Wade T Iams; Christine M Lovly
Journal:  Clin Cancer Res       Date:  2015-10-01       Impact factor: 12.531

3.  A Combination CDK4/6 and IGF1R Inhibitor Strategy for Ewing Sarcoma.

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Journal:  Clin Cancer Res       Date:  2018-11-05       Impact factor: 12.531

4.  CD39 is a promising therapeutic antibody target for the treatment of soft tissue sarcoma.

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Journal:  Am J Transl Res       Date:  2015-06-15       Impact factor: 4.060

5.  Vincristine, Ifosfamide, and Doxorubicin for Initial Treatment of Ewing Sarcoma in Adults.

Authors:  Michael J Wagner; Vancheswaran Gopalakrishnan; Vinod Ravi; J Andrew Livingston; Anthony P Conley; Dejka Araujo; Neeta Somaiah; Maria A Zarzour; Ravin Ratan; Wei-Lien Wang; Shreyaskumar R Patel; Alexander Lazar; Joseph A Ludwig; Robert S Benjamin
Journal:  Oncologist       Date:  2017-07-14

6.  Tandem high-dose chemotherapy strategy as first-line treatment of primary disseminated multifocal Ewing sarcomas in children, adolescents and young adults.

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Review 7.  Early phase clinical trials of anticancer agents in children and adolescents - an ITCC perspective.

Authors:  Lucas Moreno; Andrew D J Pearson; Xavier Paoletti; Irene Jimenez; Birgit Geoerger; Pamela R Kearns; C Michel Zwaan; Francois Doz; Andre Baruchel; Josef Vormoor; Michela Casanova; Stefan M Pfister; Bruce Morland; Gilles Vassal
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Review 8.  New advances in targeted gastric cancer treatment.

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Journal:  World J Gastroenterol       Date:  2016-08-14       Impact factor: 5.742

Review 9.  Children's Oncology Group's 2013 blueprint for research: bone tumors.

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Journal:  Pediatr Blood Cancer       Date:  2012-12-19       Impact factor: 3.167

10.  PTEN deficiency mediates a reciprocal response to IGFI and mTOR inhibition.

Authors:  Mukund Patel; Nicholas C Gomez; Andrew W McFadden; Billie M Moats-Staats; Sam Wu; Andres Rojas; Travis Sapp; Jeremy M Simon; Scott V Smith; Kathleen Kaiser-Rogers; Ian J Davis
Journal:  Mol Cancer Res       Date:  2014-07-03       Impact factor: 5.852

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