Literature DB >> 21997126

Dual properties of anticancer agents: an exploratory study on the in vitro anti-Candida properties of thirty drugs.

Madhushree M Routh1, Jayant S Raut, S Mohan Karuppayil.   

Abstract

BACKGROUND: Anticancer/antineoplastic agents could be a good resource for the discovery of novel antifungal agents and targets since human beings share a common eukaryotic heritage with fungi.
METHODS: Thirty commonly prescribed anticancer drugs belonging to 12 different classes were analyzed for their effects on the growth of Candida albicans. Minimum inhibitory concentrations (MICs) were obtained using standard CLSI-M27 A2 methodology, and minimal fungicidal concentrations (MFCs) were determined via the agar plate method.
RESULTS: Anticancer agents inhibited the growth of C. albicans in a concentration-dependent manner. Nine drugs from different classes were effective at low concentrations (≤50 μg·ml(-1)), while 15 anticancer drugs exhibited MICs of 100 μg·ml(-1). Sixteen out of 30 drugs exerted fungicidal activity in the range of 400-800 μg·ml(-1).
CONCLUSIONS: MICs and MFCs for 30 anticancer drugs were established against C. albicans. Our study highlighted the anti-Candida potential of these drugs, which may give insights to unexplored targets for antifungal chemotherapy.
Copyright © 2011 S. Karger AG, Basel.

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Year:  2011        PMID: 21997126     DOI: 10.1159/000330454

Source DB:  PubMed          Journal:  Chemotherapy        ISSN: 0009-3157            Impact factor:   2.544


  3 in total

1.  The antibacterial agent, moxifloxacin inhibits virulence factors of Candida albicans through multitargeting.

Authors:  Ashwini Jadhav; Bhagyashree Bansode; Datta Phule; Amruta Shelar; Rajendra Patil; Wasudev Gade; Kiran Kharat; Sankunny Mohan Karuppayil
Journal:  World J Microbiol Biotechnol       Date:  2017-04-13       Impact factor: 3.312

2.  The triphenylethylenes, a novel class of antifungals.

Authors:  Audrey R Odom
Journal:  MBio       Date:  2014-04-29       Impact factor: 7.867

3.  Cancer drugs inhibit morphogenesis in the human fungal pathogen, Candida albicans.

Authors:  Madhushree M Routh; Nitin M Chauhan; S Mohan Karuppayil
Journal:  Braz J Microbiol       Date:  2014-01-15       Impact factor: 2.476

  3 in total

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