Literature DB >> 21896859

Topical dexamethasone-cyclodextrin microparticle eye drops for diabetic macular edema.

Masaki Tanito1, Katsunori Hara, Yasuyuki Takai, Yotaro Matsuoka, Nobuhiro Nishimura, Phatsawee Jansook, Thorsteinn Loftsson, Einar Stefánsson, Akihiro Ohira.   

Abstract

PURPOSE: To test the safety and efficacy of topical 1.5% dexamethasone aqueous eye drops with cyclodextrin microparticles for diabetic macular edema (DME).
METHODS: Nineteen eyes of 19 consecutive patients with DME were administered dexamethasone-cyclodextrin eye drops three or six times a day for 4 weeks and then observed for 4 weeks without treatment. Visual acuity, intraocular pressure, and spectral domain optical coherent tomography-measured central macular thickness recordings at weeks 0 (baseline), 4, and 8. These parameters were compared using Bonferroni-corrected paired t-tests.
RESULTS: At weeks 0, 4, and 8, logMAR visual acuity (mean ± SD) was 0.52 ± 0.41, 0.37 ± 0.40 (P = 0.0025 vs. baseline), and 0.45 ± 0.41, respectively; central macular thickness (μm) was 512 ± 164, 399 ± 154 (P = 0.0016 vs. baseline), and 488 ± 172 (P = 0.0116 versus week 4), respectively; and intraocular pressure (mm Hg) was 15.2 ± 3.1, 17.4 ± 4.2 (P = 0.0015 vs. baseline) and 15.8 ± 4.0, respectively. At week 4, in 12 (63%) of 19 eyes, central macular thickness had decreased more than 10%, and the mean change was -20% (-65% to +10%). In 14 of 19 eyes (74%) visual acuity (logMAR) had improved more than 0.1 at week 4. No subjects showed severe adverse effects related to the eye drops.
CONCLUSIONS: Based on this short pilot study, topical dexamethasone-cyclodextrin eye drops are well tolerated, decrease central macular thickness, and improve visual acuity in DME. The results encourage comparative studies between dexamethasone cyclodextrin microparticle eye drops and other treatments for DME. (http://www.umin.ac.jp/ctr number, UMIN000001790.).

Entities:  

Mesh:

Substances:

Year:  2011        PMID: 21896859     DOI: 10.1167/iovs.11-8178

Source DB:  PubMed          Journal:  Invest Ophthalmol Vis Sci        ISSN: 0146-0404            Impact factor:   4.799


  15 in total

Review 1.  Novel Therapies in Development for Diabetic Macular Edema.

Authors:  Aniruddha Agarwal; Rubbia Afridi; Muhammad Hassan; Mohammad Ali Sadiq; Yasir J Sepah; Diana V Do; Quan Dong Nguyen
Journal:  Curr Diab Rep       Date:  2015-10       Impact factor: 4.810

Review 2.  Drug and gene delivery to the back of the eye: from bench to bedside.

Authors:  Cheryl L Rowe-Rendleman; Shelley A Durazo; Uday B Kompella; Kay D Rittenhouse; Adriana Di Polo; Alan L Weiner; Hans E Grossniklaus; Muna I Naash; Alfred S Lewin; Alan Horsager; Henry F Edelhauser
Journal:  Invest Ophthalmol Vis Sci       Date:  2014-04-28       Impact factor: 4.799

3.  Ocular Drug Distribution and Safety of a Noninvasive Ocular Drug Delivery System of Dexamethasone Sodium Phosphate in Rabbit.

Authors:  Kongnara Papangkorn; John W Higuchi; Balbir Brar; William I Higuchi
Journal:  J Ocul Pharmacol Ther       Date:  2018-02-12       Impact factor: 2.671

Review 4.  Pharmaceutical microscale and nanoscale approaches for efficient treatment of ocular diseases.

Authors:  I Bravo-Osuna; V Andrés-Guerrero; P Pastoriza Abal; I T Molina-Martínez; R Herrero-Vanrell
Journal:  Drug Deliv Transl Res       Date:  2016-12       Impact factor: 4.617

Review 5.  Novel Eye Drop Delivery Systems: Advance on Formulation Design Strategies Targeting Anterior and Posterior Segments of the Eye.

Authors:  Yaru Wang; Changhong Wang
Journal:  Pharmaceutics       Date:  2022-05-27       Impact factor: 6.525

Review 6.  Clinical Applications of Dexamethasone for Aged Eyes.

Authors:  Beatriz Abadia; Pilar Calvo; Antonio Ferreras; Fran Bartol; Guayente Verdes; Luis Pablo
Journal:  Drugs Aging       Date:  2016-09       Impact factor: 3.923

7.  Noninvasive Ocular Drug Delivery System of Dexamethasone Sodium Phosphate in the Treatment of Experimental Uveitis Rabbit.

Authors:  Kongnara Papangkorn; Eri Prendergast; John W Higuchi; Balbir Brar; William I Higuchi
Journal:  J Ocul Pharmacol Ther       Date:  2017-10-12       Impact factor: 2.671

Review 8.  Principles of pharmacology in the eye.

Authors:  Sahar Awwad; Abeer H A Mohamed Ahmed; Garima Sharma; Jacob S Heng; Peng T Khaw; Steve Brocchini; Alastair Lockwood
Journal:  Br J Pharmacol       Date:  2017-10-10       Impact factor: 8.739

9.  Solubilized ubiquinol for preserving corneal function.

Authors:  Youssef W Naguib; Sanjib Saha; Jessica M Skeie; Timothy Acri; Kareem Ebeid; Somaya Abdel-Rahman; Sandeep Kesh; Gregory A Schmidt; Darryl Y Nishimura; Jeffrey A Banas; Min Zhu; Mark A Greiner; Aliasger K Salem
Journal:  Biomaterials       Date:  2021-05-01       Impact factor: 15.304

10.  Lidocaine Cyclodextrin complex Ophthalmic Drop, a New Topical Anesthetic Choice.

Authors:  Aa Sabermoghadam Ranjbar; O Rajabi; R Salari; H Ashraf
Journal:  Iran Red Crescent Med J       Date:  2012-09-30       Impact factor: 0.611

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.