Literature DB >> 21865850

Knock-out of the potassium channel TASK-1 leads to a prolonged QT interval and a disturbed QRS complex.

Niels Decher1, Konstantin Wemhöner, Susanne Rinné, Michael F Netter, Marylou Zuzarte, Maria I Aller, Susann G Kaufmann, Xian Tao Li, Sven G Meuth, Jürgen Daut, Frank B Sachse, Sebastian K G Maier.   

Abstract

BACKGROUND/AIMS: The aim of the study was to characterize the whole cell current of the two-pore domain potassium channel TASK-1 (K2P3) in mouse ventricular cardiomyocytes (I(TASK-1)) and to analyze the cardiac phenotype of the TASK-1(-/-) mice. METHODS AND
RESULTS: We have quantified the ventricular I(TASK-1) current using the blocker A293 and TASK-1(-/-) mice. Surface electrocardiogram recordings of TASK-1(-/-) mice showed a prolonged QTc interval and a broadened QRS complex. The differences in electrocardiograms between wild type and TASK-1(-/-) mice disappeared during sympathetic stimulation of the animals. Quantitative RT-PCR, patch clamp recordings and measurements of hemodynamic performance of TASK-1(-/-) mice revealed no major compensatory changes in ion channel transcription. Action potential recordings of TASK-1(-/-) mouse cardiomyocytes indicated that I(TASK-1) modulates action potential duration. Our in vivo electrophysiological studies showed that isoflurane, which activates TASK-1, slowed heart rate and atrioventricular conduction of wild-type but not of TASK-1(-/-) mice.
CONCLUSION: The results of an invasive electrophysiological catheter protocol in combination with the observed QRS time prolongation in the surface electrocardiogram point towards a regulatory role of TASK-1 in the cardiac conduction system.
Copyright © 2011 S. Karger AG, Basel.

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Year:  2011        PMID: 21865850     DOI: 10.1159/000331715

Source DB:  PubMed          Journal:  Cell Physiol Biochem        ISSN: 1015-8987


  32 in total

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Authors:  Rikki H Chokshi; Aaron T Larsen; Brijesh Bhayana; Joseph F Cotten
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Journal:  Nature       Date:  2020-04-29       Impact factor: 49.962

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Authors:  Niels Decher; Aytug K Kiper; Caroline Rolfes; Eric Schulze-Bahr; Susanne Rinné
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7.  Physiological genomics identifies genetic modifiers of long QT syndrome type 2 severity.

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Review 8.  Investigational antiarrhythmic agents: promising drugs in early clinical development.

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Journal:  Pflugers Arch       Date:  2016-01-05       Impact factor: 3.657

10.  Ability to induce atrial fibrillation in the peri-operative period is associated with phosphorylation-dependent inhibition of TWIK protein-related acid-sensitive potassium channel 1 (TASK-1).

Authors:  Erin Harleton; Alessandra Besana; George M Comas; Peter Danilo; Tove S Rosen; Michael Argenziano; Michael R Rosen; Richard B Robinson; Steven J Feinmark
Journal:  J Biol Chem       Date:  2012-12-10       Impact factor: 5.157

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