Literature DB >> 21852469

Infectious diseases. A tropical disease hits the road.

Mitch Leslie.   

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Year:  2011        PMID: 21852469     DOI: 10.1126/science.333.6045.934

Source DB:  PubMed          Journal:  Science        ISSN: 0036-8075            Impact factor:   47.728


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  8 in total

1.  Pharmacological characterization, structural studies, and in vivo activities of anti-Chagas disease lead compounds derived from tipifarnib.

Authors:  Frederick S Buckner; Maria Terezinha Bahia; Praveen Kumar Suryadevara; Karen L White; David M Shackleford; Naveen Kumar Chennamaneni; Matthew A Hulverson; Joy U Laydbak; Eric Chatelain; Ivan Scandale; Christophe L M J Verlinde; Susan A Charman; Galina I Lepesheva; Michael H Gelb
Journal:  Antimicrob Agents Chemother       Date:  2012-07-09       Impact factor: 5.191

2.  Recent Developments in Sterol 14-demethylase Inhibitors for Chagas Disease.

Authors:  Frederick S Buckner; Julio A Urbina
Journal:  Int J Parasitol Drugs Drug Resist       Date:  2012-12       Impact factor: 4.077

3.  Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents.

Authors:  Maria V Papadopoulou; William D Bloomer; Howard S Rosenzweig; Marcel Kaiser; Eric Chatelain; Jean-Robert Ioset
Journal:  Bioorg Med Chem       Date:  2013-08-20       Impact factor: 3.641

4.  Novel 3-nitrotriazole-based amides and carbinols as bifunctional antichagasic agents.

Authors:  Maria V Papadopoulou; William D Bloomer; Galina I Lepesheva; Howard S Rosenzweig; Marcel Kaiser; Benjamín Aguilera-Venegas; Shane R Wilkinson; Eric Chatelain; Jean-Robert Ioset
Journal:  J Med Chem       Date:  2015-01-23       Impact factor: 7.446

5.  Sesquiterpene lactone in nanostructured parenteral dosage form is efficacious in experimental Chagas disease.

Authors:  Renata Tupinambá Branquinho; Vanessa Carla Furtado Mosqueira; Jaquelline Carla Valamiel de Oliveira-Silva; Marianne Rocha Simões-Silva; Dênia Antunes Saúde-Guimarães; Marta de Lana
Journal:  Antimicrob Agents Chemother       Date:  2014-01-21       Impact factor: 5.191

6.  Novel 3-nitro-1H-1,2,4-triazole-based compounds as potential anti-Chagasic drugs: in vivo studies.

Authors:  Maria V Papadopoulou; William D Bloomer; Howard S Rosenzweig; Rachel Ashworth; Shane R Wilkinson; Marcel Kaiser; Grasiella Andriani; Ana Rodriguez
Journal:  Future Med Chem       Date:  2013-10       Impact factor: 3.808

7.  Antitrypanosomal activity of 5-nitro-2-aminothiazole-based compounds.

Authors:  Maria V Papadopoulou; William D Bloomer; Howard S Rosenzweig; Shane R Wilkinson; Joanna Szular; Marcel Kaiser
Journal:  Eur J Med Chem       Date:  2016-04-08       Impact factor: 6.514

8.  Nitrotriazole-based acetamides and propanamides with broad spectrum antitrypanosomal activity.

Authors:  Maria V Papadopoulou; William D Bloomer; Howard S Rosenzweig; Shane R Wilkinson; Joanna Szular; Marcel Kaiser
Journal:  Eur J Med Chem       Date:  2016-08-09       Impact factor: 6.514

  8 in total

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