Literature DB >> 21782251

Use of insulin sensitizers for the treatment of major depressive disorder: a pilot study of pioglitazone for major depression accompanied by abdominal obesity.

David E Kemp1, Faramarz Ismail-Beigi, Stephen J Ganocy, Carla Conroy, Keming Gao, Sarah Obral, Elizabeth Fein, Robert L Findling, Joseph R Calabrese.   

Abstract

OBJECTIVE: This study was conducted to examine the safety and efficacy of pioglitazone, a thiazolidinedione insulin sensitizer, in adult outpatients with major depressive disorder.
METHOD: In a 12-week, open-label, flexible-dose study, 23 patients with major depressive disorder received pioglitazone monotherapy or adjunctive therapy initiated at 15 mg daily. Subjects were required to meet criteria for abdominal obesity (waist circumference>35 in. in women and >40 in. in men) or metabolic syndrome. The primary efficacy measure was the change from baseline to Week 12 on the Inventory of Depressive Symptomatology (IDS) total score. Partial responders (≥25% decrease in IDS total score) were eligible to participate in an optional extension phase for an additional three months.
RESULTS: Pioglitazone decreased depression symptom severity from a total IDS score of 40.3±1.8 to 19.2±1.8 at Week 12 (p<.001). Among partial responders (≥25% decrease in IDS total score), an improvement in depressive symptoms was maintained during an additional 3-month extension phase (total duration=24 weeks) according to IDS total scores (p<.001). Patients experienced a reduction in insulin resistance from baseline to Week 12 according to the log homeostasis model assessment (-0.8±0.75; p<.001) and a significant reduction in inflammation as measured by log highly- sensitive C-reactive protein (-0.87±0.72; p<.001). During the current episode, the majority of participants (74%, n=17), had already failed at least one antidepressant trial. The most common side effects were headache and dizziness; no patient discontinued due to side effects. LIMITATIONS: These data are limited by a small sample size and an open-label study design with no placebo control.
CONCLUSION: Although preliminary, pioglitazone appears to reduce depression severity and improve several markers of cardiometabolic risk, including insulin resistance and inflammation. Larger, placebo-controlled studies are indicated.
Copyright © 2011 Elsevier B.V. All rights reserved.

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Year:  2011        PMID: 21782251      PMCID: PMC3225727          DOI: 10.1016/j.jad.2011.06.033

Source DB:  PubMed          Journal:  J Affect Disord        ISSN: 0165-0327            Impact factor:   4.839


  50 in total

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2.  Bidirectional association between depression and type 2 diabetes mellitus in women.

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Journal:  Arch Intern Med       Date:  2010-11-22

3.  Acute treatment with the PPARgamma agonist pioglitazone and ibuprofen reduces glial inflammation and Abeta1-42 levels in APPV717I transgenic mice.

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4.  Ischemic preconditioning reveals that GLT1/EAAT2 glutamate transporter is a novel PPARgamma target gene involved in neuroprotection.

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5.  Long-term safety of pioglitazone versus glyburide in patients with recently diagnosed type 2 diabetes mellitus.

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6.  A pilot test of pioglitazone as an add-on in patients with relapsing remitting multiple sclerosis.

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7.  Long-term lipid effects of pioglitazone by baseline anti-hyperglycemia medication therapy and statin use from the PROactive experience (PROactive 14).

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1.  Pioglitazone is an effective treatment for patients with post-stroke depression combined with type 2 diabetes mellitus.

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Journal:  Exp Ther Med       Date:  2015-06-24       Impact factor: 2.447

2.  PPAR-γ agonism as a modulator of mood: proof-of-concept for pioglitazone in bipolar depression.

Authors:  David E Kemp; Martha Schinagle; Keming Gao; Carla Conroy; Stephen J Ganocy; Faramarz Ismail-Beigi; Joseph R Calabrese
Journal:  CNS Drugs       Date:  2014-06       Impact factor: 5.749

3.  Activation of PPARγ Attenuates the Expression of Physical and Affective Nicotine Withdrawal Symptoms through Mechanisms Involving Amygdala and Hippocampus Neurotransmission.

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Review 4.  Targeting the immune system in the treatment of bipolar disorder.

Authors:  Joshua D Rosenblat
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Review 5.  Depression and obesity among females, are sex specificities considered?

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7.  NMDA receptor involvement in antidepressant-like effect of pioglitazone in the forced swimming test in mice.

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8.  Adjuvant pioglitazone for unremitted depression: Clinical correlates of treatment response.

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Review 9.  Insulin receptor in the brain: Mechanisms of activation and the role in the CNS pathology and treatment.

Authors:  Igor Pomytkin; João P Costa-Nunes; Vladimir Kasatkin; Ekaterina Veniaminova; Anna Demchenko; Alexey Lyundup; Klaus-Peter Lesch; Eugene D Ponomarev; Tatyana Strekalova
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10.  Cardiometabolic Health in Bipolar Disorder.

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