Literature DB >> 21780776

Remarkable potential of the α-aminophosphonate/phosphinate structural motif in medicinal chemistry.

Artur Mucha1, Paweł Kafarski, Łukasz Berlicki.   

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Year:  2011        PMID： 21780776     DOI： 10.1021/jm200587f

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  52 in total

1.  A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases.

Authors:  Ewelina Węglarz-Tomczak; Łukasz Berlicki; Małgorzata Pawełczak; Bogusław Nocek; Andrzej Joachimiak; Artur Mucha
Journal:  Eur J Med Chem       Date:  2016-04-09       Impact factor: 6.514

2.  New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP).

Authors:  José Luis Viveros-Ceballos; Lizeth A Matías-Valdez; Francisco J Sayago; Carlos Cativiela; Mario Ordóñez
Journal:  Amino Acids       Date:  2021-03-01       Impact factor: 3.520

3.  Redox-neutral α-C-H bond functionalization of secondary amines with concurrent C-P bond formation/N-alkylation.

Authors:  Deepankar Das; Daniel Seidel
Journal:  Org Lett       Date:  2013-08-19       Impact factor: 6.005

4.  Bis(aminomethyl)phosphinic Acid, a Highly Promising Scaffold for the Development of Bacterial Urease Inhibitors.

Authors:  Katarzyna Macegoniuk; Anna Dziełak; Artur Mucha; Łukasz Berlicki
Journal:  ACS Med Chem Lett       Date:  2014-12-11       Impact factor: 4.345

5.  Use of the dehydrophos biosynthetic enzymes to prepare antimicrobial analogs of alaphosphin.

Authors:  Despina J Bougioukou; Chi P Ting; Spencer C Peck; Subha Mukherjee; Wilfred A van der Donk
Journal:  Org Biomol Chem       Date:  2019-01-23       Impact factor: 3.876

6.  Asymmetric homoenolate additions to acyl phosphonates through rational design of a tailored N-heterocyclic carbene catalyst.

Authors:  Ki Po Jang; Gerri E Hutson; Ryne C Johnston; Elizabeth O McCusker; Paul H-Y Cheong; Karl A Scheidt
Journal:  J Am Chem Soc       Date:  2013-12-17       Impact factor: 15.419

7.  An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and molecular modeling.

Authors:  Ewelina Węglarz-Tomczak; Marcin Poręba; Anna Byzia; Łukasz Berlicki; Bogusław Nocek; Rory Mulligan; Andrzej Joachimiak; Marcin Drąg; Artur Mucha
Journal:  Biochimie       Date:  2012-11-03       Impact factor: 4.079

Review 8.  Synthesis of α-Aminophosphonates and Related Derivatives; the Last Decade of the Kabachnik-Fields Reaction.

Authors:  Petra R Varga; György Keglevich
Journal:  Molecules       Date:  2021-04-25       Impact factor: 4.411

9.  Synthesis and Anti-Pancreatic Cancer Activity Studies of Novel 3-Amino-2-hydroxybenzofused 2-Phospha-γ-lactones.

Authors:  Satheesh Krishna Balam; Jayaprakash Soora Harinath; Suresh Kumar Krishnammagari; Raghavendra Reddy Gajjala; Kishore Polireddy; Vijaya Bhaskar Baki; Wei Gu; Koteswara Rao Valasani; Vijaya Kumar Reddy Avula; Swetha Vallela; Grigory Vasilievich Zyryanov; Visweswara Rao Pasupuleti; Suresh Reddy Cirandur
Journal:  ACS Omega       Date:  2021-04-23

10.  Highly Diastereoselective Construction of Carbon- Heteroatom Quaternary Stereogenic Centers in the Synthesis of Analogs of Bioactive Compounds: From Monofluorinated Epoxyalkylphosphonates to α-Fluoro-, β-, or γ-Amino Alcohol Derivatives of Alkylphosphonates.

Authors:  Magdalena Rapp; Klaudia Margas-Musielak; Patrycja Kaczmarek; Agnieszka Witkowska; Tomasz Cytlak; Tomasz Siodła; Henryk Koroniak
Journal:  Front Chem       Date:  2021-06-02       Impact factor: 5.221
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