Literature DB >> 21748297

Topical treatment of cutaneous metastases of malignant melanoma using combined imiquimod and 5-fluorouracil.

Valerie Florin1, Eve Desmedt, Sophie Vercambre-Darras, Laurent Mortier.   

Abstract

BACKGROUND: Despite multiple available options, the treatment of cutaneous melanoma metastases is often unsuccessful. Based on the hypothesis that imiquimod and 5-fluorouracil have synergistic antitumor properties, we used this topical combination to treat several patients. AIM: Our objective was to investigate the treatment combination in a small cohort of patients with surgically non-resectable melanoma metastases.
METHODS: The lesions of 5 patients with multiple cutaneous metastases were treated topically, 5 days per week, with 5-fluorouracil in the morning and imiquimod at night.
RESULTS: 45 lesions were treated. A clinical response was seen in 44 lesions, with a complete response in 19 lesions and a partial response in 25. Stable disease was confirmed in the 1 remaining lesion. No patients developed new lesions during treatment. However, one patient had a recurrence 6 months after treatment discontinuation, followed by a partial response when rechallenged.
CONCLUSIONS: The imiquimod and 5-fluorouracil combination is effective. That patients did not develop new, distant lesions suggests the achievement of locoregional control, probably by the induction of antitumor immune response.

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Year:  2011        PMID: 21748297     DOI: 10.1007/s10637-011-9717-2

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  20 in total

1.  Topical imiquimod treatment of a cutaneous melanoma metastasis.

Authors:  A Steinmann; J O Funk; G Schuler; P von den Driesch
Journal:  J Am Acad Dermatol       Date:  2000-09       Impact factor: 11.527

2.  Imiquimod-induced vitiligo in a patient with genital warts.

Authors:  C Stefanaki; E Nicolaidou; M Hadjivassiliou; C Antoniou; A Katsambas
Journal:  J Eur Acad Dermatol Venereol       Date:  2006-07       Impact factor: 6.166

3.  Small anti-viral compounds activate immune cells via the TLR7 MyD88-dependent signaling pathway.

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Journal:  Nat Immunol       Date:  2002-01-22       Impact factor: 25.606

Review 4.  Interferons as biomodulators of fluoropyrimidines in the treatment of colorectal cancer.

Authors:  D Makower; S Wadler
Journal:  Semin Oncol       Date:  1999-12       Impact factor: 4.929

5.  Death receptor-independent apoptosis in malignant melanoma induced by the small-molecule immune response modifier imiquimod.

Authors:  Michael P Schön; B Gregor Wienrich; Claudia Drewniok; Anne B Bong; Jürgen Eberle; Christoph C Geilen; Harald Gollnick; Margarete Schön
Journal:  J Invest Dermatol       Date:  2004-05       Impact factor: 8.551

6.  Possible mechanisms in the induction of vitiligo-like hypopigmentation by topical imiquimod.

Authors:  J Mashiah; S Brenner
Journal:  Clin Exp Dermatol       Date:  2007-11-02       Impact factor: 3.470

7.  Imiquimod and lentigo maligna: a search for prognostic features in a clinicopathological study with long-term follow-up.

Authors:  A M Powell; A M Robson; R Russell-Jones; R J Barlow
Journal:  Br J Dermatol       Date:  2009-02-16       Impact factor: 9.302

8.  Imiquimod-induced vitiligo after treatment of nodular basal cell carcinoma.

Authors:  Smitha Gowda; Donald K Tillman; James E Fitzpatrick; Anthony A Gaspari; Gary Goldenberg
Journal:  J Cutan Pathol       Date:  2009-08       Impact factor: 1.587

9.  Imiquimod, a topical immune response modifier, in the treatment of cutaneous metastases of malignant melanoma.

Authors:  Anne B Bong; Bernd Bonnekoh; Ingolf Franke; Michael P Schön; Jens Ulrich; Harald Gollnick
Journal:  Dermatology       Date:  2002       Impact factor: 5.366

10.  Modulation of TH1 and TH2 cytokine production with the immune response modifiers, R-848 and imiquimod.

Authors:  T L Wagner; C L Ahonen; A M Couture; S J Gibson; R L Miller; R M Smith; M J Reiter; J P Vasilakos; M A Tomai
Journal:  Cell Immunol       Date:  1999-01-10       Impact factor: 4.868

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  13 in total

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Authors:  Daniel E Spratt; Elizabeth A Gordon Spratt; Shenhong Wu; Antonio DeRosa; Nancy Y Lee; Mario E Lacouture; Christopher A Barker
Journal:  J Clin Oncol       Date:  2014-08-25       Impact factor: 44.544

Review 2.  Current treatment of locoregional recurrence of melanoma.

Authors:  Malcolm Hart Squires; Keith A Delman
Journal:  Curr Oncol Rep       Date:  2013-10       Impact factor: 5.075

3.  Advancements in unresectable melanoma: a multidisciplinary perspective.

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Journal:  Melanoma Manag       Date:  2016-08-16

Review 4.  Melanoma treatment: from conventional to nanotechnology.

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Journal:  J Cancer Res Clin Oncol       Date:  2018-08-09       Impact factor: 4.553

Review 5.  Developments in Intralesional Therapy for Metastatic Melanoma.

Authors:  Sarah Sloot; Omar M Rashid; Arnod A Sarnaik; Jonathan S Zager
Journal:  Cancer Control       Date:  2016-01       Impact factor: 3.302

Review 6.  Intralesional treatment of metastatic melanoma: a review of therapeutic options.

Authors:  Benjamin Weide; Dario Neri; Giuliano Elia
Journal:  Cancer Immunol Immunother       Date:  2017-01-11       Impact factor: 6.968

7.  Imidazoquinoxaline anticancer derivatives and imiquimod interact with tubulin: Characterization of molecular microtubule inhibiting mechanisms in correlation with cytotoxicity.

Authors:  Alexis Courbet; Nicole Bec; Caroline Constant; Christian Larroque; Martine Pugniere; Safia El Messaoudi; Zahraa Zghaib; Sonia Khier; Carine Deleuze-Masquefa; Florence Gattacceca
Journal:  PLoS One       Date:  2017-08-10       Impact factor: 3.240

Review 8.  Trial Watch: Toll-like receptor agonists for cancer therapy.

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9.  Anti-Melanoma immunity and local regression of cutaneous metastases in melanoma patients treated with monobenzone and imiquimod; a phase 2 a trial.

Authors:  Hansje-Eva Teulings; Esther P M Tjin; Karina J Willemsen; Stephanie van der Kleij; Sylvia Ter Meulen; E Helen Kemp; Gabrielle Krebbers; Carel J M van Noesel; Cornelis L M C Franken; Jan W Drijfhout; Cornelis J M Melief; Ludmila Nieuweboer-Krobotova; Omgo E Nieweg; Jos A van der Hage; J P Wietze van der Veen; Germaine N Relyveld; Rosalie M Luiten
Journal:  Oncoimmunology       Date:  2018-01-15       Impact factor: 8.110

10.  Protocol for the TIDAL Melanoma Study: topical imiquimod or diphenylcyclopropenone for the management of cutaneous in-transit melanoma metastases-a phase II, single centre, randomised, pilot study.

Authors:  Tavis Read; Scott Webber; Janine Thomas; Michael Wagels; Helmut Schaider; H Peter Soyer; B Mark Smithers
Journal:  BMJ Open       Date:  2017-10-06       Impact factor: 2.692

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