Literature DB >> 21739958

Synthesis of carbolines by photostimulated cyclization of anilinohalopyridines.

Joydev K Laha1, Silvia M Barolo, Roberto A Rossi, Gregory D Cuny.   

Abstract

A general synthetic route to prepare all four carboline regioisomers by photostimulated cyclization of anilinohalopyridines is described. The methodology affords various substituted carbolines in good to excellent yields. In the case of α-carbolines, the S(RN)1 methodology complements previously reported palladium-catalyzed cyclization approaches.

Entities:  

Mesh:

Substances:

Year:  2011        PMID: 21739958     DOI: 10.1021/jo200923n

Source DB:  PubMed          Journal:  J Org Chem        ISSN: 0022-3263            Impact factor:   4.354


  2 in total

1.  Rh(II)2-catalyzed synthesis of α-, β-, or δ-carbolines from aryl azides.

Authors:  Ashley L Pumphrey; Huijun Dong; Tom G Driver
Journal:  Angew Chem Int Ed Engl       Date:  2012-04-26       Impact factor: 15.336

2.  An intramolecular inverse electron demand Diels-Alder approach to annulated α-carbolines.

Authors:  Zhiyuan Ma; Feng Ni; Grace H C Woo; Sie-Mun Lo; Philip M Roveto; Scott E Schaus; John K Snyder
Journal:  Beilstein J Org Chem       Date:  2012-06-06       Impact factor: 2.883

  2 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.