Literature DB >> 21696296

A phase II trial of panobinostat, a histone deacetylase inhibitor, in the treatment of patients with refractory metastatic renal cell carcinoma.

John D Hainsworth1, Jeffrey R Infante, David R Spigel, Edward R Arrowsmith, Ralph V Boccia, Howard A Burris.   

Abstract

PURPOSE: To evaluate the activity of panobinostat in refractory renal carcinoma. PATIENTS AND METHODS: Patients with advanced clear cell renal carcinoma who had received previous therapy with at least one angiogenesis inhibitor and one mTOR inhibitor were treated with panobinostat 45 mg orally twice a week, and were reevaluated after 8 weeks.
RESULTS: Twenty patients were treated with no objective responses. All patients progressed or stopped treatment prior to the 16-week reevaluation. Panobinostat was generally well-tolerated.
CONCLUSION: Panobinostat had no activity in this group of patients with refractory renal carcinoma. Further development of panobinostat in renal carcinoma is not recommended.

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Year:  2011        PMID: 21696296     DOI: 10.3109/07357907.2011.590568

Source DB:  PubMed          Journal:  Cancer Invest        ISSN: 0735-7907            Impact factor:   2.176


  39 in total

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Journal:  Mol Clin Oncol       Date:  2014-07-15

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9.  Phase I study of the mTOR inhibitor everolimus in combination with the histone deacetylase inhibitor panobinostat in patients with advanced clear cell renal cell carcinoma.

Authors:  Anthony Wood; Saby George; Nabil Adra; Sreenivasulu Chintala; Nur Damayanti; Roberto Pili
Journal:  Invest New Drugs       Date:  2019-10-25       Impact factor: 3.850

10.  A phase 1 trial of the histone deacetylase inhibitor AR-42 in patients with neurofibromatosis type 2-associated tumors and advanced solid malignancies.

Authors:  Katharine A Collier; Hugo Valencia; Herbert Newton; Erinn M Hade; Douglas W Sborov; Robert Cavaliere; Ming Poi; Mitch A Phelps; Sophia G Liva; Christopher C Coss; Jiang Wang; Soun Khountham; Paul Monk; Charles L Shapiro; Richard Piekarz; Craig C Hofmeister; D Bradley Welling; Amir Mortazavi
Journal:  Cancer Chemother Pharmacol       Date:  2021-01-25       Impact factor: 3.333

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