Literature DB >> 21674534

Liquid formulation of pentoxifylline is a poorly tolerated treatment for duchenne dystrophy.

Angela Zimmerman1, Paula R Clemens, Carolina Tesi-Rocha, Anne Connolly, Susan T Iannaccone, Nancy Kuntz, Adrienne Arrieta, Lauren Hache, Erik Henricson, Fengming Hu, Jill Mayhew, Diana M Escolar.   

Abstract

INTRODUCTION: In this study we performed an open-label, pilot study of an orally administered liquid formulation of immediate-release pentoxifylline (PTX) on patients with Duchenne muscular dystrophy (DMD). Treatment efficacy, safety, and tolerability were assessed.
METHODS: The tolerability and safety of PTX and measures of muscle strength and function were evaluated during 12 months of treatment.
RESULTS: Seventeen boys with DMD, between 4 and 8 years of age, were enrolled at one of five Cooperative International Neuromuscular Research Group (CINRG) centers. Only 9 were able to complete the 12-month PTX treatment phase; the primary reason for discontinuation was adverse events. Intolerable gastrointestinal side effects were experienced by 65% of participants. Two participants had severe leukopenia that resolved with medication withdrawal.
CONCLUSIONS: Open-label treatment with a liquid formulation of immediate-release PTX resulted in a high incidence of adverse events in boys with DMD. Poor tolerability of this PTX formulation precluded adequate assessment of efficacy.
Copyright © 2011 Wiley Periodicals, Inc.

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Year:  2011        PMID: 21674534      PMCID: PMC3136640          DOI: 10.1002/mus.22127

Source DB:  PubMed          Journal:  Muscle Nerve        ISSN: 0148-639X            Impact factor:   3.217


  7 in total

1.  Pre-clinical screening of drugs using the mdx mouse.

Authors:  J A Granchelli; C Pollina; M S Hudecki
Journal:  Neuromuscul Disord       Date:  2000-06       Impact factor: 4.296

Review 2.  Effects of phosphodiesterase inhibition on the inflammatory response after shock: role of pentoxifylline.

Authors:  Raul Coimbra; Heidi Melbostad; David B Hoyt
Journal:  J Trauma       Date:  2004-02

3.  Relaxin restores altered ileal spontaneous contractions in dystrophic (mdx) mice.

Authors:  Maria Caterina Baccari; Franco Calamai; Laura Chiappini; Maria Giuliana Vannucchi; Daniele Bani
Journal:  Ann N Y Acad Sci       Date:  2005-05       Impact factor: 5.691

4.  Evolution of gastric electrical features and gastric emptying in children with Duchenne and Becker muscular dystrophy.

Authors:  Osvaldo Borrelli; Gennaro Salvia; Valentina Mancini; Lucio Santoro; Francesca Tagliente; Erminia Francesca Romeo; Salvatore Cucchiara
Journal:  Am J Gastroenterol       Date:  2005-03       Impact factor: 10.864

Review 5.  Immunological mechanisms of pentoxifylline in chronic heart failure.

Authors:  Steven M Shaw; Mohammed K H Shah; Simon G Williams; James E Fildes
Journal:  Eur J Heart Fail       Date:  2009-02       Impact factor: 15.534

6.  Altered tachykinergic influence on gastric mechanical activity in mdx mice.

Authors:  F Mulè; A Amato; M G Vannucchi; M S Faussone-Pellegrini; R Serio
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7.  Reversal by relaxin of altered ileal spontaneous contractions in dystrophic (mdx) mice through a nitric oxide-mediated mechanism.

Authors:  M C Baccari; S Nistri; M G Vannucchi; F Calamai; D Bani
Journal:  Am J Physiol Regul Integr Comp Physiol       Date:  2007-05-23       Impact factor: 3.619

  7 in total
  4 in total

1.  Pentoxifylline as a rescue treatment for DMD: a randomized double-blind clinical trial.

Authors:  D M Escolar; A Zimmerman; T Bertorini; P R Clemens; A M Connolly; L Mesa; K Gorni; A Kornberg; H Kolski; N Kuntz; Y Nevo; C Tesi-Rocha; K Nagaraju; S Rayavarapu; L P Hache; J E Mayhew; J Florence; F Hu; A Arrieta; E Henricson; R T Leshner; J K Mah
Journal:  Neurology       Date:  2012-03-07       Impact factor: 9.910

2.  Selective serotonin reuptake inhibitors ameliorate MEGF10 myopathy.

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3.  Pharmacological therapeutics targeting the secondary defects and downstream pathology of Duchenne muscular dystrophy.

Authors:  Janelle M Spinazzola; Louis M Kunkel
Journal:  Expert Opin Orphan Drugs       Date:  2016-10-18       Impact factor: 0.694

4.  Motor and cognitive assessment of infants and young boys with Duchenne Muscular Dystrophy: results from the Muscular Dystrophy Association DMD Clinical Research Network.

Authors:  Anne M Connolly; Julaine M Florence; Mary M Cradock; Elizabeth C Malkus; Jeanine R Schierbecker; Catherine A Siener; Charlie O Wulf; Pallavi Anand; Paul T Golumbek; Craig M Zaidman; J Philip Miller; Linda P Lowes; Lindsay N Alfano; Laurence Viollet-Callendret; Kevin M Flanigan; Jerry R Mendell; Craig M McDonald; Erica Goude; Linda Johnson; Alina Nicorici; Peter I Karachunski; John W Day; Joline C Dalton; Janey M Farber; Karen K Buser; Basil T Darras; Peter B Kang; Susan O Riley; Elizabeth Shriber; Rebecca Parad; Kate Bushby; Michelle Eagle
Journal:  Neuromuscul Disord       Date:  2013-05-28       Impact factor: 4.296

  4 in total

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