Literature DB >> 21669530

Synthesis and activities of naphthalimide azoles as a new type of antibacterial and antifungal agents.

Yi-Yi Zhang1, Cheng-He Zhou.   

Abstract

Naphthalimide-derived azoles as a new type of antimicrobial agents were synthesized and evaluated for their efficiency in vitro against eight bacteria and two fungi by two fold serial dilution technique. Most title compounds exhibited good antimicrobial potency with low MIC values ranging from 1 to 16μg/mL. Notably, some synthesized compounds displayed comparable or even better antibacterial and antifungal activities against some tested strains than the reference drugs Orbifloxacin, Chloromycin and Fluconazole, respectively.
Copyright © 2011 Elsevier Ltd. All rights reserved.

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Year:  2011        PMID： 21669530     DOI： 10.1016/j.bmcl.2011.05.042

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

1.  Evaluation of DNA Binding, Radicals Scavenging and Antimicrobial Studies of Newly Synthesized N-Substituted Naphthalimides: Spectroscopic and Molecular Docking Investigations.

Authors:  Pattan Sirajuddin Nayab; Madhusudana Pulaganti; Suresh Kumar Chitta; Mohammad Abid; Rahis Uddin
Journal:  J Fluoresc       Date:  2015-10-13       Impact factor: 2.217

Review 2.  An Updated Review on the Synthesis and Antibacterial Activity of Molecular Hybrids and Conjugates Bearing Imidazole Moiety.

Authors:  Renzo Rossi; Maurizio Ciofalo
Journal:  Molecules       Date:  2020-11-04       Impact factor: 4.411

3.  Synthesis and sensor activity of a PET-based 1,8-naphthalimide Probe for Zn(2+) and pH determination.

Authors:  Stefan M Dimov; Nikolai I Georgiev; Abdullah M Asiri; Vladimir B Bojinov
Journal:  J Fluoresc       Date:  2014-09-09       Impact factor: 2.217

4.  6-Bromo-2-(diprop-2-ynyl-amino)-1H-benzo[de]isoquinoline-1,3(2H)-dione.

Authors:  Jing-Song Lv; Jun-Lei Wang; Cheng-He Zhou
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-05-23

5.  Crystal structure of 2-[4-(4-chloro-phen-yl)-1-(4-meth-oxy-phen-yl)-2-oxoazetidin-3-yl]benzo[de]iso-quinoline-1,3-dione dimethyl sulfoxide monosolvate.

Authors:  Ísmail Çelik; Mehmet Akkurt; Aliasghar Jarrahpour; Javad Ameri Rad; Ömer Çelik
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2015-01-28

6.  Synthesis and the Biological Activity of Phosphonylated 1,2,3-Triazolenaphthalimide Conjugates.

Authors:  Iwona E Głowacka; Rafał Gulej; Piotr Grzonkowski; Graciela Andrei; Dominique Schols; Robert Snoeck; Dorota G Piotrowska
Journal:  Molecules       Date:  2016-10-26       Impact factor: 4.411
  6 in total

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