Literature DB >> 21615166

Cu(I)- and Ru(II)-mediated "click" cyclization of tripeptides toward vancomycin-inspired mimics.

Jinqiang Zhang1, Johan Kemmink, Dirk T S Rijkers, Rob M J Liskamp.   

Abstract

Structural mimics comprising 1,4- and 1,5-disubstituted triazole-containing cyclic tripeptides with excellent resemblance toward the DE-ring of vancomycin are conveniently accessible using Cu(I)- or Ru(II)-assisted "click" cyclization.

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Year:  2011        PMID： 21615166     DOI： 10.1021/ol201184b

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  6 in total

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  6 in total

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