Literature DB >> 21492993

Atazanavir in pregnancy: impact on neonatal hyperbilirubinemia.

Laurent Mandelbrot1, Fabienne Mazy, Corinne Floch-Tudal, Françoise Meier, Elie Azria, Catherine Crenn-Hebert, Jean Marc Treluyer, Evelyne Herinomenzanahary, Claudia Ferreira, Gilles Peytavin.   

Abstract

OBJECTIVE: To study the impact on the neonate of maternal antiretroviral therapy with atazanavir (ATV). STUDY
DESIGN: An observational study of 22 HIV-infected women receiving, for clinical indications, antiretroviral therapy with ATV 300 mg and ritonavir 100mg during pregnancy and their 23 HIV infants (including a twin pair).
RESULTS: Mothers had received ATV for a median duration of 19 months [range 3-49] by delivery. At delivery, plasma HIV-RNA was <40 copies/mL in all patients. Liver enzymes were normal in 19/22 patients, but one woman had grade 3-4 liver toxicity. Maternal serum bilirubin concentrations were above the upper limit of normal in most patients, with grade 3 toxicity in 5 patients. All but one woman had trough ATV concentrations during pregnancy above the minimum effective concentration. The median cord blood ATV concentration was 130 ng/mL [range<30-758]; the cord/maternal ratio was 21%. All neonates were born at term [median 38.2 weeks]. Three neonates had mildly elevated AST transaminase levels. Bilirubin concentrations at birth were significantly higher than maternal concentrations, with a median of 44 μm/L [range 24-129]; values on days 2-3 were 63 [8-212]. Five neonates had jaundice requiring phototherapy, without liver damage, and recovered without sequelae.
CONCLUSION: Neonates whose mothers were treated with ATV should be monitored for hyperbilirubinemia, which may be due to placental transfer of unconjugated bilirubin from the mother and/or a direct effect of transplacental ATV on bilirubin metabolism in the fetus.
Copyright © 2011 Elsevier Ireland Ltd. All rights reserved.

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Year:  2011        PMID: 21492993     DOI: 10.1016/j.ejogrb.2011.02.005

Source DB:  PubMed          Journal:  Eur J Obstet Gynecol Reprod Biol        ISSN: 0301-2115            Impact factor:   2.435


  14 in total

1.  Meconium Atazanavir Concentrations and Early Language Outcomes in HIV-Exposed Uninfected Infants With Prenatal Atazanavir Exposure.

Authors:  Sarah K Himes; Yanling Huo; George K Siberry; Paige L Williams; Mabel L Rice; Patricia A Sirois; Toni Frederick; Rohan Hazra; Marilyn A Huestis
Journal:  J Acquir Immune Defic Syndr       Date:  2015-06-01       Impact factor: 3.731

2.  Infant peripheral blood repetitive element hypomethylation associated with antiretroviral therapy in utero.

Authors:  Carmen J Marsit; Sean S Brummel; Deborah Kacanek; George R Seage; Stephen A Spector; David A Armstrong; Barry M Lester; Kenneth Rich
Journal:  Epigenetics       Date:  2015       Impact factor: 4.528

3.  Placental transfer of darunavir in an ex vivo human cotyledon perfusion model.

Authors:  Laurent Mandelbrot; Dominique Duro; Emilie Belissa; Gilles Peytavin
Journal:  Antimicrob Agents Chemother       Date:  2014-06-30       Impact factor: 5.191

4.  Atazanavir exposure in utero and neurodevelopment in infants: a comparative safety study.

Authors:  Ellen C Caniglia; Kunjal Patel; Yanling Huo; Paige L Williams; Suad Kapetanovic; Kenneth C Rich; Patricia A Sirois; Denise L Jacobson; Sonia Hernandez-Diaz; Miguel A Hernán; George R Seage
Journal:  AIDS       Date:  2016-05-15       Impact factor: 4.177

5.  Safety of perinatal exposure to antiretroviral medications: developmental outcomes in infants.

Authors:  Patricia A Sirois; Yanling Huo; Paige L Williams; Kathleen Malee; Patricia A Garvie; Betsy Kammerer; Kenneth Rich; Russell B Van Dyke; Molly L Nozyce
Journal:  Pediatr Infect Dis J       Date:  2013-06       Impact factor: 2.129

Review 6.  HIV protease inhibitors in pregnancy : pharmacology and clinical use.

Authors:  Nisha Andany; Mona R Loutfy
Journal:  Drugs       Date:  2013-03       Impact factor: 9.546

7.  Pharmacokinetics of an increased atazanavir dose with and without tenofovir during the third trimester of pregnancy.

Authors:  Regis Kreitchmann; Brookie M Best; Jiajia Wang; Alice Stek; Edmund Caparelli; D Heather Watts; Elizabeth Smith; David E Shapiro; Steve Rossi; Sandra K Burchett; Elizabeth Hawkins; Mark Byroads; Tim R Cressey; Mark Mirochnick
Journal:  J Acquir Immune Defic Syndr       Date:  2013-05-01       Impact factor: 3.731

8.  Evaluation of risk for late language emergence after in utero antiretroviral drug exposure in HIV-exposed uninfected infants.

Authors:  Mabel L Rice; Bret Zeldow; George K Siberry; Murli Purswani; Kathleen Malee; Howard J Hoffman; Toni Frederick; Ashley Buchanan; Patricia A Sirois; Susannah M Allison; Paige L Williams
Journal:  Pediatr Infect Dis J       Date:  2013-10       Impact factor: 2.129

Review 9.  Protecting the fetus against HIV infection: a systematic review of placental transfer of antiretrovirals.

Authors:  Shelley A McCormack; Brookie M Best
Journal:  Clin Pharmacokinet       Date:  2014-11       Impact factor: 6.447

10.  Clinical and pharmacogenetic factors affecting neonatal bilirubinemia following atazanavir treatment of mothers during pregnancy.

Authors:  Timothy Eley; Shu-Pang Huang; Francesca Conradie; Carmen D Zorrilla; Deirdre Josipovic; Mariëtte Botes; Olayemi Osiyemi; Hélène Hardy; Richard Bertz; Donnie McGrath
Journal:  AIDS Res Hum Retroviruses       Date:  2013-07-19       Impact factor: 2.205

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