Literature DB >> 21431166

Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G.

Eugen Merkul1, Elisabeth Schäfer, Thomas J J Müller.   

Abstract

3-(Hetero)aryl substituted indoles, 7-azaindoles, and pyrroles can be obtained in a very concise fashion via a one-pot Masuda borylation-Suzuki coupling sequence. The concise total syntheses of the marine natural products meridianins A (5) and G (4i) nicely illustrate the utility of this methodology.

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Year:  2011        PMID： 21431166     DOI： 10.1039/c1ob05310h

Source DB:  PubMed          Journal:  Org Biomol Chem        ISSN： 1477-0520            Impact factor:   3.876


  4 in total

1.  Asymmetrically bridged aroyl-S,N-ketene acetal-based multichromophores with aggregation-induced tunable emission.

Authors:  Lukas Biesen; Julius Krenzer; Nithiya Nirmalananthan-Budau; Ute Resch-Genger; Thomas J J Müller
Journal:  Chem Sci       Date:  2022-04-12       Impact factor: 9.969

2.  Transition-metal-free synthesis of pyrimidines from lignin β-O-4 segments via a one-pot multi-component reaction.

Authors:  Bo Zhang; Tenglong Guo; Zhewei Li; Fritz E Kühn; Ming Lei; Zongbao K Zhao; Jianliang Xiao; Jian Zhang; Dezhu Xu; Tao Zhang; Changzhi Li
Journal:  Nat Commun       Date:  2022-06-11       Impact factor: 17.694

3.  Room-temperature borylation and one-pot two-step borylation/Suzuki-Miyaura cross-coupling reaction of aryl chlorides.

Authors:  Hong Ji; Li-Yang Wu; Jiang-Hong Cai; Guo-Rong Li; Na-Na Gan; Zhao-Hua Wang
Journal:  RSC Adv       Date:  2018-04-11       Impact factor: 4.036

4.  Concise Syntheses of Marine (Bis)indole Alkaloids Meridianin C, D, F, and G and Scalaridine A via One-Pot Masuda Borylation-Suzuki Coupling Sequence.

Authors:  Marco Kruppa; Gereon A Sommer; Thomas J J Müller
Journal:  Molecules       Date:  2022-03-30       Impact factor: 4.411
  4 in total

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