Literature DB >> 21387512

Design and synthesis of Selenazole-containing peptides for cocrystallization with P-glycoprotein.

Houchao Tao1, Yue Weng, Rupeng Zhuo, Geoffrey Chang, Ina L Urbatsch, Qinghai Zhang.   

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Year:  2011        PMID： 21387512      PMCID： PMC4814162          DOI： 10.1002/cbic.201100048

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  19 in total

1.  Peptide-embedded heterocycles by mild single and multiple Aza-Wittig ring closures.

Authors:  Matthias Riedrich; Surendra Harkal; Hans-Dieter Arndt
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Review 2.  ABC efflux pump-based resistance to chemotherapy drugs.

Authors:  Paul D W Eckford; Frances J Sharom
Journal:  Chem Rev       Date:  2009-07       Impact factor: 60.622

3.  New cyclic peptides from the ascidian Lissoclinum patella.

Authors:  X Fu; T Do; F J Schmitz; V Andrusevich; M H Engel
Journal:  J Nat Prod       Date:  1998-12       Impact factor: 4.050

4.  Dendroamides, new cyclic hexapeptides from a blue-green alga. Multidrug-resistance reversing activity of dendroamide A.

Authors:  J Ogino; R E Moore; G M Patterson; C D Smith
Journal:  J Nat Prod       Date:  1996-06       Impact factor: 4.050

5.  Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"?

Authors:  Tip W Loo; David M Clarke
Journal:  Biochem Biophys Res Commun       Date:  2005-04-08       Impact factor: 3.575

6.  A biomimetic synthesis of thiazolines using hexaphenyloxodiphosphonium trifluoromethanesulfonate.

Authors:  Shu-Li You; Hossein Razavi; Jeffery W Kelly
Journal:  Angew Chem Int Ed Engl       Date:  2003-01-03       Impact factor: 15.336

Review 7.  Targeting multidrug resistance in cancer.

Authors:  Gergely Szakács; Jill K Paterson; Joseph A Ludwig; Catherine Booth-Genthe; Michael M Gottesman
Journal:  Nat Rev Drug Discov       Date:  2006-03       Impact factor: 84.694

8.  Modeling conformational changes in cyclosporin A.

Authors:  M F O'Donohue; A W Burgess; M D Walkinshaw; H R Treutlein
Journal:  Protein Sci       Date:  1995-10       Impact factor: 6.725

9.  Simultaneous binding of two different drugs in the binding pocket of the human multidrug resistance P-glycoprotein.

Authors:  Tip W Loo; M Claire Bartlett; David M Clarke
Journal:  J Biol Chem       Date:  2003-08-07       Impact factor: 5.157

10.  Cyclosporin A and its analogues as modifiers of adriamycin and vincristine resistance in a multi-drug resistant human lung cancer cell line.

Authors:  P R Twentyman; N E Fox; D J White
Journal:  Br J Cancer       Date:  1987-07       Impact factor: 7.640
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  11 in total

Review 1.  Molecular basis of the polyspecificity of P-glycoprotein (ABCB1): recent biochemical and structural studies.

Authors:  Eduardo E Chufan; Hong-May Sim; Suresh V Ambudkar
Journal:  Adv Cancer Res       Date:  2015-01-08       Impact factor: 6.242

Review 2.  Inhibit or Evade Multidrug Resistance P-Glycoprotein in Cancer Treatment.

Authors:  Deepali Waghray; Qinghai Zhang
Journal:  J Med Chem       Date:  2017-12-28       Impact factor: 7.446

3.  Design, synthesis, and biological evaluation of (S)-valine thiazole-derived cyclic and noncyclic peptidomimetic oligomers as modulators of human P-glycoprotein (ABCB1).

Authors:  Satyakam Singh; Nagarajan Rajendra Prasad; Khyati Kapoor; Eduardo E Chufan; Bhargav A Patel; Suresh V Ambudkar; Tanaji T Talele
Journal:  Chembiochem       Date:  2013-11-29       Impact factor: 3.164

4.  Understanding polyspecificity within the substrate-binding cavity of the human multidrug resistance P-glycoprotein.

Authors:  Lorena Martinez; Ophélie Arnaud; Emilie Henin; Houchao Tao; Vincent Chaptal; Rupak Doshi; Thibault Andrieu; Sébastien Dussurgey; Michel Tod; Attilio Di Pietro; Qinghai Zhang; Geoffrey Chang; Pierre Falson
Journal:  FEBS J       Date:  2014-01-17       Impact factor: 5.542

5.  Localization and substrate selectivity of sea urchin multidrug (MDR) efflux transporters.

Authors:  Tufan Gökirmak; Joseph P Campanale; Lauren E Shipp; Gary W Moy; Houchao Tao; Amro Hamdoun
Journal:  J Biol Chem       Date:  2012-11-02       Impact factor: 5.157

6.  Mass spectrometry reveals synergistic effects of nucleotides, lipids, and drugs binding to a multidrug resistance efflux pump.

Authors:  Julien Marcoux; Sheila C Wang; Argyris Politis; Eamonn Reading; Jerome Ma; Philip C Biggin; Min Zhou; Houchao Tao; Qinghai Zhang; Geoffrey Chang; Nina Morgner; Carol V Robinson
Journal:  Proc Natl Acad Sci U S A       Date:  2013-05-20       Impact factor: 11.205

7.  Snapshots of ligand entry, malleable binding and induced helical movement in P-glycoprotein.

Authors:  Paul Szewczyk; Houchao Tao; Aaron P McGrath; Mark Villaluz; Steven D Rees; Sung Chang Lee; Rupak Doshi; Ina L Urbatsch; Qinghai Zhang; Geoffrey Chang
Journal:  Acta Crystallogr D Biol Crystallogr       Date:  2015-02-26

8.  Multiple transport-active binding sites are available for a single substrate on human P-glycoprotein (ABCB1).

Authors:  Eduardo E Chufan; Khyati Kapoor; Hong-May Sim; Satyakam Singh; Tanaji T Talele; Stewart R Durell; Suresh V Ambudkar
Journal:  PLoS One       Date:  2013-12-05       Impact factor: 3.240

9.  Design and synthesis of human ABCB1 (P-glycoprotein) inhibitors by peptide coupling of diverse chemical scaffolds on carboxyl and amino termini of (S)-valine-derived thiazole amino acid.

Authors:  Satyakam Singh; Nagarajan Rajendra Prasad; Eduardo E Chufan; Bhargav A Patel; Yi-Jun Wang; Zhe-Sheng Chen; Suresh V Ambudkar; Tanaji T Talele
Journal:  J Med Chem       Date:  2014-05-07       Impact factor: 7.446

10.  An enzymatic route to selenazolines.

Authors:  Jesko Koehnke; Falk Morawitz; Andrew F Bent; Wael E Houssen; Sally L Shirran; Matthew A Fuszard; Iain A Smellie; Catherine H Botting; Margaret C M Smith; Marcel Jaspars; James H Naismith
Journal:  Chembiochem       Date:  2013-02-18       Impact factor: 3.164
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